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Results: 1-13 |
Results: 13

Authors: FASSLER A BOLD G STEINER H
Citation: A. Fassler et al., A CONCISE SYNTHESIS OF AZA-DIPEPTIDE ISOSTERES, Tetrahedron letters, 39(27), 1998, pp. 4925-4928

Authors: BOLD G FASSLER A CAPRARO HG COZENS R KLIMKAIT T LAZDINS J MESTAN J PONCIONI B ROSEL J STOVER D TINTELNOTBLOMLEY M ACEMOGLU F BECK W BOSS E ESCHBACH M HURLIMANN T MASSO E ROUSSEL S UCCISTOLL K WYSS D LANG R
Citation: G. Bold et al., NEW AZA-DIPEPTIDE ANALOGS AS POTENT AND ORALLY ABSORBED HIV-1 PROTEASE INHIBITORS - CANDIDATES FOR CLINICAL DEVELOPMENT, Journal of medicinal chemistry, 41(18), 1998, pp. 3387-3401

Authors: TRAXLER P BOLD G FREI J LANG M LYDON N METT H BUCHDUNGER E MEYER T MUELLER M FURET P
Citation: P. Traxler et al., USE OF A PHARMACOPHORE MODEL FOR THE DESIGN OF EGF-R TYROSINE KINASE INHIBITORS - 4-(PHENYLAMINO)PYRAZOLO[3,4-D]PYRIMIDINES, Journal of medicinal chemistry, 40(22), 1997, pp. 3601-3616

Authors: LAZDINS JK MESTAN J GOUTTE G WALKER MR BOLD G CAPRARO HG KLIMKAIT T
Citation: Jk. Lazdins et al., IN-VITRO EFFECT OF ALPHA(1)-ACID GLYCOPROTEIN ON THE ANTI-HUMAN-IMMUNODEFICIENCY-VIRUS (HIV) ACTIVITY OF THE PROTEASE INHIBITOR CGP-61755 -A COMPARATIVE-STUDY WITH OTHER RELEVANT HIV PROTEASE INHIBITORS, The Journal of infectious diseases, 175(5), 1997, pp. 1063-1070

Authors: SOLLADIECAVALLO A ROCHE D BOLD G ACEMOGLU F TINTELNOTBLOMLEY M FISCHER J DECIAN A
Citation: A. Solladiecavallo et al., STEREOSELECTIVE SYNTHESIS OF (4S,5R,6S)-4-(5,6-EPOXY-6-PHENYL)-GAMMA-LACTONE, Tetrahedron : asymmetry, 7(6), 1996, pp. 1797-1810

Authors: COZENS RM BOLD G CAPRARO HG FASSLER A MESTAN J LANG M PONCIONI B STOVER D ROSEL JL
Citation: Rm. Cozens et al., SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF CGP-57813 AND CGP-61755, HIV-1 PROTEASE INHIBITORS FROM THE PHE-C-PHE PEPTIDOMIMETIC CLASS, Antiviral chemistry & chemotherapy, 7(6), 1996, pp. 294-299

Authors: CAPRARO HG BOLD G FASSLER A COZENS R KLIMKAIT T LAZDINS J PONCIONI B ROSEL JL STOVER D LANG M
Citation: Hg. Capraro et al., SYNTHESIS OF POTENT AND ORALLY-ACTIVE HIV-PROTEASE INHIBITORS, Archiv der pharmazie, 329(6), 1996, pp. 273-278

Authors: LAZDINS JK BOLD G CAPRARO HG COZENS R FASSLER A FLESCH G KLIMKAIT T LANG M MESTAN J PONCIONI B ROSEL J STOVER D TINTELNOTBLOMLEY M WALKER MR WOODSCOOK K
Citation: Jk. Lazdins et al., PROFILE OF CGP-61755 - A NOVEL AND POTENT HIV-1 PROTEASE INHIBITOR THAT SHOWS ENHANCED ANTI-HIV ACTIVITY WHEN COMBINED WITH OTHER ANTIRETROVIRAL AGENTS IN-VITRO, Schweizerische medizinische Wochenschrift, 126(43), 1996, pp. 1849-1851

Authors: FASSLER A BOLD G CAPRARO HG COZENS R MESTAN J PONCIONI B ROSEL J TINTELNOTBLOMLEY M LANG M
Citation: A. Fassler et al., AZA-PEPTIDE ANALOGS AS POTENT HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 PROTEASE INHIBITORS WITH ORAL BIOAVAILABILITY, Journal of medicinal chemistry, 39(16), 1996, pp. 3203-3216

Authors: DUTHALER RO HAFNER A ALSTERS PL BOLD G RIHS G ROTHESTREIT P WYSS B
Citation: Ro. Duthaler et al., THE PREPARATION OF CHIRAL TITANIUM REAGENTS - A COMPARISON OF NEW ANDKNOWN LIGANDS, Inorganica Chimica Acta, 222(1-2), 1994, pp. 95-113

Authors: FASSLER A ROSEL J GRUTTER M TINTELNOTBLOMLEY M ALTERI E BOLD G LANG M
Citation: A. Fassler et al., NOVEL PSEUDOSYMMETRIC INHIBITORS OF HIV-1 PROTEASE, Bioorganic & medicinal chemistry letters, 3(12), 1993, pp. 2837-2842

Authors: ALTERI E BOLD G COZENS R FAESSLER A KLIMKAIT T LANG M LAZDINS J PONCIONI B ROESEL JL SCHNEIDER P WALKER M WOODSCOOK K
Citation: E. Alteri et al., CGP-53437, AN ORALLY BIOAVAILABLE INHIBITOR OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 PROTEASE WITH POTENT ANTIVIRAL ACTIVITY, Antimicrobial agents and chemotherapy, 37(10), 1993, pp. 2087-2092

Authors: DEREPPE C BOLD G GHISALBA O EBERT E SCHAR HP
Citation: C. Dereppe et al., PURIFICATION AND CHARACTERIZATION OF DIHYDRODIPICOLINATE SYNTHASE FROM PEA, Plant physiology, 98(3), 1992, pp. 813-821
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