AAAAAA

   
Results: 1-12 |
Results: 12
PEPTIDE ALDEHYDE INHIBITORS OF CATHEPSIN-K INHIBIT BONE-RESORPTION BOTH IN-VITRO AND IN-VIVO
Authors: VOTTA BJ LEVY MA BADGER A BRADBEER J DODDS RA JAMES IE THOMPSON S BOSSARD MJ CARR T CONNOR JR TOMASZEK TA SZEWCZUK L DRAKE FH VEBER DF GOWEN M
Citation: Bj. Votta et al., PEPTIDE ALDEHYDE INHIBITORS OF CATHEPSIN-K INHIBIT BONE-RESORPTION BOTH IN-VITRO AND IN-VIVO, Journal of bone and mineral research, 12(9), 1997, pp. 1396-1406
DESIGN OF POTENT AND SELECTIVE HUMAN CATHEPSIN-K INHIBITORS THAT SPANTHE ACTIVE-SITE
Authors: THOMPSON SK HALBERT SM BOSSARD MJ TOMASZEK TA LEVY MA ZHAO BG SMITH WW ABDELMEGUID SS JANSON CA DALESSIO KJ MCQUENEY MS AMEGADZIE BY HANNING CR DESJARLAIS RL BRIAND J SARKAR SK HUDDLESTON MJ IJAMES CF CARR SA GARNES KT SHU A HEYS JR BRADBEER J ZEMBRYKI D LEERYKACZEWSKI L JAMES IE LARK MW DRAKE FH GOWEN M GLEASON JG VEBER DF
Citation: Sk. Thompson et al., DESIGN OF POTENT AND SELECTIVE HUMAN CATHEPSIN-K INHIBITORS THAT SPANTHE ACTIVE-SITE, Proceedings of the National Academy of Sciences of the United Statesof America, 94(26), 1997, pp. 14249-14254
STRUCTURE AND DESIGN OF POTENT AND SELECTIVE CATHEPSIN-K INHIBITORS
Authors: YAMASHITA DS SMITH WW ZHAO BG JANSON CA TOMASZEK TA BOSSARD MJ LEVY MA OH HJ CARR TJ THOMPSON SK IJAMES CF CARR SA MCQUENEY M DALESSIO KJ AMEGADZIE BY HANNING CR ABDELMEGUID S DESJARLAIS RL GLEASON JG VEBER DF
Citation: Ds. Yamashita et al., STRUCTURE AND DESIGN OF POTENT AND SELECTIVE CATHEPSIN-K INHIBITORS, Journal of the American Chemical Society, 119(46), 1997, pp. 11351-11352
PEPTIDE ALDEHYDE INHIBITORS OF CATHEPSIN-K INHIBIT BONE-RESORPTION BOTH IN-VITRO AND IN-VIVO
Authors: DRAKE F VOTTA BJ BADGER A DODDS RA JAMES I LEVY MA THOMPSON S BOSSARD MJ CARR T CONNOR JR TOMASZEK TA SZEWCZUK L VEBER D GOWEN M
Citation: F. Drake et al., PEPTIDE ALDEHYDE INHIBITORS OF CATHEPSIN-K INHIBIT BONE-RESORPTION BOTH IN-VITRO AND IN-VIVO, Journal of bone and mineral research, 11, 1996, pp. 246-246
PROTEOLYTIC ACTIVITY OF HUMAN OSTEOCLAST CATHEPSIN-K - EXPRESSION, PURIFICATION, ACTIVATION, AND SUBSTRATE IDENTIFICATION
Authors: BOSSARD MJ TOMASZEK TA THOMPSON SK AMEGADZIE BY HANNING CR JONES C KURDYLA JT MCNULTY DE DRAKE FH GOWEN M LEVY MA
Citation: Mj. Bossard et al., PROTEOLYTIC ACTIVITY OF HUMAN OSTEOCLAST CATHEPSIN-K - EXPRESSION, PURIFICATION, ACTIVATION, AND SUBSTRATE IDENTIFICATION, The Journal of biological chemistry, 271(21), 1996, pp. 12517-12524
STRUCTURE-ACTIVITY STUDIES OF RAPAMYCIN ANALOGS - EVIDENCE THAT THE C-7 METHOXY GROUP IS PART OF THE EFFECTOR DOMAIN AND POSITIONED AT THE FKBP12-FRAP INTERFACE
Authors: LUENGO JI YAMASHITA DS DUNNINGTON D BECK AK ROZAMUS LW YEN HK BOSSARD MJ LEVY MA HAND A NEWMANTARR T BADGER A FAUCETTE L JOHNSON RK DALESSIO K PORTER T SHU AYL HEYS R CHOI JW KONGSAEREE P CLARDY J HOLT DA
Citation: Ji. Luengo et al., STRUCTURE-ACTIVITY STUDIES OF RAPAMYCIN ANALOGS - EVIDENCE THAT THE C-7 METHOXY GROUP IS PART OF THE EFFECTOR DOMAIN AND POSITIONED AT THE FKBP12-FRAP INTERFACE, Chemistry & biology, 2(7), 1995, pp. 471-481
STRUCTURE-ACTIVITY STUDIES OF SYNTHETIC FKBP LIGANDS AS PEPTIDYL-PROLYL ISOMERASE INHIBITORS
Authors: HOLT DA KONIALIANBECK AL OH HJ YEN HK ROZAMUS LW KROG AJ ERHARD KF ORTIZ E LEVY MA BRANDT M BOSSARD MJ LUENGO JI
Citation: Da. Holt et al., STRUCTURE-ACTIVITY STUDIES OF SYNTHETIC FKBP LIGANDS AS PEPTIDYL-PROLYL ISOMERASE INHIBITORS, Bioorganic & medicinal chemistry letters, 4(2), 1994, pp. 315-320
DESIGN, SYNTHESIS AND EVALUATION OF DUAL DOMAIN FKBP LIGANDS
Authors: YAMASHITA DS OH HJ YEN HK BOSSARD MJ BRANDT M LEVY MA NEWMANTARR T BADGER A LUENGO JI HOLT DA
Citation: Ds. Yamashita et al., DESIGN, SYNTHESIS AND EVALUATION OF DUAL DOMAIN FKBP LIGANDS, Bioorganic & medicinal chemistry letters, 4(2), 1994, pp. 325-328
CATALYTIC AND LIGAND-BINDING PROPERTIES OF THE FK506 BINDING-PROTEIN FKBP12 - EFFECTS OF THE SINGLE AMINO-ACID SUBSTITUTION OF TYR(82) TO LEU
Authors: BOSSARD MJ BERGSMA DJ BRANDT M LIVI GP ENG WK JOHNSON RK LEVY MA
Citation: Mj. Bossard et al., CATALYTIC AND LIGAND-BINDING PROPERTIES OF THE FK506 BINDING-PROTEIN FKBP12 - EFFECTS OF THE SINGLE AMINO-ACID SUBSTITUTION OF TYR(82) TO LEU, Biochemical journal, 297, 1994, pp. 365-372
STRUCTURE-ACTIVITY STUDIES OF NONMACROCYCLIC RAPAMYCIN DERIVATIVES
Authors: HOLT DA KONIALIAN AL BRANDT M LEVY MA BOSSARD MJ LUENGO JI NEWMANTARR T BADGER A
Citation: Da. Holt et al., STRUCTURE-ACTIVITY STUDIES OF NONMACROCYCLIC RAPAMYCIN DERIVATIVES, Bioorganic & medicinal chemistry letters, 3(10), 1993, pp. 1977-1980
THE TYROSINE89 RESIDUE OF YEAST FKBP12 IS REQUIRED FOR RAPAMYCIN BINDING
Authors: KOSER PL ENG WK BOSSARD MJ MCLAUGHLIN MM CAFFERKEY R SATHE GM FAUCETTE L LEVY MA JOHNSON RK BERGSMA DJ LIVI GP
Citation: Pl. Koser et al., THE TYROSINE89 RESIDUE OF YEAST FKBP12 IS REQUIRED FOR RAPAMYCIN BINDING, Gene, 129(2), 1993, pp. 159-165
DESIGN, SYNTHESIS, AND KINETIC EVALUATION OF HIGH-AFFINITY FKBP LIGANDS AND THE X-RAY CRYSTAL-STRUCTURES OF THEIR COMPLEXES WITH FKBP12
Authors: HOLT DA LUENGO JI YAMASHITA DS OH HJ KONIALIAN AL YEN HK ROZAMUS LW BRANDT M BOSSARD MJ LEVY MA EGGLESTON DS LIANG J SCHULTZ LW STOUT TJ CLARDY J
Citation: Da. Holt et al., DESIGN, SYNTHESIS, AND KINETIC EVALUATION OF HIGH-AFFINITY FKBP LIGANDS AND THE X-RAY CRYSTAL-STRUCTURES OF THEIR COMPLEXES WITH FKBP12, Journal of the American Chemical Society, 115(22), 1993, pp. 9925-9938
Risultati: 1-12 |