Authors:
SALL DJ
BASTIAN JA
BRIGGS SL
BUBEN JA
CHIRGADZE NY
CLAWSON DK
DENNEY ML
GIERA DD
GIFFORDMOORE DS
HARPER RW
HAUSER KL
KLIMKOWSKI VJ
KOHN TJ
LIN HS
MCCOWAN JR
PALKOWITZ AD
SMITH GF
TAKEUCHI K
THRASHER KJ
TINSLEY JM
UTTERBACK BG
YAN SCB
ZHANG MS
Citation: Dj. Sall et al., DIBASIC BENZO[B]THIOPHENE DERIVATIVES AS A NOVEL CLASS OF ACTIVE-SITE-DIRECTED THROMBIN INHIBITORS .1. DETERMINATION OF THE SERINE-PROTEASESELECTIVITY, STRUCTURE-ACTIVITY-RELATIONSHIPS, AND BINDING ORIENTATION, Journal of medicinal chemistry, 40(22), 1997, pp. 3489-3493
Authors:
RAFFA RB
HASLEGO ML
MARYANOFF CA
VILLANI FJ
CODD EE
CONNELLY CD
MARTINEZ RP
SCHUPSKY JJ
BUBEN JA
WU WN
TAKACS AN
MCKOWN LA
Citation: Rb. Raffa et al., UNEXPECTED ANTINOCICEPTIVE EFFECT OF THE N-OXIDE (RWJ-38705) OF TRAMADOL HYDROCHLORIDE, The Journal of pharmacology and experimental therapeutics, 278(3), 1996, pp. 1098-1104
Authors:
CRANE HM
MENALDINO DS
JAGDMANN GE
DARGES JW
BUBEN JA
Citation: Hm. Crane et al., INCREASING THE CELLULAR PKC INHIBITORY ACTIVITY OF BALANOL - A STUDY OF ESTER ANALOGS, Bioorganic & medicinal chemistry letters, 5(18), 1995, pp. 2133-2138
Authors:
JAGDMANN GE
DEFAUW JM
LAI YS
CRANE HM
HALL SE
BUBEN JA
HU H
GOSNELL PA
Citation: Ge. Jagdmann et al., NOVEL PKC INHIBITORY ANALOGS OF BALANOL WITH REPLACEMENT OF THE ESTERFUNCTIONALITY, Bioorganic & medicinal chemistry letters, 5(17), 1995, pp. 2015-2020