AAAAAA

   
Results: 1-12 |
Results: 12
A convenient synthesis of N-Fmoc-N,N '-bis-Boc-7-guanyl-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (Fmoc-N,N '-bis-Boc-7-guanyl-Tic-OH, GTIC)
Authors: Santagada, V Fiorino, F Severino, B Salvadori, S Lazarus, LH Bryant, SD Caliendo, G
Citation: V. Santagada et al., A convenient synthesis of N-Fmoc-N,N '-bis-Boc-7-guanyl-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (Fmoc-N,N '-bis-Boc-7-guanyl-Tic-OH, GTIC), TETRAHEDR L, 42(20), 2001, pp. 3507-3509
Inhibition of human multidrug resistance P-glycoprotein 1 by analogues of a potent delta-opioid antagonist
Authors: Lovekamp, T Cooper, PS Hardison, J Bryant, SD Guerrini, R Balboni, G Salvadori, S Lazarus, LH
Citation: T. Lovekamp et al., Inhibition of human multidrug resistance P-glycoprotein 1 by analogues of a potent delta-opioid antagonist, BRAIN RES, 902(1), 2001, pp. 131-134
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues
Authors: Santagada, V Balboni, G Caliendo, G Guerrini, R Salvadori, S Bianchi, C Bryant, SD Lazarus, LH
Citation: V. Santagada et al., Assessment of substitution in the second pharmacophore of Dmt-Tic analogues, BIOORG MED, 10(24), 2000, pp. 2745-2748
Characterization of N,N(Me)(2)-Dmt-Tic-OH, a delta selective opioid dipeptide antagonist
Authors: Monory, K Bryant, SD Kertesz, I Balboni, G Guerrini, R Toth, G Salvadori, S Lazarus, LH Borsodi, A
Citation: K. Monory et al., Characterization of N,N(Me)(2)-Dmt-Tic-OH, a delta selective opioid dipeptide antagonist, NEUROREPORT, 11(10), 2000, pp. 2083-2086
Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei
Authors: Balboni, G Salvadori, S Guerrini, R Bianchi, C Santagada, V Calliendo, G Bryant, SD Lazarus, LH
Citation: G. Balboni et al., Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei, PEPTIDES, 21(11), 2000, pp. 1663-1671
Inverse agonism by Dmt-Tic analogues and H5 378, a naltrindole analogue
Authors: Labarre, M Butterworth, J St-Onge, S Payza, K Schmidhammer, H Salvadori, S Balboni, G Guerrini, R Bryant, SD Lazarus, LH
Citation: M. Labarre et al., Inverse agonism by Dmt-Tic analogues and H5 378, a naltrindole analogue, EUR J PHARM, 406(1), 2000, pp. R1-R3
Synthesis of stereoisomeric analogues of endomorphin-2, H-Tyr-Pro-Phe-Phe-NH2, and examination of their opioid receptor binding activities and solution conformation
Authors: Okada, Y Fukumizu, A Takahashi, M Shimizu, Y Tsuda, Y Yokoi, T Bryant, SD Lazarus, LH
Citation: Y. Okada et al., Synthesis of stereoisomeric analogues of endomorphin-2, H-Tyr-Pro-Phe-Phe-NH2, and examination of their opioid receptor binding activities and solution conformation, BIOC BIOP R, 276(1), 2000, pp. 7-11
Acylcarnitine analogues as topical, microbicidal spermicides.
Authors: Savle, PS Doncel, GF Bryant, SD Hubieki, MP Robinette, RG Gandour, RD
Citation: Ps. Savle et al., Acylcarnitine analogues as topical, microbicidal spermicides., BIOORG MED, 9(17), 1999, pp. 2545-2548
What peptides these deltorphins be
Authors: Lazarus, LH Bryant, SD Cooper, PS Salvadori, S
Citation: Lh. Lazarus et al., What peptides these deltorphins be, PROG NEUROB, 57(4), 1999, pp. 377-420
Amino acids and peptides. LVI. Synthesis of pyrazinone ring-containing opioid mimetics and examination of their opioid receptor binding activity
Authors: Okada, Y Fukumizu, A Takahashi, M Yamazaki, J Yokoi, T Tsuda, Y Bryant, SD Lazarus, LH
Citation: Y. Okada et al., Amino acids and peptides. LVI. Synthesis of pyrazinone ring-containing opioid mimetics and examination of their opioid receptor binding activity, TETRAHEDRON, 55(50), 1999, pp. 14391-14406
Further studies on the Dmt-Tic pharmacophore: Hydrophobic substituents at the C-terminus endow delta antagonists to manifest mu agonism or mu antagonism
Authors: Salvadori, S Guerrini, R Balboni, G Bianchi, C Bryant, SD Cooper, PS Lazarus, LH
Citation: S. Salvadori et al., Further studies on the Dmt-Tic pharmacophore: Hydrophobic substituents at the C-terminus endow delta antagonists to manifest mu agonism or mu antagonism, J MED CHEM, 42(24), 1999, pp. 5010-5019
Synthesis of pyrazinone ring-containing opioid mimetics and examination oftheir opioid receptor-binding activity
Authors: Okada, Y Fukumizu, A Takahashi, M Yokoi, T Tsuda, Y Bryant, SD Lazarus, LH
Citation: Y. Okada et al., Synthesis of pyrazinone ring-containing opioid mimetics and examination oftheir opioid receptor-binding activity, CHEM PHARM, 47(8), 1999, pp. 1193-1195
Risultati: 1-12 |