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Results: 1-21 |
Results: 21
Non-nucleoside reverse transcriptase inhibitors: perspectives on novel therapeutic compounds and strategies for the treatment of HIV infection
Authors: Buckheit, RW
Citation: Rw. Buckheit, Non-nucleoside reverse transcriptase inhibitors: perspectives on novel therapeutic compounds and strategies for the treatment of HIV infection, EXPERT OP I, 10(8), 2001, pp. 1423-1442
Synthesis and anti-HIV activity of cosalane analogues incorporating two dichlorodisalicylmethane pharmacophore fragments
Authors: Casimiro-Garcia, A De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Fanwick, PE Cushman, M
Citation: A. Casimiro-garcia et al., Synthesis and anti-HIV activity of cosalane analogues incorporating two dichlorodisalicylmethane pharmacophore fragments, BIO MED CH, 9(11), 2001, pp. 2827-2841
SJ-3366, a unique and highly potent nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1 (HIV-1) that also inhibits HIV-2
Authors: Buckheit, RW Watson, K Fliakas-Boltz, V Russell, J Loftus, TL Osterling, MC Turpin, JA Pallansch, LA White, EL Lee, JW Lee, SH Oh, JW Kwon, HS Chung, SG Cho, EH
Citation: Rw. Buckheit et al., SJ-3366, a unique and highly potent nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1 (HIV-1) that also inhibits HIV-2, ANTIM AG CH, 45(2), 2001, pp. 393-400
Synthesis and anti-HIV activity of a bile acid analog of cosalane
Authors: Kannan, A De Clercq, E Pannecouque, C Witvrouw, M Hartman, TL Turpin, JA Buckheit, RW Cushman, M
Citation: A. Kannan et al., Synthesis and anti-HIV activity of a bile acid analog of cosalane, TETRAHEDRON, 57(46), 2001, pp. 9385-9391
Solid-phase synthesis of the alkenyldiarylmethane (ADAM) series of non-nucleoside HIV-1 reverse transcriptase inhibitors
Authors: Xu, GZ Loftus, TL Wargo, H Turpin, JA Buckheit, RW Cushman, M
Citation: Gz. Xu et al., Solid-phase synthesis of the alkenyldiarylmethane (ADAM) series of non-nucleoside HIV-1 reverse transcriptase inhibitors, J ORG CHEM, 66(18), 2001, pp. 5958-5964
Correlation of anti-HIV activity with anion spacing in a series of cosalane analogues with extended polycarboxylate pharmacophores
Authors: Santhosh, KC Paul, GC De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Kc. Santhosh et al., Correlation of anti-HIV activity with anion spacing in a series of cosalane analogues with extended polycarboxylate pharmacophores, J MED CHEM, 44(5), 2001, pp. 703-714
The biological effects of structural variation at the meta position of thearomatic rings and at the end of the alkenyl chain in the alkenyldiarylmethane series of non-nucleoside reverse transcriptase inhibitors
Authors: Xu, GZ Micklatcher, M Silvestri, MA Hartman, TL Burrier, J Osterling, MC Wargo, H Turpin, JA Buckheit, RW Cushman, M
Citation: Gz. Xu et al., The biological effects of structural variation at the meta position of thearomatic rings and at the end of the alkenyl chain in the alkenyldiarylmethane series of non-nucleoside reverse transcriptase inhibitors, J MED CHEM, 44(24), 2001, pp. 4092-4113
Synthesis and anti-HIV activity of cosalane analogues incorporating nitrogen in the linker chain
Authors: Casimiro-Garcia, A De Clercq, E Pannecouque, C Witvrouw, M Stup, TL Turpin, JA Buckheit, RW Cushman, M
Citation: A. Casimiro-garcia et al., Synthesis and anti-HIV activity of cosalane analogues incorporating nitrogen in the linker chain, BIO MED CH, 8(1), 2000, pp. 191-200
Anti-HIV activity of a series of cosalane amino acid conjugates
Authors: Santhosh, KC De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Kc. Santhosh et al., Anti-HIV activity of a series of cosalane amino acid conjugates, BIOORG MED, 10(22), 2000, pp. 2505-2508
Identification of optimal anion spacing for anti-HIV activity in a series of cosalane tetracarboxylates
Authors: Paul, GC De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Gc. Paul et al., Identification of optimal anion spacing for anti-HIV activity in a series of cosalane tetracarboxylates, BIOORG MED, 10(18), 2000, pp. 2149-2152
Anti-HIV-1 activity of calanolides used in combination with other mechanistically diverse inhibitors of HIV-1 replication
Authors: Buckheit, RW Russell, JD Xu, ZQ Flavin, M
Citation: Rw. Buckheit et al., Anti-HIV-1 activity of calanolides used in combination with other mechanistically diverse inhibitors of HIV-1 replication, ANTIVIR CHE, 11(5), 2000, pp. 321-327
Plant-derived and semi-synthetic calanolide compounds with in vitro activity against both human immunodeficiency virus type 1 and human cytomegalovirus
Authors: Xu, ZQ Kern, ER Westbrook, L Allen, LB Buckheit, RW Tseng, CKH Jenta, T Flavin, MT
Citation: Zq. Xu et al., Plant-derived and semi-synthetic calanolide compounds with in vitro activity against both human immunodeficiency virus type 1 and human cytomegalovirus, ANTIVIR CHE, 11(1), 2000, pp. 23-29
Antiviral activity of 2 '-deoxy-3 '-oxa-4 '-thiocytidine (BCH-10652) against lamivudine-resistant human immunodeficiency virus type 1 in SCID-hu Thy/Liv mice
Authors: Stoddart, CA Moreno, ME Linquist-Stepps, VD Bare, C Bogan, MR Gobbi, A Buckheit, RW Bedard, J Rando, RF McCune, JM
Citation: Ca. Stoddart et al., Antiviral activity of 2 '-deoxy-3 '-oxa-4 '-thiocytidine (BCH-10652) against lamivudine-resistant human immunodeficiency virus type 1 in SCID-hu Thy/Liv mice, ANTIM AG CH, 44(3), 2000, pp. 783-786
Discovery of novel HIV-1 reverse transcriptase inhibitors using a combination of 3D database searching and 3D QSAR
Authors: Zaharevitz, DW Gussio, R Wiegand, A Jalluri, R Pattabiraman, N Kellogg, GE Pallansch, LA Yang, SS Buckheit, RW
Citation: Dw. Zaharevitz et al., Discovery of novel HIV-1 reverse transcriptase inhibitors using a combination of 3D database searching and 3D QSAR, MED CHEM RE, 9(7-8), 1999, pp. 551-564
Anti-human immunodeficiency virus type 1 (HIV-1) activity of 2 '-fluoro-2 ',3 '-dideoxyarabinosyladenine (F-ddA) used in combination with other mechanistically diverse inhibitors of HIV-1 replication
Authors: Buckheit, RW Russell, JD Pallansch, LA Driscoll, JS
Citation: Rw. Buckheit et al., Anti-human immunodeficiency virus type 1 (HIV-1) activity of 2 '-fluoro-2 ',3 '-dideoxyarabinosyladenine (F-ddA) used in combination with other mechanistically diverse inhibitors of HIV-1 replication, ANTIVIR CHE, 10(3), 1999, pp. 115-119
PMTI, a broadly active unusual single-stranded polyribonucleotide, inhibits human immunodeficiency virus replication by multiple mechanisms
Authors: Buckheit, RW Lackman-Smith, C Snow, MJ Halliday, SM White, EL Ross, LJ Agrawal, VK Broom, AD
Citation: Rw. Buckheit et al., PMTI, a broadly active unusual single-stranded polyribonucleotide, inhibits human immunodeficiency virus replication by multiple mechanisms, ANTIVIR CHE, 10(1), 1999, pp. 23-32
Unique anti-human immunodeficiency virus activities of the nonnucleoside reverse transcriptase inhibitors calanolide A, costatolide, and dihydrocostatolide
Authors: Buckheit, RW White, EL Fliakas-Boltz, V Russell, J Stup, TL Kinjerski, TL Osterling, MC Weigand, A Bader, JP
Citation: Rw. Buckheit et al., Unique anti-human immunodeficiency virus activities of the nonnucleoside reverse transcriptase inhibitors calanolide A, costatolide, and dihydrocostatolide, ANTIM AG CH, 43(8), 1999, pp. 1827-1834
Synthesis and anti-HIV activity of cosalane analogues with substituted benzoic acid rings attached to the pharmacophore through methylene and amide linkers
Authors: Ruell, JA De Clercq, E Pannecouque, C Witvrouw, M Stup, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Ja. Ruell et al., Synthesis and anti-HIV activity of cosalane analogues with substituted benzoic acid rings attached to the pharmacophore through methylene and amide linkers, J ORG CHEM, 64(16), 1999, pp. 5858-5866
Novel modifications in the alkenyldiarylmethane (ADAM) series of non-nucleoside reverse transcriptase inhibitors
Authors: Casimiro-Garcia, A Micklatcher, M Turpin, JA Stup, TL Watson, K Buckheit, RW Cushman, M
Citation: A. Casimiro-garcia et al., Novel modifications in the alkenyldiarylmethane (ADAM) series of non-nucleoside reverse transcriptase inhibitors, J MED CHEM, 42(23), 1999, pp. 4861-4874
Synthesis and biological activity of 2 '-fluoro-D-arabinofuranosylpyrazolo[3,4-d]pyrimidine nucleosides
Authors: Shortnacy-Fowler, AT Tiwari, KN Montgomery, JA Buckheit, RW Secrist, JA Seela, FA
Citation: At. Shortnacy-fowler et al., Synthesis and biological activity of 2 '-fluoro-D-arabinofuranosylpyrazolo[3,4-d]pyrimidine nucleosides, HELV CHIM A, 82(12), 1999, pp. 2240-2245
Antiviral oligo- and polyribonucleotides containing selected triazolo[2,3-a]purines
Authors: Tutonda, MG Buckheit, RW Agrawal, VK Broom, AD
Citation: Mg. Tutonda et al., Antiviral oligo- and polyribonucleotides containing selected triazolo[2,3-a]purines, J MED CHEM, 41(25), 1998, pp. 4958-4964
Risultati: 1-21 |