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Results: 1-21 |
Results: 21
SYNTHESIS AND ANTICHOLINESTERASE ACTIVITY OF HUPERZINE-A ANALOGS CONTAINING PHENOL AND CATECHOL REPLACEMENTS FOR THE PYRIDONE RING
Authors: CAMPIANI G KOZIKOWSKI AP WANG SM MING L NACCI V SAXENA A DOCTOR BP
Citation: G. Campiani et al., SYNTHESIS AND ANTICHOLINESTERASE ACTIVITY OF HUPERZINE-A ANALOGS CONTAINING PHENOL AND CATECHOL REPLACEMENTS FOR THE PYRIDONE RING, Bioorganic & medicinal chemistry letters, 8(11), 1998, pp. 1413-1418
NEW ANTIPSYCHOTIC AGENTS WITH SEROTONIN AND DOPAMINE ANTAGONIST PROPERTIES BASED ON A PYRROLO[2,1-B][1,3]BENZOTHIAZEPINE STRUCTURE
Authors: CAMPIANI G NACCI V BECHELLI S CIANI SM GAROFALO A FIORINI I WIKSTROM H DEBOER P LIAO Y TEPPER PG CAGNOTTO A MENNINI T
Citation: G. Campiani et al., NEW ANTIPSYCHOTIC AGENTS WITH SEROTONIN AND DOPAMINE ANTAGONIST PROPERTIES BASED ON A PYRROLO[2,1-B][1,3]BENZOTHIAZEPINE STRUCTURE, Journal of medicinal chemistry, 41(20), 1998, pp. 3763-3772
ANTIPROLIFERATIVE ACTION OF PYRROLOBENZOXAZEPINE DERIVATIVES IN CULTURED-CELLS - ABSENCE OF CORRELATION WITH BINDING TO THE PERIPHERAL-TYPEBENZODIAZEPINE BINDING-SITE
Authors: ZISTERER DM HANCE N CAMPIANI G GAROFALO A NACCI V WILLIAMS DC
Citation: Dm. Zisterer et al., ANTIPROLIFERATIVE ACTION OF PYRROLOBENZOXAZEPINE DERIVATIVES IN CULTURED-CELLS - ABSENCE OF CORRELATION WITH BINDING TO THE PERIPHERAL-TYPEBENZODIAZEPINE BINDING-SITE, Biochemical pharmacology, 55(4), 1998, pp. 397-403
NEW PYRROLOBENZOTHIAZEPINE DERIVATIVES AS MOLECULAR PROBES OF THE PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR (PBR) BINDING-SITE
Authors: CAMPIANI G NACCI V FIORINI I DEFILIPPIS MP GAROFALO A CIANI SM GRECO G NOVELLINO E MANZONI C MENNINI T
Citation: G. Campiani et al., NEW PYRROLOBENZOTHIAZEPINE DERIVATIVES AS MOLECULAR PROBES OF THE PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR (PBR) BINDING-SITE, European journal of medicinal chemistry, 32(3), 1997, pp. 241-251
NOVEL AND HIGHLY POTENT 5-HT3 RECEPTOR AGONISTS BASED ON A PYRROLOQUINOXALINE STRUCTURE
Authors: CAMPIANI G CAPPELLI A NACCI V ANZINI M VOMERO S HAMON M CAGNOTTO A FRACASSO C UBOLDI C CACCIA S CONSOLO S MENNINI T
Citation: G. Campiani et al., NOVEL AND HIGHLY POTENT 5-HT3 RECEPTOR AGONISTS BASED ON A PYRROLOQUINOXALINE STRUCTURE, Journal of medicinal chemistry, 40(22), 1997, pp. 3670-3678
DILTIAZEM-LIKE CALCIUM-ENTRY BLOCKERS - A HYPOTHESIS OF THE RECEPTOR-BINDING SITE BASED ON A COMPARATIVE MOLECULAR-FIELD ANALYSIS MODEL
Authors: CORELLI F MANETTI F TAFI A CAMPIANI G NACCI V BOTTA M
Citation: F. Corelli et al., DILTIAZEM-LIKE CALCIUM-ENTRY BLOCKERS - A HYPOTHESIS OF THE RECEPTOR-BINDING SITE BASED ON A COMPARATIVE MOLECULAR-FIELD ANALYSIS MODEL, Journal of medicinal chemistry, 40(1), 1997, pp. 125-131
AN APPROACH TO MODIFIED HETEROCYCLIC-ANALOGS OF HUPERZINE-A AND ISOHUPERZINE-A - SYNTHESIS OF THE PYRIMIDONE AND PYRAZOLE ANALOGS, AND THEIR ANTICHOLINESTERASE ACTIVITY
Authors: KOZIKOWSKI AP CAMPIANI G NACCI V SEGA A SAXENA A DOCTOR BP
Citation: Ap. Kozikowski et al., AN APPROACH TO MODIFIED HETEROCYCLIC-ANALOGS OF HUPERZINE-A AND ISOHUPERZINE-A - SYNTHESIS OF THE PYRIMIDONE AND PYRAZOLE ANALOGS, AND THEIR ANTICHOLINESTERASE ACTIVITY, Journal of the Chemical Society. Perkin transactions. I, (11), 1996, pp. 1287-1297
POLYCONDENSED HETEROCYCLES .9. PYRROLO[2,1-C][1,4]BENZOTHIAZEPINES - SYNTHESIS OF 3-(DIMETHYLAMINO)METHYL DERIVATIVES
Authors: GAROFALO A CAMPIANI G CIANI SM FIORINI I NACCI V
Citation: A. Garofalo et al., POLYCONDENSED HETEROCYCLES .9. PYRROLO[2,1-C][1,4]BENZOTHIAZEPINES - SYNTHESIS OF 3-(DIMETHYLAMINO)METHYL DERIVATIVES, Tetrahedron, 52(22), 1996, pp. 7745-7754
SYNTHESIS, BIOLOGICAL-ACTIVITY, AND SARS OF PYRROLOBENZOXAZEPINE DERIVATIVES, A NEW CLASS OF SPECIFIC PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR LIGANDS
Authors: CAMPIANI G NACCI V FIORINI I DEFILIPPIS MP GAROFALO A CIANI SM GRECO G NOVELLINO E WILLIAMS DC ZISTERER DM WOODS MJ MIHAI C MANZONI C MENNINI T
Citation: G. Campiani et al., SYNTHESIS, BIOLOGICAL-ACTIVITY, AND SARS OF PYRROLOBENZOXAZEPINE DERIVATIVES, A NEW CLASS OF SPECIFIC PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR LIGANDS, Journal of medicinal chemistry, 39(18), 1996, pp. 3435-3450
CARDIOVASCULAR CHARACTERIZATION OF PYRROLO[2,1-D][1,5]BENZOTHIAZEPINEDERIVATIVES BINDING SELECTIVELY TO THE PERIPHERAL-TYPE BENZODIAZEPINERECEPTOR (PBR) - FROM DUAL PBR AFFINITY AND CALCIUM-ANTAGONIST ACTIVITY TO NOVEL AND SELECTIVE CALCIUM-ENTRY BLOCKERS
Authors: CAMPIANI G FIORINI I DEFILIPPIS MP CIANI SM GAROFALO A NACCI V GIORGI G SEGA A BOTTA M CHIARINI A BUDRIESI R BRUNI G ROMEO MR MANZONI C MENNINI T
Citation: G. Campiani et al., CARDIOVASCULAR CHARACTERIZATION OF PYRROLO[2,1-D][1,5]BENZOTHIAZEPINEDERIVATIVES BINDING SELECTIVELY TO THE PERIPHERAL-TYPE BENZODIAZEPINERECEPTOR (PBR) - FROM DUAL PBR AFFINITY AND CALCIUM-ANTAGONIST ACTIVITY TO NOVEL AND SELECTIVE CALCIUM-ENTRY BLOCKERS, Journal of medicinal chemistry, 39(15), 1996, pp. 2922-2938
PYRROLOBENZOTHIAZEPINONES AND PYRROLOBENZOXAZEPINONES - NOVEL AND SPECIFIC NONNUCLEOSIDE HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS WITH ANTIVIRAL ACTIVITY
Authors: CAMPIANI G NACCI V FIORINI I DEFILIPPIS MP GAROFALO A GRECO G NOVELLINO E ALTAMURA S DIRENZO L
Citation: G. Campiani et al., PYRROLOBENZOTHIAZEPINONES AND PYRROLOBENZOXAZEPINONES - NOVEL AND SPECIFIC NONNUCLEOSIDE HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS WITH ANTIVIRAL ACTIVITY, Journal of medicinal chemistry, 39(14), 1996, pp. 2672-2680
IDENTIFICATION OF A MORE POTENT ANALOG OF THE NATURALLY-OCCURRING ALKALOID HUPERZINE-A - PREDICTIVE MOLECULAR MODELING OF ITS INTERACTION WITH ACHE
Authors: KOZIKOWSKI AP CAMPIANI G SUN LQ WANG SM SAXENA A DOCTOR BP
Citation: Ap. Kozikowski et al., IDENTIFICATION OF A MORE POTENT ANALOG OF THE NATURALLY-OCCURRING ALKALOID HUPERZINE-A - PREDICTIVE MOLECULAR MODELING OF ITS INTERACTION WITH ACHE, Journal of the American Chemical Society, 118(46), 1996, pp. 11357-11362
SYNTHESIS AND ACETYLCHOLINESTERASE INHIBITORY ACTIVITY OF SEVERAL PYRIMIDONE ANALOGS OF HUPERZINE-A
Authors: KOZIKOWSKI AP CAMPIANI G SAXENA A DOCTOR BP
Citation: Ap. Kozikowski et al., SYNTHESIS AND ACETYLCHOLINESTERASE INHIBITORY ACTIVITY OF SEVERAL PYRIMIDONE ANALOGS OF HUPERZINE-A, Journal of the Chemical Society, Chemical Communications, (2), 1995, pp. 283-285
A CONCERTED STUDY USING BINDING MEASUREMENTS, X-RAY STRUCTURAL DATA, AND MOLECULAR MODELING ON THE STEREOCHEMICAL FEATURES RESPONSIBLE FOR THE AFFINITY OF 6-ARYLPYRROLO[2,1-D][1,5]BENZOTHIAZEPINES TOWARD MITOCHONDRIAL BENZODIAZEPINE RECEPTORS
Authors: DALPIAZ A BERTOLASI V BOREA PA NACCI V FIORINI I CAMPIANI G MENNINI T MANZONI C NOVELLINO E GRECO G
Citation: A. Dalpiaz et al., A CONCERTED STUDY USING BINDING MEASUREMENTS, X-RAY STRUCTURAL DATA, AND MOLECULAR MODELING ON THE STEREOCHEMICAL FEATURES RESPONSIBLE FOR THE AFFINITY OF 6-ARYLPYRROLO[2,1-D][1,5]BENZOTHIAZEPINES TOWARD MITOCHONDRIAL BENZODIAZEPINE RECEPTORS, Journal of medicinal chemistry, 38(23), 1995, pp. 4730-4738
PYRROLO[2,1-C][1,4] BENZOTHIAZINES - SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, MOLECULAR MODELING STUDIES, AND CARDIOVASCULAR ACTIVITY
Authors: CAMPIANI G GAROFALO A FIORINI I BETTA M NACCI V TAFI A CHIARINI A BUDRIESI R BRUNI G ROMEO MR
Citation: G. Campiani et al., PYRROLO[2,1-C][1,4] BENZOTHIAZINES - SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, MOLECULAR MODELING STUDIES, AND CARDIOVASCULAR ACTIVITY, Journal of medicinal chemistry, 38(22), 1995, pp. 4393-4410
SYNTHESIS AND IN-VITRO CARDIOVASCULAR ACTIVITY OF TRAHYDRO-1H-PYRROLO[2,1-C][1,4]BENZOTHIAZIN-1-ONES AND TETRAHYDROPYRROLO[2,1-D][1,5]BENZOTHIAZEPIN-10-ONE
Authors: CAMPIANI G GAROFALO A FIORINI I NACCI V BOTTA M TAFI A CHIARINI A BUDRIESI R BRUNI G ROMEO MR
Citation: G. Campiani et al., SYNTHESIS AND IN-VITRO CARDIOVASCULAR ACTIVITY OF TRAHYDRO-1H-PYRROLO[2,1-C][1,4]BENZOTHIAZIN-1-ONES AND TETRAHYDROPYRROLO[2,1-D][1,5]BENZOTHIAZEPIN-10-ONE, Bioorganic & medicinal chemistry letters, 4(10), 1994, pp. 1235-1240
AN APPROACH TO OPEN-CHAIN AND MODIFIED HETEROCYCLIC-ANALOGS OF THE ACETYLCHOLINESTERASE INHIBITOR, HUPERZINE-A, THROUGH A BICYCLO[3.3.1]NONANE INTERMEDIATE
Authors: KOZIKOWSKI AP CAMPIANI G TUCKMANTEL W
Citation: Ap. Kozikowski et al., AN APPROACH TO OPEN-CHAIN AND MODIFIED HETEROCYCLIC-ANALOGS OF THE ACETYLCHOLINESTERASE INHIBITOR, HUPERZINE-A, THROUGH A BICYCLO[3.3.1]NONANE INTERMEDIATE, Heterocycles, 39(1), 1994, pp. 101-116
A COMPARATIVE MOLECULAR-FIELD ANALYSIS MODEL FOR 6-ARYLPYRROLO[2,1-D][1,5]BENZOTHIAZEPINES BINDING SELECTIVELY TO THE MITOCHONDRIAL BENZODIAZEPINE RECEPTOR
Authors: GRECO G NOVELLINO E FIORINI I NACCI V CAMPIANI G CIANI SM GAROFALO A BERNASCONI P MENNINI T
Citation: G. Greco et al., A COMPARATIVE MOLECULAR-FIELD ANALYSIS MODEL FOR 6-ARYLPYRROLO[2,1-D][1,5]BENZOTHIAZEPINES BINDING SELECTIVELY TO THE MITOCHONDRIAL BENZODIAZEPINE RECEPTOR, Journal of medicinal chemistry, 37(24), 1994, pp. 4100-4108
NOVEL LIGANDS SPECIFIC FOR MITOCHONDRIAL BENZODIAZEPINE RECEPTORS - 6-ARYLPYRROLO[2,1-D][1,5]BENZOTHIAZEPINE DERIVATIVES - SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, AND MOLECULAR MODELING STUDIES
Authors: FIORINI I NACCI V CIANI SM GAROFALO A CAMPIANI G SAVINI L NOVELLINO E GRECO G BERNASCONI P MENNINI T
Citation: I. Fiorini et al., NOVEL LIGANDS SPECIFIC FOR MITOCHONDRIAL BENZODIAZEPINE RECEPTORS - 6-ARYLPYRROLO[2,1-D][1,5]BENZOTHIAZEPINE DERIVATIVES - SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, AND MOLECULAR MODELING STUDIES, Journal of medicinal chemistry, 37(10), 1994, pp. 1427-1438
AN IMPROVED SYNTHETIC ROUTE TO HUPERZINE-A - NEW ANALOGS AND THEIR INHIBITION OF ACETYLCHOLINESTERASE
Authors: KOZIKOWSKI AP CAMPIANI G AAGAARD P MCKINNEY M
Citation: Ap. Kozikowski et al., AN IMPROVED SYNTHETIC ROUTE TO HUPERZINE-A - NEW ANALOGS AND THEIR INHIBITION OF ACETYLCHOLINESTERASE, Journal of the Chemical Society, Chemical Communications, (10), 1993, pp. 860-862
A PALLADIUM-CATALYZED ROUTE TO HUPERZINE-A AND ITS ANALOGS AND THEIR ANTICHOLINESTERASE ACTIVITY
Authors: CAMPIANI G SUN LQ KOZIKOWSKI AP AAGAARD P MCKINNEY M
Citation: G. Campiani et al., A PALLADIUM-CATALYZED ROUTE TO HUPERZINE-A AND ITS ANALOGS AND THEIR ANTICHOLINESTERASE ACTIVITY, Journal of organic chemistry, 58(27), 1993, pp. 7660-7669
Risultati: 1-21 |