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Results: 1-12 |
Results: 12
2-AMINO-4H-3,1-BENZOXAZIN-4-ONES AS INHIBITORS OF C1R SERINE-PROTEASE
Authors: HAYS SJ CAPRATHE BW GILMORE JL AMIN N EMMERLING MR MICHAEL W NADIMPALLI R NATH R RASER KJ STAFFORD D WATSON D WANG K JAEN JC
Citation: Sj. Hays et al., 2-AMINO-4H-3,1-BENZOXAZIN-4-ONES AS INHIBITORS OF C1R SERINE-PROTEASE, Journal of medicinal chemistry, 41(7), 1998, pp. 1060-1067
DESIGN AND SYNTHESIS OF M1-SELECTIVE MUSCARINIC AGONISTS - (R)-(-)-(Z)-1-AZABICYCLO[2.2.1]HEPTAN-3-ONE, O-(3-(3'-METHOXYPHENYL)-2-PROPYNYL)OXIME MALEATE (CI-1017), A FUNCTIONALLY M1-SELECTIVE MUSCARINIC AGONIST
Authors: TECLE H BARRETT SD LAUFFER DJ AUGELLISZAFRAN C BRANN MR CALLAHAN MJ CAPRATHE BW DAVIS RE DOYLE PD EUBANKS D LIPINISKI W MIRZADEGAN T MOOS WH MORELAND DW NELSON CB PAVIA MR RABY C SCHWARZ RD SPENCER CJ THOMAS AJ JAEN JC
Citation: H. Tecle et al., DESIGN AND SYNTHESIS OF M1-SELECTIVE MUSCARINIC AGONISTS - (R)-(-)-(Z)-1-AZABICYCLO[2.2.1]HEPTAN-3-ONE, O-(3-(3'-METHOXYPHENYL)-2-PROPYNYL)OXIME MALEATE (CI-1017), A FUNCTIONALLY M1-SELECTIVE MUSCARINIC AGONIST, Journal of medicinal chemistry, 41(14), 1998, pp. 2524-2536
EFFICIENT SYNTHESIS OF EXO-1-AZABICYCLO[2.2.1]HEPTAN-3-OL
Authors: BARRETT SD JAEN JC CAPRATHE BW THOMAS AJ TECLE H
Citation: Sd. Barrett et al., EFFICIENT SYNTHESIS OF EXO-1-AZABICYCLO[2.2.1]HEPTAN-3-OL, Organic preparations and procedures international, 29(3), 1997, pp. 330-335
SYNTHESIS AND EVALUATION OF 2-ARYL-4H-3,1-BENZOXAZIN-4-ONES AS C1R SERINE-PROTEASE INHIBITORS
Authors: GILMORE JL HAYS SJ CAPRATHE BW LEE C EMMERLING MR MICHAEL W JAEN JC
Citation: Jl. Gilmore et al., SYNTHESIS AND EVALUATION OF 2-ARYL-4H-3,1-BENZOXAZIN-4-ONES AS C1R SERINE-PROTEASE INHIBITORS, Bioorganic & medicinal chemistry letters, 6(6), 1996, pp. 679-682
IDENTIFICATION OF A 3-HYDROXYLATED TACRINE METABOLITE IN RAT AND MAN - METABOLIC PROFILING IMPLICATIONS AND PHARMACOLOGY
Authors: POOL WF WOOLF TF REILY MD CAPRATHE BW EMMERLING MR JAEN JC
Citation: Wf. Pool et al., IDENTIFICATION OF A 3-HYDROXYLATED TACRINE METABOLITE IN RAT AND MAN - METABOLIC PROFILING IMPLICATIONS AND PHARMACOLOGY, Journal of medicinal chemistry, 39(15), 1996, pp. 3014-3018
Z-(+ -)-1-AZABICYCLO [2.2.1]HEPTAN-3-ONE, O-(3-ARYL-2-PROPYNYL) OXIMES AS POTENTIAL M1-SUBTYPE SELECTIVE MUSCARINIC AGONISTS/
Authors: TECLE H JAEN JC AUGELLISZAFRAN C BARRETT SD CAPRATHE BW LAUFFER DJ MIRZADEGAN T MOOS WH MORELAND DW PAVIA MR SCHWARZ RD THOMAS AJ DAVIS RE
Citation: H. Tecle et al., Z-(+ -)-1-AZABICYCLO [2.2.1]HEPTAN-3-ONE, O-(3-ARYL-2-PROPYNYL) OXIMES AS POTENTIAL M1-SUBTYPE SELECTIVE MUSCARINIC AGONISTS/, Bioorganic & medicinal chemistry letters, 5(6), 1995, pp. 631-636
CI-1007, A DOPAMINE PARTIAL AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT.1. NEUROCHEMICAL EFFECTS
Authors: PUGSLEY TA DAVIS MD AKUNNE HC COOKE LW WHETZEL SZ MACKENZIE RG SHIH YH VANLEEUWEN DH DEMATTOS SB GEORGIC LM CAPRATHE BW WRIGHT JC JAEN JC WISE LD HEFFNER TG
Citation: Ta. Pugsley et al., CI-1007, A DOPAMINE PARTIAL AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT.1. NEUROCHEMICAL EFFECTS, The Journal of pharmacology and experimental therapeutics, 274(2), 1995, pp. 898-911
KYNURENIC ACID-DERIVATIVES INHIBIT THE BINDING OF NERVE GROWTH-FACTOR(NGF) TO THE LOW-AFFINITY P75 NGF RECEPTOR
Authors: JAEN JC LABORDE E BUCSH RA CAPRATHE BW SORENSON RJ FERGUS J SPIEGEL K MARKS J DICKERSON MR DAVIS RE
Citation: Jc. Jaen et al., KYNURENIC ACID-DERIVATIVES INHIBIT THE BINDING OF NERVE GROWTH-FACTOR(NGF) TO THE LOW-AFFINITY P75 NGF RECEPTOR, Journal of medicinal chemistry, 38(22), 1995, pp. 4439-4445
THE DISCOVERY AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF YDRO-4-PHENYL-1-[(ARYLCYCLOHEXENYL)ALKYL]PYRIDINES - DOPAMINE AUTORECEPTOR AGONISTS AND POTENTIAL ANTIPSYCHOTIC AGENTS
Authors: WRIGHT JL CAPRATHE BW DOWNING DM GLASE SA HEFFNER TG JAEN JC JOHNSON SJ KESTEN SR MACKENZIE RG MELTZER LT PUGSLEY TA SMITH SJ WISE LD WUSTROW DJ
Citation: Jl. Wright et al., THE DISCOVERY AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF YDRO-4-PHENYL-1-[(ARYLCYCLOHEXENYL)ALKYL]PYRIDINES - DOPAMINE AUTORECEPTOR AGONISTS AND POTENTIAL ANTIPSYCHOTIC AGENTS, Journal of medicinal chemistry, 37(21), 1994, pp. 3523-3533
ASSESSMENT OF MUTAGENIC POTENTIAL IN A SERIES OF COMPOUNDS STRUCTURALLY RELATED TO 2-AMINO-3-METHYLIMIDAZO [4,5-F]QUINOLINE (IQ)
Authors: JAEN JC KROPKO ML THEISS JC WOLD S CAPRATHE BW WISE LD
Citation: Jc. Jaen et al., ASSESSMENT OF MUTAGENIC POTENTIAL IN A SERIES OF COMPOUNDS STRUCTURALLY RELATED TO 2-AMINO-3-METHYLIMIDAZO [4,5-F]QUINOLINE (IQ), European journal of medicinal chemistry, 28(7-8), 1993, pp. 547-553
PHARMACOLOGICAL PROFILE OF THE DOPAMINE PARTIAL AGONIST, (+ --PD-128483 AND ITS ENANTIOMERS/
Authors: MELTZER LT CAPRATHE BW CHRISTOFFERSEN CL CORBIN AE JAEN JC NINTEMAN FW PUGSLEY TA SERPA KA SHIH YH WHETZEL SZ WILEY JN WISE LD HEFFNER TG
Citation: Lt. Meltzer et al., PHARMACOLOGICAL PROFILE OF THE DOPAMINE PARTIAL AGONIST, (+ --PD-128483 AND ITS ENANTIOMERS/, The Journal of pharmacology and experimental therapeutics, 266(3), 1993, pp. 1177-1189
EVALUATION OF THE EFFECTS OF THE ENANTIOMERS OF REDUCED HALOPERIDOL, AZAPEROL, AND RELATED 4-AMINO-1-ARYLBUTANOLS ON DOPAMINE AND SIGMA-RECEPTORS
Authors: JAEN JC CAPRATHE BW PUGSLEY TA WISE LD AKUNNE H
Citation: Jc. Jaen et al., EVALUATION OF THE EFFECTS OF THE ENANTIOMERS OF REDUCED HALOPERIDOL, AZAPEROL, AND RELATED 4-AMINO-1-ARYLBUTANOLS ON DOPAMINE AND SIGMA-RECEPTORS, Journal of medicinal chemistry, 36(24), 1993, pp. 3929-3936
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