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Results: 1-23 |
Results: 23
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A(2B) adenosine receptor antagonists
Authors: Baraldi, PG Cacciari, B Romagnoli, R Klotz, KN Spalluto, G Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A(2B) adenosine receptor antagonists, DRUG DEV R, 53(2-3), 2001, pp. 225-235
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new pharmacological tool for the characterization of the human A(3) adenosine receptor
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Varani, K Cessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new pharmacological tool for the characterization of the human A(3) adenosine receptor, DRUG DEV R, 52(1-2), 2001, pp. 406-415
Fluorosulfonyl- and bis-(beta-chloroethyl)amino-phenylamino functionalizedpyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: Irreversible antagonists at the human A(3) adenosine receptor and molecular modeling studies
Authors: Baraldi, PG Cacciari, B Moro, S Romagnoli, R Ji, XD Jacobson, KA Gessi, S Borea, PA Spalluto, G
Citation: Pg. Baraldi et al., Fluorosulfonyl- and bis-(beta-chloroethyl)amino-phenylamino functionalizedpyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: Irreversible antagonists at the human A(3) adenosine receptor and molecular modeling studies, J MED CHEM, 44(17), 2001, pp. 2735-2742
[2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding totranscription factor Sp1
Authors: Baraldi, PG Cacciari, B Guiotto, A Romagnoli, R Spalluto, G Leoni, A Bianchi, N Feriotto, G Rutigliano, C Mischiati, C Gambari, R
Citation: Pg. Baraldi et al., [2,1-c][1,4]benzodiazepine (PBD)-distamycin hybrid inhibits DNA binding totranscription factor Sp1, NUCLEOS NUC, 19(8), 2000, pp. 1219-1229
DNA minor groove alkylating agents structurally related to distamycin A
Authors: Baraldi, PG Spalluto, G Cacciari, B Romagnoli, R
Citation: Pg. Baraldi et al., DNA minor groove alkylating agents structurally related to distamycin A, EXPERT OP T, 10(6), 2000, pp. 891-904
CC-1065 and the duocarmycins: recent developments
Authors: Cacciari, B Romagnoli, R Baraldi, PG Da Ros, T Spalluto, G
Citation: B. Cacciari et al., CC-1065 and the duocarmycins: recent developments, EXPERT OP T, 10(12), 2000, pp. 1853-1871
Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors
Authors: Baraldi, PG Cacciari, B Romagnoli, R Varani, K Merighi, S Gessi, S Borea, PA Leung, E Hickey, SL Spalluto, G
Citation: Pg. Baraldi et al., Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors, BIOORG MED, 10(3), 2000, pp. 209-211
Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors (vol 10, pg 209, 2000)
Authors: Baraldi, PG Cacciari, B Romagnoli, R Varani, K Merighi, S Gessi, S Borea, PA Leung, E Hickey, SL Spalluto, G
Citation: Pg. Baraldi et al., Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors (vol 10, pg 209, 2000), BIOORG MED, 10(12), 2000, pp. 1403-1403
A(3) adenosine receptor ligands: History and perspectives
Authors: Baraldi, PG Cacciari, B Romagnoli, R Merighi, S Varani, K Borea, PA Spalluto, G
Citation: Pg. Baraldi et al., A(3) adenosine receptor ligands: History and perspectives, MED RES REV, 20(2), 2000, pp. 103-128
[H-3]MRE 3008F20: A novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors
Authors: Varani, K Merighi, S Gessi, S Klotz, KN Leung, E Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Borea, PA
Citation: K. Varani et al., [H-3]MRE 3008F20: A novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors, MOLEC PHARM, 57(5), 2000, pp. 968-975
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: Influence of thechain at the N-8 pyrazole nitrogen
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Moro, S Klotz, KN Leung, E Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: Influence of thechain at the N-8 pyrazole nitrogen, J MED CHEM, 43(25), 2000, pp. 4768-4780
Design, radiosynthesis, and biodistribution of a new potent and selective ligand for in vivo imaging of the adenosine A(2A) receptor system using positron emission tomography
Authors: Todde, S Moresco, RM Simonelli, F Baraldi, PG Cacciari, B Spalluto, G Varani, K Monopoli, A Matarrese, M Carpinelli, A Magni, F Kienle, MG Fazio, F
Citation: S. Todde et al., Design, radiosynthesis, and biodistribution of a new potent and selective ligand for in vivo imaging of the adenosine A(2A) receptor system using positron emission tomography, J MED CHEM, 43(23), 2000, pp. 4359-4362
A(1) and A(3) adenosine receptor agonists: an overview
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G
Citation: Pg. Baraldi et al., A(1) and A(3) adenosine receptor agonists: an overview, EXPERT OP T, 9(5), 1999, pp. 515-527
Resolution of a CPzI precursor, synthesis and biological evaluation of (+)and (-)-N-Boc-CPzI: A further validation of the relationship between chemical solvolytic stability and cytotoxicity
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Boyce, CW Boger, DL
Citation: Pg. Baraldi et al., Resolution of a CPzI precursor, synthesis and biological evaluation of (+)and (-)-N-Boc-CPzI: A further validation of the relationship between chemical solvolytic stability and cytotoxicity, BIOORG MED, 9(21), 1999, pp. 3087-3092
Selective binding to human genomic sequences of two synthetic analogues structurally related to U-71184 and adozelesin
Authors: Bianchi, N Spalluto, G Cacciari, B Romagnoli, R Feriotto, G Mischiati, C Rutigliano, C Borsetti, E Baraldi, PG Gambari, R
Citation: N. Bianchi et al., Selective binding to human genomic sequences of two synthetic analogues structurally related to U-71184 and adozelesin, DRUG DEV R, 46(2), 1999, pp. 96-106
Comparative molecular field analysis (CoMFA) of a series of selective adenosine receptor A(2A) antagonists
Authors: Baraldi, PG Borea, PA Bergonzoni, M Cacciari, B Ongini, E Recanatini, M Spalluto, G
Citation: Pg. Baraldi et al., Comparative molecular field analysis (CoMFA) of a series of selective adenosine receptor A(2A) antagonists, DRUG DEV R, 46(2), 1999, pp. 126-133
An efficient procedure for the synthesis of 5H-6-substituted-pyrazolo[1,5-d]-1,2,4-triazine-4,7-diones
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G
Citation: Pg. Baraldi et al., An efficient procedure for the synthesis of 5H-6-substituted-pyrazolo[1,5-d]-1,2,4-triazine-4,7-diones, SYNTHESIS-S, (3), 1999, pp. 453-458
Synthesis, in vitro antiproliferative activity, and DNA-binding propertiesof hybrid molecules containing pyrrolo[2,1-c][1,4]benzodiazepine and minor-groove-binding oligopyrrole carriers
Authors: Baraldi, PG Balboni, G Cacciari, B Guiotto, A Manfredini, S Romagnoli, R Spalluto, G Thurston, DE Howard, PW Bianchi, N Rutigliano, C Mischiati, C Gambari, R
Citation: Pg. Baraldi et al., Synthesis, in vitro antiproliferative activity, and DNA-binding propertiesof hybrid molecules containing pyrrolo[2,1-c][1,4]benzodiazepine and minor-groove-binding oligopyrrole carriers, J MED CHEM, 42(25), 1999, pp. 5131-5141
Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]-pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Klotz, KN Leung, E Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]-pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists, J MED CHEM, 42(22), 1999, pp. 4473-4478
Effect of A-ring modifications on the DNA-binding behavior and cytotoxicity of pyrrolo[2,1-c] [1,4]benzodiazepines
Authors: Thurston, DE Bose, DS Howard, PW Jenkins, TC Leoni, A Baraldi, PG Guiotto, A Cacciari, B Kelland, LR Foloppe, MP Rault, S
Citation: De. Thurston et al., Effect of A-ring modifications on the DNA-binding behavior and cytotoxicity of pyrrolo[2,1-c] [1,4]benzodiazepines, J MED CHEM, 42(11), 1999, pp. 1951-1964
DNA minor-groove binders: results and design of new antitumor agents
Authors: Baraldi, PG Cacciari, B Guiotto, A Romagnoli, R Zaid, AN Spalluto, G
Citation: Pg. Baraldi et al., DNA minor-groove binders: results and design of new antitumor agents, FARMACO, 54(1-2), 1999, pp. 15-25
1H-pyrazolo[2,3-d][1,2,4]triazine-3,7-diones as a new class of human leukocyte elastase inhibitors
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G
Citation: Pg. Baraldi et al., 1H-pyrazolo[2,3-d][1,2,4]triazine-3,7-diones as a new class of human leukocyte elastase inhibitors, ARZNEI-FOR, 49(12), 1999, pp. 997-1000
Heterocyclic analogs of pyrrolo [2,1-c] [1,4] benzodiazepines. Synthesis and structural requirements for their biological activity
Authors: Baraldi, PG Cacciari, B Guiotto, A Romagnoli, R Spalluto, G
Citation: Pg. Baraldi et al., Heterocyclic analogs of pyrrolo [2,1-c] [1,4] benzodiazepines. Synthesis and structural requirements for their biological activity, RRD ORG CHE, 2, 1998, pp. 567-591
Risultati: 1-23 |