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Results:
1-25
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Results: 25
Authors:
Lobaton, E
Velazquez, S
Perez-Perez, MJ
Jimeno, ML
San-Felix, A
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: E. Lobaton et al., "Second generation" of TSAO compounds directed against HIV-1 TSAO-resistant strains, NUCLEOS NUC, 20(4-7), 2001, pp. 707-710
Authors:
Lobaton, E
Velazquez, S
San-Felix, A
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: E. Lobaton et al., 4 ''-H-TSAO-T, a novel prototype in the HIV-1 specific TSAO family, NUCLEOS NUC, 20(4-7), 2001, pp. 711-714
Authors:
Chamorro, C
Lobaton, E
Bonache, MC
De Clercq, E
Balzarini, J
Velazquez, S
San-Felix, A
Camarasa, MJ
Citation: C. Chamorro et al., Identification of a novel family of nucleosides that specifically inhibit HIV-1 reverse transcriptase, BIOORG MED, 11(23), 2001, pp. 3085-3088
Authors:
Chamorro, C
Perez-Perez, MJ
Rodriguez-Barrios, F
Gago, F
De Clercq, E
Balzarini, J
San-Felix, A
Camarasa, MJ
Citation: C. Chamorro et al., Exploring the role of the 5 '-position of TSAO-T. Synthesis and anti-HIV evaluation of novel TSAO-T derivatives, ANTIVIR RES, 50(3), 2001, pp. 207-222
Authors:
Pelemans, H
Aertsen, A
Van Laethem, K
Vandamme, AM
De Clercq, E
Perez-Perez, MJ
San-Felix, A
Velazquez, S
Camarasa, MJ
Balzarini, J
Citation: H. Pelemans et al., Site-directed mutagenesis of human immunodeficiency virus type 1 reverse transcriptase at amino acid position 138, VIROLOGY, 280(1), 2001, pp. 97-106
Authors:
Priego, EM
Camarasa, MJ
Perez-Perez, MJ
Citation: Em. Priego et al., Efficient synthesis of N-3-substituted 6-aminouracil derivatives via N-6-[(Dimethylamino)methylene] protection, SYNTHESIS-S, (3), 2001, pp. 478-482
Authors:
Balzarini, J
Camarasa, MJ
Perez-Perez, MJ
San-Fleix, A
Velazquez, S
Perno, CF
De Clercq, E
Anderson, JN
Karlsson, A
Citation: J. Balzarini et al., Exploitation of the low fidelity of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase and the nucleotide composition bias in the HIV-1 genome to alter the drug resistance development of HIV, J VIROLOGY, 75(13), 2001, pp. 5772-5777
Authors:
Rodriguez-Barrios, F
Perez, C
Lobaton, E
Velazquez, S
Chamorro, C
San-Felix, A
Perez-Perez, MJ
Camarasa, MJ
Pelemans, H
Balzarini, J
Gago, F
Citation: F. Rodriguez-barrios et al., Identification of a putative binding site for [2 ',5 '-bis-O-(tert-butyldimethylsilyl)beta-D-ribofuranosyl]-3 '-spiro-5 ''-(4 ''-amino-1 '',2 ''-oxathiole-2 '',2 ''-dioxide)thymine (TSAO) derivatives at the p51-p66 interfaceof HIV-1 reverse transcriptase, J MED CHEM, 44(12), 2001, pp. 1853-1865
Authors:
Menendez-Arias, L
Abraha, A
Quinones-Mateu, ME
Mas, A
Camarasa, MJ
Arts, EJ
Citation: L. Menendez-arias et al., Functional characterization of chimeric reverse transcriptases with polypeptide subunits of highly divergent HIV-1 group M and O strains, J BIOL CHEM, 276(29), 2001, pp. 27470-27479
Authors:
Chamorro, C
De Clercq, E
Balzarini, J
Camarasa, MJ
San-Felix, A
Citation: C. Chamorro et al., TSAO-T analogues bearing amino acids at position N-3 of thymine: synthesisand anti-human immunodeficiency virus activity, ANTIVIR CHE, 11(1), 2000, pp. 61-69
Authors:
Lobaton, E
Camarasa, MJ
Velazquez, S
Citation: E. Lobaton et al., An efficient synthesis of 3 '-spiro sultone nucleosides functionalized on the sultone moiety via Pd-catalyzed cross-coupling reaction, SYNLETT, (9), 2000, pp. 1312-1314
Authors:
Van Laethem, K
Schmit, JC
Pelemans, H
Balzarini, J
Witvrouw, M
Perez-Perez, MJ
Camarasa, MJ
Esnouf, RM
Aquaro, S
Cenci, A
Perno, CF
Hermans, P
Sprecher, S
Ruiz, L
Clotet, B
Van Wijngaerden, E
Van Ranst, M
Desmyter, J
De Clercq, E
Vandamme, AM
Citation: K. Van Laethem et al., Presence of 2 ',5 '-bis-O-(tert-butyldimethylsilyl)-3 '-spiro-5 ''-(4 ''-amino-1 '',2 ''-oxathiole-2 '',2 ''-dioxide) (TSAO)-resistant virus strains in TSAO-inexperienced HIV patients, AIDS RES H, 16(9), 2000, pp. 825-833
Authors:
Camarasa, MJ
San-Felix, A
Perez-Perez, MJ
Velazquez, S
Alvarez, R
Chamorro, C
Jimeno, ML
Perez, C
Gago, F
De Clercq, E
Balzarini, J
Citation: Mj. Camarasa et al., HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique?, J CARB CHEM, 19(4-5), 2000, pp. 451-469
Authors:
San-Felix, A
Chamorro, C
Perez-Perez, MJ
Velazquez, S
de Clercq, E
Balzarini, J
Camarasa, MJ
Citation: A. San-felix et al., Synthesis of novel 5 '-substituted TSAO-T analogues with anti-HIV-1 activity, J CARB CHEM, 19(4-5), 2000, pp. 635-640
Authors:
Balzarini, J
Zhu, CY
De Clercq, E
Perez-Perez, MJ
Chamorro, C
Camarasa, MJ
Karlsson, A
Citation: J. Balzarini et al., Novel ribofuranosylnucleoside lead compounds for potent and selective inhibitors of mitochondrial thymidine kinase-2, BIOCHEM J, 351, 2000, pp. 167-171
Authors:
Esteban-Gamboa, A
Balzarini, J
Esnouf, R
De Clercq, E
Camarasa, MJ
Perez-Perez, MJ
Citation: A. Esteban-gamboa et al., Design, synthesis, and enzymatic evaluation of multisubstrate analogue inhibitors of Escherichia coli thymidine phosphorylase, J MED CHEM, 43(5), 2000, pp. 971-983
Authors:
Balzarini, J
Degreve, B
Esteban-Gamboa, A
Esnouf, R
De Clercq, E
Engelborghs, Y
Camarasa, MJ
Perez-Perez, MJ
Citation: J. Balzarini et al., Kinetic analysis of novel multisubstrate analogue inhibitors of thymidine phosphorylase, FEBS LETTER, 483(2-3), 2000, pp. 181-185
Authors:
Sluis-Cremer, N
Dmitrienko, GI
Balzarini, J
Camarasa, MJ
Parniak, MA
Citation: N. Sluis-cremer et al., Human immunodeficiency virus type 1 reverse transcriptase dimer destabilization by 1-{spiro[4 ''-amino-2 '',2 ''-dioxo-1 '',2 ''-oxathiole-5 '',3 '-[2 ',5 '-bis-O-(tert-butyldimethylsilyl)-beta-D-ribofuranosyl]]}-3-ethylthymine, BIOCHEM, 39(6), 2000, pp. 1427-1433
Authors:
Lobaton, E
Velazquez, S
San-Felix, A
Chamorro, C
Tunon, V
Esteban-Gamboa, A
De Clercq, E
Balzarini, J
Camarasa, MJ
Perez-Perez, MJ
Citation: E. Lobaton et al., Novel TSAO derivatives modified at positions 3 '' and 4 '' of the spiro moiety, NUCLEOS NUC, 18(4-5), 1999, pp. 675-676
Authors:
Chamorro, C
Velazquez, S
Jimeno, ML
Perez-Perez, MJ
Lobaton, E
Tunon, V
Esteban-Gamboa, A
Gago, F
De Clercq, E
Balzarini, J
Camarasa, MJ
San-Felix, A
Citation: C. Chamorro et al., Unexpected results in the reaction of 5 '-tosyl TSAO-m(3)t with amines, NUCLEOS NUC, 18(4-5), 1999, pp. 715-716
Authors:
Velazquez, S
Tunon, V
Jimeno, ML
Perez-Perez, MJ
San-Felix, A
Chamorro, C
Lobaton, E
Esteban-Gamboa, A
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: S. Velazquez et al., Novel series of [ddN]-[TSAO-T] heterodimers as potential bi-functional inhibitors of HIV-1 RT. Studies in the linker and ddN region, NUCLEOS NUC, 18(4-5), 1999, pp. 1029-1030
Authors:
Perez-Perez, MJ
Alvarez, R
Jimeno, ML
San-Felix, A
Lozano, A
Camarasa, MJ
Citation: Mj. Perez-perez et al., Steric and electronic properties of the 3 '-spiro moiety of TSAO-T and analogues, NUCLEOS NUC, 18(4-5), 1999, pp. 1107-1108
Authors:
Camarasa, MJ
Jimeno, ML
Perez-Perez, MJ
Alvarez, R
Velazquez, S
Lozano, A
Citation: Mj. Camarasa et al., Synthesis, NMR studies and theoretical calculations of novel 3-spiro-branched ribofuranoses, TETRAHEDRON, 55(41), 1999, pp. 12187-12200
Authors:
Velazquez, S
Tunon, V
Jimeno, ML
Chamorro, C
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: S. Velazquez et al., Potential multifunctional inhibitors of HIV-1 reverse transcriptase. Novel[AZT]-[TSAO-T] and [d4T]-[TSAO-T] heterodimers modified in the linker and in the dideoxynucleoside region, J MED CHEM, 42(25), 1999, pp. 5188-5196
Authors:
Velazquez, S
Alvarez, R
Perez, C
Gago, F
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: S. Velazquez et al., Regiospecific synthesis and anti-human immunodeficiency virus activity of novel 5-substituted N-alkylcarbamoyl and N,N-dialkyl carbamoyl 1,2,3-triazole-TSAO analogues, ANTIVIR CHE, 9(6), 1998, pp. 481-489
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