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Results: 1-14 |
Results: 14
Novel and potent tacrine-related hetero- and homobivalent ligands for acetylcholinesterase and butyrylcholinesterase
Authors: Savini, L Campiani, G Gaeta, A Pellerano, C Fattorusso, C Chiasserini, L Fedorko, JM Saxena, A
Citation: L. Savini et al., Novel and potent tacrine-related hetero- and homobivalent ligands for acetylcholinesterase and butyrylcholinesterase, BIOORG MED, 11(13), 2001, pp. 1779-1782
Pyrrolo-1,5-benzoxazepines: a new class of apoptotic agents
Authors: Zisterer, DM McGee, MM Campiani, G Ramunno, A Fattorusso, C Nacci, V Lawler, M Williams, DC
Citation: Dm. Zisterer et al., Pyrrolo-1,5-benzoxazepines: a new class of apoptotic agents, BIOCH SOC T, 29, 2001, pp. 704-706
Pyrrolo-1,5-benzoxazepines induce apoptosis in chronic myelogenous leukemia (CML) cells by bypassing the apoptotic suppressor Bcr-Abl
Authors: Mc Gee, MM Campiani, G Ramunno, A Fattorusso, C Nacci, V Lawler, M Williams, DC Zisterer, DM
Citation: Mm. Mc Gee et al., Pyrrolo-1,5-benzoxazepines induce apoptosis in chronic myelogenous leukemia (CML) cells by bypassing the apoptotic suppressor Bcr-Abl, J PHARM EXP, 296(1), 2001, pp. 31-40
Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent
Authors: Campiani, G Aiello, F Fabbrini, M Morelli, E Ramunno, A Armaroli, S Nacci, V Garofalo, A Greco, G Novellino, E Maga, G Spadari, S Bergamini, A Ventura, L Bongiovanni, B Capozzi, M Bolacchi, F Marini, S Coletta, M Guiso, G Caccia, S
Citation: G. Campiani et al., Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent, J MED CHEM, 44(3), 2001, pp. 305-315
A rational approach to the design of selective substrates and potent nontransportable inhibitors of the excitatory amino acid transporter EAAC1 (EAAT3). New glutamate and aspartate analogues as potential neuroprotective agents
Authors: Campiani, G De Angelis, M Armaroli, S Fattorusso, C Catalanotti, B Ramunno, A Nacci, V Novellino, E Grewer, C Ionescu, D Rauen, T Griffiths, R Sinclair, C Fumagalli, E Mennini, T
Citation: G. Campiani et al., A rational approach to the design of selective substrates and potent nontransportable inhibitors of the excitatory amino acid transporter EAAC1 (EAAT3). New glutamate and aspartate analogues as potential neuroprotective agents, J MED CHEM, 44(16), 2001, pp. 2507-2510
The stereoselective targeting of a specific enzyme-substrate complex is the molecular mechanism for the synergic inhibition of HIV-1 reverse transcriptase by (R)-(-)-PPO464 - A novel generation of nonnucleoside inhibitors
Authors: Maga, G Ramunno, A Nacci, V Locatelli, GA Spadari, S Fiorini, I Baldanti, F Paolucci, S Zavattoni, M Bergamini, A Galletti, B Muck, S Hubscher, U Giorgi, G Guiso, G Caccia, S Campiani, G
Citation: G. Maga et al., The stereoselective targeting of a specific enzyme-substrate complex is the molecular mechanism for the synergic inhibition of HIV-1 reverse transcriptase by (R)-(-)-PPO464 - A novel generation of nonnucleoside inhibitors, J BIOL CHEM, 276(48), 2001, pp. 44653-44662
Non-nucleoside HIV-1 reverse transcriptase inhibitors: synthesis and biological evaluation of novel quinoxalinylethylpyridylthioureas as potent antiviral agents
Authors: Campiani, G Fabbrini, M Morelli, E Nacci, V Greco, G Novellino, E Maga, G Spadari, S Bergamini, A Faggioli, E Uccella, I Bolacchi, F Marini, S Coletta, M Fracasso, C Caccia, S
Citation: G. Campiani et al., Non-nucleoside HIV-1 reverse transcriptase inhibitors: synthesis and biological evaluation of novel quinoxalinylethylpyridylthioureas as potent antiviral agents, ANTIVIR CHE, 11(2), 2000, pp. 141-155
Polycondensed heterocycles. Part 11: Preparation and regioselective reductions of 5-phenyl-4H-pyrrolo[1,2-a][1]benzazepin-4-one
Authors: Garofalo, A Ragno, G Campiani, G Brizzi, A Nacci, V
Citation: A. Garofalo et al., Polycondensed heterocycles. Part 11: Preparation and regioselective reductions of 5-phenyl-4H-pyrrolo[1,2-a][1]benzazepin-4-one, TETRAHEDRON, 56(47), 2000, pp. 9351-9355
Pyrrolo-1,5-benzoxazepines induce apoptosis in HL-60, Jurkat, and Hut-78 cells: A new class of apoptotic agents
Authors: Zisterer, DM Campiani, G Nacci, V Williams, DC
Citation: Dm. Zisterer et al., Pyrrolo-1,5-benzoxazepines induce apoptosis in HL-60, Jurkat, and Hut-78 cells: A new class of apoptotic agents, J PHARM EXP, 293(1), 2000, pp. 48-59
Preparation and biological properties of biotinylated PhTX derivatives
Authors: Hashimoto, M Liu, Y Fang, K Li, HY Campiani, G Nakanishi, K
Citation: M. Hashimoto et al., Preparation and biological properties of biotinylated PhTX derivatives, BIO MED CH, 7(6), 1999, pp. 1181-1194
Polycondensed heterocycles. X. A new method for the preparation of pyrrolo[2,1-c][1,4]benzothiazepines by intramolecular Mitsunobu cyclisation.
Authors: Garofalo, A Campiani, G Fiorini, I Nacci, V
Citation: A. Garofalo et al., Polycondensed heterocycles. X. A new method for the preparation of pyrrolo[2,1-c][1,4]benzothiazepines by intramolecular Mitsunobu cyclisation., TETRAHEDRON, 55(5), 1999, pp. 1479-1490
Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT3 receptor agonists: Synthesis, further structure-activity relationships, and biological studies
Authors: Campiani, G Morelli, E Gemma, S Nacci, V Butini, S Hamon, M Novellino, E Greco, G Cagnotto, A Goegan, M Cervo, L Dalla Valle, F Fracasso, C Caccia, S Mennini, T
Citation: G. Campiani et al., Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT3 receptor agonists: Synthesis, further structure-activity relationships, and biological studies, J MED CHEM, 42(21), 1999, pp. 4362-4379
Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: Further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity
Authors: Campiani, G Morelli, E Fabbrini, M Nacci, V Greco, G Novellino, E Ramunno, A Maga, G Spadari, S Caliendo, G Bergamini, A Faggioli, E Uccella, I Bolacchi, F Marini, S Coletta, M Nacca, A Caccia, S
Citation: G. Campiani et al., Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: Further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity, J MED CHEM, 42(21), 1999, pp. 4462-4470
Thiazolothiazepine inhibitors of HIV-1 integrase
Authors: Neamati, N Turpin, JA Winslow, HE Christensen, JL Williamson, K Orr, A Rice, WG Pommier, Y Garofalo, A Brizzi, A Campiani, G Fiorini, I Nacci, V
Citation: N. Neamati et al., Thiazolothiazepine inhibitors of HIV-1 integrase, J MED CHEM, 42(17), 1999, pp. 3334-3341
Risultati: 1-14 |