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Results: 1-16 |
Results: 16
Human beta(3) adrenergic receptor agonists containing cyanoguanidine and nitroethylenediamine moieties
Authors: Brockunier, LL Candelore, MR Cascieri, MA Liu, Y Tota, L Wyvratt, MJ Fisher, MH Weber, AE Parmee, ER
Citation: Ll. Brockunier et al., Human beta(3) adrenergic receptor agonists containing cyanoguanidine and nitroethylenediamine moieties, BIOORG MED, 11(3), 2001, pp. 379-382
beta(3)-adrenoceptor agonist-induced increases in lipolysis, metabolic rate, racial flushing, and reflex tachycardia in anesthetized rhesus monkeys
Authors: Hom, GJ Forrest, MJ Bach, TJ Brady, E Candelore, MR Cascieri, MA Fletcher, DJ Fisher, MH Iliff, SA Mathvink, R Metzger, J Pecore, V Saperstein, R Shih, T Weber, AE Wyvratt, M Zafian, P Macintyre, DE
Citation: Gj. Hom et al., beta(3)-adrenoceptor agonist-induced increases in lipolysis, metabolic rate, racial flushing, and reflex tachycardia in anesthetized rhesus monkeys, J PHARM EXP, 297(1), 2001, pp. 299-307
Tetrahydroisoquinoline derivatives containing a benzenesulfonamide moiety as potent, selective human beta(3) adrenergic receptor agonists
Authors: Parmee, ER Brockunier, LL He, JF Singh, SB Candelore, MR Cascieri, MA Deng, LP Liu, Y Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Er. Parmee et al., Tetrahydroisoquinoline derivatives containing a benzenesulfonamide moiety as potent, selective human beta(3) adrenergic receptor agonists, BIOORG MED, 10(20), 2000, pp. 2283-2286
Human beta 3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides
Authors: Brockunier, LL Parmee, ER Ok, HO Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Ll. Brockunier et al., Human beta 3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides, BIOORG MED, 10(18), 2000, pp. 2111-2114
Potent, selective 3-pyridylethanolamine beta(3) adrenergic receptor agonists possessing a thiazole benzenesulfonamide pharmacophore
Authors: Mathvink, RJ Tolman, JS Chitty, D Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Rj. Mathvink et al., Potent, selective 3-pyridylethanolamine beta(3) adrenergic receptor agonists possessing a thiazole benzenesulfonamide pharmacophore, BIOORG MED, 10(17), 2000, pp. 1971-1973
Substituted oxazole benzenesulfonamides as potent human beta(3) adrenergicreceptor agonists
Authors: Ok, HO Reigle, LB Candelore, MR Cascieri, MA Colwell, LF Deng, L Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Strader, CD Tota, L Wang, P Wyvratt, MJ Fisher, MH Weber, AE
Citation: Ho. Ok et al., Substituted oxazole benzenesulfonamides as potent human beta(3) adrenergicreceptor agonists, BIOORG MED, 10(14), 2000, pp. 1531-1534
Discovery of an orally bioavailable alkyl oxadiazole beta(3) adrenergic receptor agonist
Authors: Feng, DQD Biftu, T Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Strader, CD Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Dqd. Feng et al., Discovery of an orally bioavailable alkyl oxadiazole beta(3) adrenergic receptor agonist, BIOORG MED, 10(13), 2000, pp. 1427-1429
Synthesis and SAR of benzyl and phenoxymethylene oxadiazole benzenesulfonamides as selective beta(3) adrenergic receptor agonist antiobesity agents
Authors: Biftu, T Feng, DD Liang, GB Kuo, H Qian, XX Naylor, EM Colandrea, VJ Candelore, MR Cascieri, MA Colwell, LF Forrest, MJ Hom, GJ MacIntyre, DE Stearns, RA Strader, CD Wyvratt, MJ Fisher, MH Weber, AE
Citation: T. Biftu et al., Synthesis and SAR of benzyl and phenoxymethylene oxadiazole benzenesulfonamides as selective beta(3) adrenergic receptor agonist antiobesity agents, BIOORG MED, 10(13), 2000, pp. 1431-1434
Discovery of a potent, orally bioavailable beta(3) adrenergic receptor agonist, (R)-N-[4-[2-[[2-hydroxy-2-(3-pyridinyl)ethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethyl)phenyl]thiazol-2-yl]benzenesulfonamide
Authors: Mathvink, RJ Tolman, JS Chitty, D Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Rj. Mathvink et al., Discovery of a potent, orally bioavailable beta(3) adrenergic receptor agonist, (R)-N-[4-[2-[[2-hydroxy-2-(3-pyridinyl)ethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethyl)phenyl]thiazol-2-yl]benzenesulfonamide, J MED CHEM, 43(21), 2000, pp. 3832-3836
L-750355, a human beta 3-adrenoceptor agonist; in vitro pharmacology and profile of activity in vivo in the rhesus monkey
Authors: Forrest, MJ Hom, G Bach, T Candelore, MR Cascieri, MA Strader, C Tota, L Fisher, MH Szumiloski, J Ok, HO Weber, AE Wyvratt, M Vicario, P Marko, O Deng, LP Cioffe, C Hegarty-Friscino, B MacIntyre, E
Citation: Mj. Forrest et al., L-750355, a human beta 3-adrenoceptor agonist; in vitro pharmacology and profile of activity in vivo in the rhesus monkey, EUR J PHARM, 407(1-2), 2000, pp. 175-181
L-770,644: A potent and selective human beta(3) adrenergic receptor agonist with improved oral bioavailability
Authors: Shih, TL Candelore, MR Cascieri, MA Chiu, SHL Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Strader, CD Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Tl. Shih et al., L-770,644: A potent and selective human beta(3) adrenergic receptor agonist with improved oral bioavailability, BIOORG MED, 9(9), 1999, pp. 1251-1254
Human beta(3) adrenergic receptor agonists containing cyclic ureidobenzenesulfonamides
Authors: Parmee, ER Naylor, EM Perkins, L Colandrea, VJ Ok, HO Candelore, MR Cascieri, MA Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Miller, RR Stearns, RA Strader, CD Tota, L Wyvratt, MJ Fisher, MH Weber, AE
Citation: Er. Parmee et al., Human beta(3) adrenergic receptor agonists containing cyclic ureidobenzenesulfonamides, BIOORG MED, 9(5), 1999, pp. 749-754
Human beta(3) adrenergic receptor agonists containing imidazolidinone and imidazolone benzenesulfonamides
Authors: Naylor, EM Parmee, ER Colandrea, VJ Perkins, L Brockunier, L Candelore, MR Cascieri, MA Colwell, LF Deng, LP Feeney, WP Forrest, MJ Hom, GJ MacIntyre, DE Strader, CD Tota, L Wang, PR Wyvratt, MJ Fisher, MH Weber, AE
Citation: Em. Naylor et al., Human beta(3) adrenergic receptor agonists containing imidazolidinone and imidazolone benzenesulfonamides, BIOORG MED, 9(5), 1999, pp. 755-758
Potent, selective human beta(3) adrenergic receptor agonists containing a substituted indoline-5-sulfonamide pharmacophore
Authors: Mathvink, RJ Barritta, AM Candelore, MR Cascieri, MA Deng, LP Tota, L Strader, CD Wyvratt, MJ Fisher, MH Weber, AE
Citation: Rj. Mathvink et al., Potent, selective human beta(3) adrenergic receptor agonists containing a substituted indoline-5-sulfonamide pharmacophore, BIOORG MED, 9(13), 1999, pp. 1869-1874
Acute effect of ephedrine on 24-h energy balance
Authors: Shannon, JR Gottesdiener, K Jordan, J Chen, K Flattery, S Larson, PJ Candelore, MR Gertz, B Robertson, D Sun, M
Citation: Jr. Shannon et al., Acute effect of ephedrine on 24-h energy balance, CLIN SCI, 96(5), 1999, pp. 483-491
Potent and selective human beta(3)-adrenergic receptor antagonists
Authors: Candelore, MR Deng, LP Tota, L Guan, XM Amend, A Liu, Y Newbold, R Cascieri, MA Weber, AE
Citation: Mr. Candelore et al., Potent and selective human beta(3)-adrenergic receptor antagonists, J PHARM EXP, 290(2), 1999, pp. 649-655
Risultati: 1-16 |