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Authors:
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Muschaweck, NM
Maeda, DY
Coop, A
Ticku, MK
Citation: Ak. Mehta et al., Binding characteristics of the gamma-hydroxybutyric acid receptor antagonist [H-3](2E)-(5-hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene)ethanoic acid in the rat brain, J PHARM EXP, 299(3), 2001, pp. 1148-1153
Authors:
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Ullrich, T
Rothman, RB
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Jacobson, AE
Rice, KC
Citation: S. Mclamore et al., Effect of N-alkyl and N-alkenyl substituents in noroxymorphindole, 17-substituted-6,7-dehydro-4,5 alpha-epoxy-3,14-dihydroxy-6,7 : 2 ',3 '-indolomorphinans, on opioid receptor affinity, selectivity, and efficacy, J MED CHEM, 44(9), 2001, pp. 1471-1474
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Petros, TJ
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Citation: Sm. Huang et al., Identification of a new class of molecules, the arachidonyl amino acids, and characterization of one member that inhibits pain, J BIOL CHEM, 276(46), 2001, pp. 42639-42644
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Citation: A. Coop et al., N-cyclohexylethyl-N-noroxymorphindole: A mu-opioid preferring analogue of naltrindole, BIOORG MED, 10(21), 2000, pp. 2449-2451
Citation: Dy. Maeda et al., A sigma-1 receptor selective analogue of BD1008. A potential substitute for (+)-opioids in sigma receptor binding assays, BIOORG MED, 10(1), 2000, pp. 17-18
Authors:
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Coop, A
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Citation: I. Derrick et al., Perchloric acid induced epimerisation of the thevinones: an improved synthesis of 7 beta-dihydrothevinones, TETRAHEDR L, 41(39), 2000, pp. 7571-7576
Citation: Dy. Maeda et A. Coop, Studies into the direct conversion of indolomorphinans to their 4-phenolicderivatives, TETRAHEDRON, 56(38), 2000, pp. 7399-7402
Authors:
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Citation: Dc. Broom et al., BU48: A novel buprenorphine analog that exhibits delta-opioid-mediated convulsions but not delta-opioid-mediated antinociception in mice, J PHARM EXP, 294(3), 2000, pp. 1195-1200
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Citation: A. Coop et al., Structural determinants of opioid activity in the orvinols and related structures: Ethers of orvinol and isoorvinol, J MED CHEM, 43(9), 2000, pp. 1852-1857
Authors:
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Citation: Ms. Furness et al., Probes for narcotic receptor-mediated phenomena. 27. Synthesis and pharmacological evaluation of selective delta-opioid receptor agonists from 4-[(alpha R)-alpha-(2S,5R)-4-substituted-2,5-dimethyl-1-piperazinyl-3-methoxybenzyl]-N,N-diethylbenzamides and their enantiomers, J MED CHEM, 43(16), 2000, pp. 3193-3196
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Burnside, J
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Husbands, SM
Lewis, JW
Citation: A. Coop et al., Structural determinants of opioid activity in the orvinols and related structures. Ethers of 7,8-cyclopenta-fused analogs of buprenorphine, HELV CHIM A, 83(4), 2000, pp. 687-693
Citation: A. Coop et Ae. Jacobson, The LMC delta opioid recognition pharmacophore: Comparison of SNC80 and oxymorphindole, BIOORG MED, 9(3), 1999, pp. 357-362
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Guo, L
Coop, A
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Citation: Jr. Traynor et al., Ring-constrained orvinols as analogs of buprenorphine: Differences in opioid activity related to configuration of C-20 hydroxyl group, J PHARM EXP, 291(3), 1999, pp. 1093-1099
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Citation: A. Coop et al., delta opioid affinity and selectivity of 4-hydroxy-3-methoxyindolomorphinan analogues related to naltrindole, J MED CHEM, 42(9), 1999, pp. 1673-1679
Authors:
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Rice, KC
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Rothman, RB
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Citation: Xy. Zhang et al., Probes for narcotic receptor mediated phenomena. 26. Synthesis and biological evaluation of diarylmethylpiperazines and diarylmethylpiperidines as novel, nonpeptidic delta opioid receptor ligands, J MED CHEM, 42(26), 1999, pp. 5455-5463
Authors:
Breeden, SW
Coop, A
Husbands, SM
Lewis, JW
Citation: Sw. Breeden et al., 6-O-demethylation of the thevinols with lithium aluminium hydride: Selective demethylation of a tertiary alkyl methyl ether in the presence of an aryl methyl ether, HELV CHIM A, 82(11), 1999, pp. 1978-1980