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Results: 1-13 |
Results: 13
SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF PYRIDINE-MODIFIED ANALOGS OF 3-[2-((S)-PYRROLIDINYL)METHOXY]PYRIDINE, A-84543, A POTENT NICOTINIC ACETYLCHOLINE-RECEPTOR AGONIST
Authors: LIN NH GUNN DE LI YH HE Y BAI H RYTHER KB KUNTZWEILER T DONNELLYROBERTS DL ANDERSON DJ CAMPBELL JE SULLIVAN JP ARNERIC SP HOLLADAY MW
Citation: Nh. Lin et al., SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF PYRIDINE-MODIFIED ANALOGS OF 3-[2-((S)-PYRROLIDINYL)METHOXY]PYRIDINE, A-84543, A POTENT NICOTINIC ACETYLCHOLINE-RECEPTOR AGONIST, Bioorganic & medicinal chemistry letters, 8(3), 1998, pp. 249-254
STRUCTURE-ACTIVITY STUDIES RELATED TO ABT-594, A POTENT NONOPIOID ANALGESIC AGENT - EFFECT OF PYRIDINE AND AZETIDINE RING SUBSTITUTIONS ON NICOTINIC ACETYLCHOLINE-RECEPTOR BINDING-AFFINITY AND ANALGESIC ACTIVITY IN MICE
Authors: HOLLADAY MW BAI H LI YH LIN NH DAANEN JF RYTHER KB WASICAK JT KINCAID JF HE Y HETTINGER AM HUANG P ANDERSON DJ BANNON AW BUCKLEY MJ CAMPBELL JE DONNELLYROBERTS DL GUNTHER KL KIM DJB KUNTZWEILER TA SULLIVAN JP DECKER MW ARNERIC SP
Citation: Mw. Holladay et al., STRUCTURE-ACTIVITY STUDIES RELATED TO ABT-594, A POTENT NONOPIOID ANALGESIC AGENT - EFFECT OF PYRIDINE AND AZETIDINE RING SUBSTITUTIONS ON NICOTINIC ACETYLCHOLINE-RECEPTOR BINDING-AFFINITY AND ANALGESIC ACTIVITY IN MICE, Bioorganic & medicinal chemistry letters, 8(19), 1998, pp. 2797-2802
THE ROLE OF NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS IN ANTINOCICEPTION - EFFECTS OF ABT-594
Authors: DECKER MW CURZON P HOLLADAY MW NIKKEL AL BITNER RS BANNON AW DONNELLYROBERTS DL PUTTFARCKEN PS KUNTZWEILER TA BRIGGS CA WILLIAMS M ARNERIC SP
Citation: Mw. Decker et al., THE ROLE OF NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS IN ANTINOCICEPTION - EFFECTS OF ABT-594, J PHYSL-PAR, 92(3-4), 1998, pp. 221-224
RAPID ASSESSMENT OF LIGAND ACTIONS WITH NICOTINIC ACETYLCHOLINE-RECEPTORS USING CALCIUM DYNAMICS AND FLIPR
Authors: KUNTZWEILER TA ARNERIC SP DONNELLYROBERTS DL
Citation: Ta. Kuntzweiler et al., RAPID ASSESSMENT OF LIGAND ACTIONS WITH NICOTINIC ACETYLCHOLINE-RECEPTORS USING CALCIUM DYNAMICS AND FLIPR, Drug development research, 44(1), 1998, pp. 14-20
ABT-594 [(R)-5-(2-AZETIDINYLMETHOXY)-2-CHLOROPYRIDINE] - A NOVEL, ORALLY EFFECTIVE ANALGESIC ACTING VIA NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS - I - IN-VITRO CHARACTERIZATION
Authors: DONNELLYROBERTS DL PUTTFARCKEN PS KUNTZWEILER TA BRIGGS CA ANDERSON DJ CAMPBELL JE PIATTONIKAPLAN M MCKENNA DG WASICAK JT HOLLADAY MW WILLIAMS M ARNERIC SP
Citation: Dl. Donnellyroberts et al., ABT-594 [(R)-5-(2-AZETIDINYLMETHOXY)-2-CHLOROPYRIDINE] - A NOVEL, ORALLY EFFECTIVE ANALGESIC ACTING VIA NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS - I - IN-VITRO CHARACTERIZATION, The Journal of pharmacology and experimental therapeutics, 285(2), 1998, pp. 777-786
IDENTIFICATION AND INITIAL STRUCTURE-ACTIVITY-RELATIONSHIPS OF 5-(2-AZETIDINYLMETHOXY)-2-CHLOROPYRIDINE(ABT-594), A POTENT, ORALLY-ACTIVE, NONOPIATE ANALGESIC AGENT ACTING VIA NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS
Authors: HOLLADAY MW WASICAK JT LIN NH HE Y RYTHER KB BANNON AW BUCKLEY MJ KIM DJB DECKER MW ANDERSON DJ CAMPBELL JE KUNTZWEILER TA DONNELLYROBERTS DL PIATTONIKAPLAN M BRIGGS CA WILLIAMS M ARNERIC SP
Citation: Mw. Holladay et al., IDENTIFICATION AND INITIAL STRUCTURE-ACTIVITY-RELATIONSHIPS OF 5-(2-AZETIDINYLMETHOXY)-2-CHLOROPYRIDINE(ABT-594), A POTENT, ORALLY-ACTIVE, NONOPIATE ANALGESIC AGENT ACTING VIA NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS, Journal of medicinal chemistry, 41(4), 1998, pp. 407-412
EVIDENCE FOR NICOTINIC RECEPTORS POTENTIALLY MODULATING NOCICEPTIVE TRANSMISSION AT THE LEVEL OF THE PRIMARY SENSORY NEURON - STUDIES WITH F11 CELLS
Authors: PUTTFARCKEN PS MANELLI AM ARNERIC SP DONNELLYROBERTS DL
Citation: Ps. Puttfarcken et al., EVIDENCE FOR NICOTINIC RECEPTORS POTENTIALLY MODULATING NOCICEPTIVE TRANSMISSION AT THE LEVEL OF THE PRIMARY SENSORY NEURON - STUDIES WITH F11 CELLS, Journal of neurochemistry, 69(3), 1997, pp. 930-938
STRUCTURE-ACTIVITY STUDIES ON 2-METHYL-3-(2(S)-PYRROLIDINYLMETHOXY)PYRIDINE (ABT-089) - AN ORALLY BIOAVAILABLE 3-PYRIDYL ETHER NICOTINIC ACETYLCHOLINE-RECEPTOR LIGAND WITH COGNITION-ENHANCING PROPERTIES
Authors: LIN NH GUNN DE RYTHER KB GARVEY DS DONNELLYROBERTS DL DECKER MW BRIONI JD BUCKLEY MJ RODRIGUES AD MARSH KG ANDERSON DJ BUCCAFUSCO JJ PRENDERGAST MA SULLIVAN JP WILLIAMS M ARNERIC SP HOLLADAY MW
Citation: Nh. Lin et al., STRUCTURE-ACTIVITY STUDIES ON 2-METHYL-3-(2(S)-PYRROLIDINYLMETHOXY)PYRIDINE (ABT-089) - AN ORALLY BIOAVAILABLE 3-PYRIDYL ETHER NICOTINIC ACETYLCHOLINE-RECEPTOR LIGAND WITH COGNITION-ENHANCING PROPERTIES, Journal of medicinal chemistry, 40(3), 1997, pp. 385-390
NOVEL 3-PYRIDYL ETHERS WITH SUBNANOMOLAR AFFINITY FOR CENTRAL NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS
Authors: ABREO MA LIN NH GARVEY DS GUNN DE HETTINGER AM WASICAK JT PAVLIK PA MARTIN YC DONNELLYROBERTS DL ANDERSON DJ SULLIVAN JP WILLIAMS M AMERIC SP HOLLADAY MW
Citation: Ma. Abreo et al., NOVEL 3-PYRIDYL ETHERS WITH SUBNANOMOLAR AFFINITY FOR CENTRAL NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS, Journal of medicinal chemistry, 39(4), 1996, pp. 817-825
ERYSODINE, A COMPETITIVE ANTAGONIST AT NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS
Authors: DECKER MW ANDERSON DJ BRIONI JD DONNELLYROBERTS DL KANG CH ONEILL AB PIATTONIKAPLAN M SWANSON S SULLIVAN JP
Citation: Mw. Decker et al., ERYSODINE, A COMPETITIVE ANTAGONIST AT NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS, European journal of pharmacology, 280(1), 1995, pp. 79-89
FUNCTIONAL MODULATION OF HUMAN GANGLIONIC-LIKE NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS (NACHRS) BY L-TYPE CALCIUM-CHANNEL ANTAGONISTS
Authors: DONNELLYROBERTS DL ARNERIC SP SULLIVAN JP
Citation: Dl. Donnellyroberts et al., FUNCTIONAL MODULATION OF HUMAN GANGLIONIC-LIKE NEURONAL NICOTINIC ACETYLCHOLINE-RECEPTORS (NACHRS) BY L-TYPE CALCIUM-CHANNEL ANTAGONISTS, Biochemical and biophysical research communications, 213(2), 1995, pp. 657-662
SODIUM DODECYL SULFATE-INDUCED AND CARBAMYLCHOLINE-INDUCED CHANGES INCIRCULAR-DICHROISM SPECTRA OF ACETYLCHOLINE-RECEPTOR SYNTHETIC PEPTIDES
Authors: DONNELLYROBERTS DL LENTZ TL
Citation: Dl. Donnellyroberts et Tl. Lentz, SODIUM DODECYL SULFATE-INDUCED AND CARBAMYLCHOLINE-INDUCED CHANGES INCIRCULAR-DICHROISM SPECTRA OF ACETYLCHOLINE-RECEPTOR SYNTHETIC PEPTIDES, Molecular brain research, 19(1-2), 1993, pp. 55-61
EFFECTS OF MUTATIONS OF TORPEDO ACETYLCHOLINE-RECEPTOR ALPHA-1 SUBUNIT RESIDUES 184-200 ON ALPHA-BUNGAROTOXIN BINDING IN A RECOMBINANT FUSION PROTEIN
Authors: CHATURVEDI V DONNELLYROBERTS DL LENTZ TL
Citation: V. Chaturvedi et al., EFFECTS OF MUTATIONS OF TORPEDO ACETYLCHOLINE-RECEPTOR ALPHA-1 SUBUNIT RESIDUES 184-200 ON ALPHA-BUNGAROTOXIN BINDING IN A RECOMBINANT FUSION PROTEIN, Biochemistry, 32(37), 1993, pp. 9570-9576
Risultati: 1-13 |