Authors:
AZZOLINA B
ELLSWORTH K
ANDERSSON S
GEISSLER W
BULL HG
HARRIS GS
Citation: B. Azzolina et al., INHIBITION OF RAT ALPHA-REDUCTASES BY FINASTERIDE - EVIDENCE FOR ISOZYME DIFFERENCES IN THE MECHANISM OF INHIBITION, Journal of steroid biochemistry and molecular biology, 61(1-2), 1997, pp. 55-64
Authors:
ELLSWORTH K
AZZOLINA B
BAGINSKY W
BULL H
CHANG B
CIMIS G
MITRA S
TONEY J
BAKSHI RK
RASMUSSON GR
TOLMAN RL
HARRIS GS
Citation: K. Ellsworth et al., MK386 - A POTENT, SELECTIVE INHIBITOR OF THE HUMAN TYPE-1 5-ALPHA-REDUCTASE, Journal of steroid biochemistry and molecular biology, 58(4), 1996, pp. 377-384
Citation: K. Ellsworth et al., EFFECTS OF FINASTERIDE AND DIHYDROFINASTERIDE ON RAT 5-ALPHA-REDUCTASE TYPE-1 AND TYPE-2 IN TRANSFECTED COS CELLS, The FASEB journal, 10(6), 1996, pp. 2211-2211
Authors:
HARRIS GS
ELLSWORTH K
WITZEL BE
TOLMAN RL
Citation: Gs. Harris et al., STEROID 5-ALPHA-REDUCTASE - COMPARATIVE-STUDY OF MECHANISM OF INHIBITION BY NONSTEROIDS ONO-3805 AND LY191704, Bioorganic chemistry, 24(4), 1996, pp. 386-400
Authors:
BAKSHI RK
RASMUSSON GH
PATEL GF
MOSLEY RT
CHANG B
ELLSWORTH K
HARRIS GS
TOLMAN RL
Citation: Rk. Bakshi et al., O-5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYLCARBOXAMIDES AS DUAL INHIBITORSOF HUMAN TYPE-1 AND TYPE-2 STEROID 5-ALPHA-REDUCTASES - DRAMATIC EFFECT OF N-ARYL SUBSTITUENTS ON TYPE-1 AND TYPE-2 5-ALPHA-REDUCTASE INHIBITORY POTENCY (VOL 38, PG 3190, 1995), Journal of medicinal chemistry, 39(5), 1996, pp. 1192-1192
Authors:
TOLMAN RL
ASTER S
BAKSHI RK
BERGMAN JP
BULL HG
CHANG B
CIMIS G
DOLENGA MP
DURETTE P
ELLSWORTH K
ESSER C
GRAHAM DW
HAGMANN WK
HARRIS G
KOPKA I
LANZA T
PATEL G
POLO S
RASMUSSON GH
SAHOO S
TONEY JH
VONLANGEN D
WITZEL B
Citation: Rl. Tolman et al., 4-AZASTEROIDS AS 5-ALPHA-REDUCTASE INHIBITORS - IDENTIFICATION OF 4,7-BETA-DIMETHYL-4-AZA-5-ALPHA-CHOLESTAN-3-ONE (MK-386) AS A SCALP ISOZYME-SELECTIVE INHIBITOR, European journal of medicinal chemistry, 30, 1995, pp. 311-316
Authors:
BAKSHI RK
RASMUSSON GH
PATEL GF
MOSLEY RT
CHANG B
ELLSWORTH K
HARRIS GS
TOLMAN RL
Citation: Rk. Bakshi et al., -5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYL-CARBOXAMIDES AS DUAL INHIBITORSOF HUMAN TYPE-1 AND TYPE-2 STEROID 5-ALPHA-REDUCTASES - DRAMATIC EFFECT OF N-ARYL SUBSTITUENTS ON TYPE-1 AND TYPE-2 5-ALPHA-REDUCTASE INHIBITORY POTENCY, Journal of medicinal chemistry, 38(17), 1995, pp. 3189-3192
Citation: K. Ellsworth et G. Harris, EXPRESSION OF THE TYPE-1 AND TYPE-2 STEROID 5-ALPHA-REDUCTASES IN HUMAN FETAL TISSUES, Biochemical and biophysical research communications, 215(2), 1995, pp. 774-780
Authors:
BAKSHI RK
PATEL GF
RASMUSSON GH
BAGINSKY WF
CIMIS G
ELLSWORTH K
CHANG B
BULL H
TOLMAN RL
HARRIS GS
Citation: Rk. Bakshi et al., 4,7-BETA-DIMETHYL-4-AZACHOLESTAN-3-ONE (MK-386) AND RELATED 4-AZASTEROIDS AS SELECTIVE INHIBITORS OF HUMAN TYPE-1 5-ALPHA-REDUCTASE, Journal of medicinal chemistry, 37(23), 1994, pp. 3871-3874
Citation: K. Ellsworth et G. Harris, EXPRESSION OF THE TYPE-1 AND TYPE-2 5-ALPHA-REDUCTASES IN HUMAN FETALTISSUE, Journal of investigative dermatology, 102(4), 1994, pp. 608-608