Citation: Mr. Reddy et al., RAPID ESTIMATION OF RELATIVE BINDING AFFINITIES OF ENZYME-INHIBITORS, Perspectives in drug discovery and design, 9-11, 1998, pp. 85-98
Authors:
REDDY MR
ERION MD
AGARWAL A
VISWANADHAN VN
MCDONALD DQ
STILL WC
Citation: Mr. Reddy et al., SOLVATION FREE-ENERGIES CALCULATED USING THE GB SA MODEL - SENSITIVITY OF RESULTS ON CHARGE SETS, PROTOCOLS, AND FORCE-FIELDS/, Journal of computational chemistry, 19(7), 1998, pp. 769-780
Citation: Md. Erion et Mr. Reddy, CALCULATION OF RELATIVE HYDRATION FREE-ENERGY DIFFERENCES FOR HETEROAROMATIC-COMPOUNDS - USE IN THE DESIGN OF ADENOSINE-DEAMINASE AND CYTIDINE DEAMINASE INHIBITORS, Journal of the American Chemical Society, 120(14), 1998, pp. 3295-3304
Authors:
ERION MD
UGARKAR BG
DARE J
CASTELLINO AJ
FUJITAKI JM
DIXON R
APPLEMAN JR
WIESNER JB
Citation: Md. Erion et al., DESIGN, SYNTHESIS AND ANTICONVULSANT ACTIVITY OF THE POTENT ADENOSINEKINASE INHIBITOR GP3269, Nucleosides & nucleotides, 16(7-9), 1997, pp. 1013-1021
Citation: Md. Erion et Rm. Rydzewski, AMOYL-3(5)-(2-DEOXY-BETA-D-RIBOFURANOSYL)PYRAZOLES - APPLICATION OF PALLADIUM-CATALYZED GLYCAL COUPLING METHODOLOGY TO THE SYNTHESIS OF PYRAZOFURIN ANALOGS, Nucleosides & nucleotides, 16(3), 1997, pp. 315-337
Authors:
JENG AY
FUJIMOTO RA
CHOU M
TAN J
ERION MD
Citation: Ay. Jeng et al., SUPPRESSION OF SUBSTANCE-P BIOSYNTHESIS IN SENSORY NEURONS OF DORSAL-ROOT GANGLION BY PRODRUG ESTERS OF POTENT PEPTIDYLGLYCINE ALPHA-AMIDATING MONOOXYGENASE INHIBITORS, The Journal of biological chemistry, 272(23), 1997, pp. 14666-14671
Authors:
STOECKLER JD
POIROT AF
SMITH RM
PARKS RE
EALICK SE
TAKABAYASHI K
ERION MD
Citation: Jd. Stoeckler et al., PURINE NUCLEOSIDE PHOSPHORYLASE .3. REVERSAL OF PURINE BASE SPECIFICITY BY SITE-DIRECTED MUTAGENESIS, Biochemistry, 36(39), 1997, pp. 11749-11756
Citation: Q. Dang et al., 5-AMINOPYRAZOLES AS DIENOPHILES IN THE INVERSE ELECTRON DEMAND DIELS-ALDER REACTIONS OF 2,4,6-TRIS(ETHOXY-CARBONYL)-1,3,5-TRIAZINE - SYNTHESES OF PYRAZOLOPYRIMIDINES, Journal of organic chemistry, 61(16), 1996, pp. 5204-5205
Authors:
WONG M
TAN J
FUJIMOTO RA
ERION MD
JENG AY
Citation: M. Wong et al., SUPPRESSION OF SUBSTANCE-P BIOSYNTHESIS IN SENSORY NEURONS OF DORSAL-ROOT GANGLIA BY PROESTERS OF A POTENT PEPTIDYLGLYCINE ALPHA-AMIDATING MONOOXYGENASE INHIBITOR, The FASEB journal, 9(6), 1995, pp. 1491-1491
Citation: Md. Erion et Mr. Reddy, CALCULATION OF RELATIVE FREE-ENERGY DIFFERENCES FOR THE COVALENT HYDRATION OF ORGANIC-COMPOUNDS - A COMBINED QUANTUM-MECHANICAL AND FREE-ENERGY PERTURBATION STUDY, Journal of computational chemistry, 16(12), 1995, pp. 1513-1521
Authors:
FIRESTEIN GS
BULLOUGH DA
ERION MD
JIMENEZ R
RAMIREZWEINHOUSE M
BARANKIEWICZ J
SMITH CW
GRUBER HE
MULLANE KM
Citation: Gs. Firestein et al., INHIBITION OF NEUTROPHIL ADHESION BY ADENOSINE AND AN ADENOSINE KINASE INHIBITOR - THE ROLE OF SELECTINS, The Journal of immunology, 154(1), 1995, pp. 326-334
Authors:
WALTER RL
SYMERSKY J
POIROT AF
STOECKLER JD
ERION MD
EALICK SE
Citation: Rl. Walter et al., X-RAY CRYSTALLOGRAPHIC AND KINETIC-ANALYSIS OF HUMAN PURINE NUCLEOSIDE PHOSPHORYLASE COMPLEXES WITH -BETA-D-RIBOFURANOSYL-1,2,4-TRIAZOLE-3-CARBOXAMIDE AND ETA-D-RIBOFURANOSYL-1,2,4-TRIAZOLE-3-CARBOXAMIDINE, Nucleosides & nucleotides, 13(1-3), 1994, pp. 689
Authors:
TRAPANI AJ
BELL ME
COTE DT
DELOMBAERT S
ERION MD
GERLOCK TE
GHAI RD
HOPKINS MF
PEPPARD JV
WEBB RL
LAPPE RW
WORCEL M
Citation: Aj. Trapani et al., PHARMACOLOGICAL PROFILE OF CGS-24128, A POTENT, LONG-ACTING INHIBITOROF NEUTRAL ENDOPEPTIDASE-24.11, Journal of cardiovascular pharmacology, 23(3), 1994, pp. 358-364
Authors:
GUIDA WC
ELLIOTT RD
THOMAS HJ
SECRIST JA
BABU YS
BUGG CE
ERION MD
EALICK SE
MONTGOMERY JA
Citation: Wc. Guida et al., STRUCTURE-BASED DESIGN OF INHIBITORS OF PURINE NUCLEOSIDE PHOSPHORYLASE .4. A STUDY OF PHOSPHATE MIMICS, Journal of medicinal chemistry, 37(8), 1994, pp. 1109-1114
Authors:
ERION MD
NIWAS S
ROSE JD
ANANTHAN S
ALLEN M
SECRIST JA
BABU YS
BUGG CE
GUIDA WC
EALICK SE
MONTGOMERY JA
Citation: Md. Erion et al., STRUCTURE-BASED DESIGN OF INHIBITORS OF PURINE NUCLEOSIDE PHOSPHORYLASE .3. 9-ARYLMETHYL DERIVATIVES OF 9-DEAZAGUANINE SUBSTITUTED ON THE METHYLENE GROUP (VOL 36, PG 3773, 1993), Journal of medicinal chemistry, 37(7), 1994, pp. 1034-1034
Authors:
DELOMBAERT S
ERION MD
TAN J
BLANCHARD L
ELCHEHABI L
GHAI RD
SAKANE Y
BERRY C
TRAPANI AJ
Citation: S. Delombaert et al., N-PHOSPHONOMETHYL DIPEPTIDES AND THEIR PHOSPHONATE PRODRUGS, A NEW-GENERATION OF NEUTRAL ENDOPEPTIDASE (NEP,EC-3.4.24.11) INHIBITORS, Journal of medicinal chemistry, 37(4), 1994, pp. 498-511