Authors:
DESCHAMPS JR
GEORGE C
FLIPPENANDERSON JL
DEMILO AB
BORDAS B
Citation: Jr. Deschamps et al., X-RAY CRYSTALLOGRAPHIC AND MOLECULAR MODELING STUDIES OF 1-(2,6-DIFLUOROBENZOYL)-5-(4-CHLOROPHENYL)BIURET, Journal of chemical crystallography, 28(6), 1998, pp. 453-459
Authors:
THOMAS JB
ZHENG XL
MASCARELLA SW
ROTHMAN RB
DERSCH CM
PARTILLA JS
FLIPPENANDERSON JL
GEORGE CF
CANTRELL BE
ZIMMERMAN DM
CARROLL FI
Citation: Jb. Thomas et al., N-SUBSTITUTED 9-BETA-METHYL-5-(3-HYDROXYPHENYL)MORPHANS ARE OPIOID RECEPTOR PURE ANTAGONISTS, Journal of medicinal chemistry, 41(21), 1998, pp. 4143-4149
Authors:
KOZIKOWSKI AP
ARALDI GL
BOJA J
MEIL WM
JOHNSON KM
FLIPPENANDERSON JL
GEORGE C
SAIAH E
Citation: Ap. Kozikowski et al., CHEMISTRY AND PHARMACOLOGY OF THE PIPERIDINE-BASED ANALOGS OF COCAINE- IDENTIFICATION OF POTENT DAT INHIBITORS LACKING THE TROPANE SKELETON, Journal of medicinal chemistry, 41(11), 1998, pp. 1962-1969
Authors:
SMITH MP
JOHNSON KM
ZHANG M
FLIPPENANDERSON JL
KOZIKOWSKI AP
Citation: Mp. Smith et al., TUNING THE SELECTIVITY OF MONOAMINE TRANSPORTER INHIBITORS BY THE STEREOCHEMISTRY OF THE NITROGEN LONE-PAIR, Journal of the American Chemical Society, 120(35), 1998, pp. 9072-9073
Authors:
FLIPPENANDERSON JL
DESCHAMPS JR
GEORGE C
REDDY PA
LEWIN AH
BRINE GA
SHELDRICK G
NIKIFOROVICH G
Citation: Jl. Flippenanderson et al., X-RAY STRUCTURE OF TYR-D-TIC-PHE-PHE-NH2 (D-TIPP-NH2), A HIGHLY POTENT MU-RECEPTOR SELECTIVE OPIOID AGONIST, The journal of peptide research, 49(5), 1997, pp. 384-393
Authors:
CALDERON SN
RICE KC
ROTHMAN RB
PORRECA F
FLIPPENANDERSON JL
KAYAKIRI H
XU H
BECKETTS K
SMITH LE
BILSKY EJ
DAVIS P
HORVATH R
Citation: Sn. Calderon et al., PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .23. SYNTHESIS, OPIOID RECEPTOR-BINDING, AND BIOASSAY OF THE HIGHLY SELECTIVE DELTA-AGONISTPIPERAZINYL)-3-METHOXYBENZYL]-N,N-DIETHYLBENZAMIDE (SNC-80) AND RELATED NOVEL NONPEPTIDE DELTA-OPIOID RECEPTOR LIGANDS()), Journal of medicinal chemistry, 40(5), 1997, pp. 695-704
Authors:
KATSURA Y
ZHANG XY
HOMMA K
RICE KC
CALDERON SN
ROTHMAN RB
YAMAMURA HI
DAVIS P
FLIPPENANDERSON JL
XU H
BECKETTS K
FOLTZ EJ
PORRECA F
Citation: Y. Katsura et al., PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .25. SYNTHESIS AND EVALUATION OF N-ALKYL-SUBSTITUTED (ALPHA-PIPERAZINYLBENZYL)BENZAMIDES ASNOVEL, HIGHLY SELECTIVE DELTA-OPIOID RECEPTOR AGONISTS, Journal of medicinal chemistry, 40(18), 1997, pp. 2936-2947
Authors:
KAYAKIRI H
JACOBSON AE
RICE KC
ROTHMAN RB
XU H
FLIPPENANDERSON JL
GEORGE C
ACETO MD
BOWMAN ER
HARRIS LS
MAY EL
PARTILLA JS
BECKETTS K
Citation: H. Kayakiri et al., PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .24. SYNTHESIS, SINGLE-CRYSTAL X-RAY ANALYSES, IN-VITRO AND IN-VIVO PROPERTIES OF -3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN AND -3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN, Medicinal chemistry research, 6(6), 1996, pp. 427-438
Authors:
GEORGE C
FLIPPENANDERSON JL
BIANCO A
CRISMA M
FORMAGGIO F
TONIOLO C
Citation: C. George et al., CRYSTALLOGRAPHIC CHARACTERIZATION OF TRYPTOPHAN-CONTAINING PEPTIDE 3(10)-HELICES, Peptide research, 9(6), 1996, pp. 315-321
Authors:
FLIPPENANDERSON JL
GEORGE C
VALLE G
VALENTE E
BIANCO A
FORMAGGIO F
CRISMA M
TONIOLO C
Citation: Jl. Flippenanderson et al., CRYSTALLOGRAPHIC CHARACTERIZATION OF GEOMETRY AND CONFORMATION OF TOAC, A NITROXIDE SPIN-LABELED C-ALPHA,C-ALPHA-DISUBSTITUTED GLYCINE, IN SIMPLE DERIVATIVES AND MODEL PEPTIDES, International journal of peptide & protein research, 47(4), 1996, pp. 231-238
Citation: Jr. Deschamps et al., A DIACETYLMORPHINE POLYMORPH, Acta crystallographica. Section C, Crystal structure communications, 52, 1996, pp. 698-700
Authors:
YAMADA K
RICE KC
FLIPPENANDERSON JL
EISSENSTAT MA
WARD SJ
JOHNSON MR
HOWLETT AC
Citation: K. Yamada et al., (AMINOALKYL)INDOLE ISOTHIOCYANATES AS POTENTIAL ELECTROPHILIC AFFINITY LIGANDS FOR THE BRAIN CANNABINOID RECEPTOR, Journal of medicinal chemistry, 39(10), 1996, pp. 1967-1974
Authors:
BERTHA CM
ELLIS M
FLIPPENANDERSON JL
PORRECA F
ROTHMAN RB
DAVIS P
XU H
BECKETTS K
RICE KC
Citation: Cm. Bertha et al., PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .21. NOVEL DERIVATIVES OF L-2,6-METHANO-6H-AZOCINO[4,5-B]INDOL-6-YL)-PHENOLS WITH IMPROVED DELTA-OPIOID RECEPTOR SELECTIVITY, Journal of medicinal chemistry, 39(10), 1996, pp. 2081-2086
Citation: Jr. Deschamps et al., STRUCTURAL STUDIES OF OPIOID-PEPTIDES - A REVIEW OF RECENT PROGRESS IN X-RAY-DIFFRACTION STUDIES, Biopolymers, 40(1), 1996, pp. 121-139
Authors:
COLLINS N
FLIPPENANDERSON JL
HAASETH RC
DESCHAMPS JR
GEORGE C
KOVER R
HRUBY VJ
Citation: N. Collins et al., CONFORMATIONAL DETERMINANTS OF AGONIST VERSUS ANTAGONIST PROPERTIES OF [D-PEN(2),D-PEN(5)]ENKEPHALIN (DPDPE) ANALOGS AT OPIOID RECEPTORS - COMPARISON OF X-RAY CRYSTALLOGRAPHIC STRUCTURE, SOLUTION H-1-NMR DATA,AND MOLECULAR DYNAMIC SIMULATIONS OF [L-ALA(3)]DPDPE AND [D-ALA(3)]DPDPE, Journal of the American Chemical Society, 118(9), 1996, pp. 2143-2152
Authors:
NIKIFOROVICH GV
KOVER KE
KOLODZIEJ SA
NOCK B
GEORGE C
DESCHAMPS JR
FLIPPENANDERSON JL
MARSHALL GR
Citation: Gv. Nikiforovich et al., DESIGN AND COMPREHENSIVE CONFORMATIONAL STUDIES OF TYR(1)-CYCLO(D-PEN(2)-GLY(3)-PHE(4)-L-3-MPT(5)) AND TYR(1)-CYCLO(D-PEN(2)-GLY(3)-PHE(4)-D-3-MPT(5)) - NOVEL CONFORMATIONALLY CONSTRAINED OPIOID-PEPTIDES, Journal of the American Chemical Society, 118(5), 1996, pp. 959-969
Authors:
BERTHA CM
FLIPPENANDERSON JL
ROTHMAN RB
PORRECA F
DAVIS P
XU H
BECKETTS K
CHA XY
RICE KC
Citation: Cm. Bertha et al., PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .20. ALTERATION OF OPIOID RECEPTOR SUBTYPE SELECTIVITY OF THE 5-(3-HYDROXYPHENYL)MORPHANS BY APPLICATION OF THE MESSAGE-ADDRESS CONCEPT - PREPARATION OF DELTA-OPIOID RECEPTOR LIGANDS, Journal of medicinal chemistry, 38(9), 1995, pp. 1523-1537
Authors:
BERTHA CM
VILNER BJ
MATTSON MV
BOWEN WD
BECKETTS K
XU H
ROTHMAN RB
FLIPPENANDERSON JL
RICE KC
Citation: Cm. Bertha et al., (E)-8-BENZYLIDENE DERIVATIVES OF 2-METHYL-5-(3-HYDROXYPHENYL)MORPHANS- HIGHLY SELECTIVE LIGANDS FOR THE SIGMA(2) RECEPTOR SUBTYPE, Journal of medicinal chemistry, 38(24), 1995, pp. 4776-4785
Authors:
LEI PS
OGAWA Y
FLIPPENANDERSON JL
KOVAC P
Citation: Ps. Lei et al., SYNTHESIS AND CRYSTAL-STRUCTURE OF METHYL O-TETRONAMIDO)-2-O-METHYL-ALPHA-D-MANNOPYRANOSIDE, THE METHYL ALPHA-GLYCOSIDE OF THE TERMINAL UNIT, AND PRESUMED ANTIGENIC DETERMINANT, OF THE O-SPECIFIC POLYSACCHARIDE OF VIBRIO-CHOLERAE O 1, SEROTYPE OGAWA/, Carbohydrate research, 275(1), 1995, pp. 117-129
Authors:
KARLE IL
FLIPPENANDERSON JL
GURUNATH R
BALARAM P
Citation: Il. Karle et al., FACILE TRANSITION BETWEEN 3(10)-HELIX AND ALPHA-HELIX - STRUCTURES OF8-RESIDUE, 9-RESIDUE, AND 10-RESIDUE PEPTIDES CONTAINING THE -(LEU-AIB-ALA)(2)-PHE-AIB- FRAGMENT, Protein science, 3(9), 1994, pp. 1547-1555