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Results: 1-18 |
Results: 18
(4-METHYL-PIPERIDIN-1-YL)PROPYL]BENZENESULFONAMIDE - THE FIRST SELECTIVE 5-HT7 RECEPTOR ANTAGONIST
Authors: FORBES IT DABBS S DUCKWORTH DM JENNINGS AJ KING FD LOVELL PJ BROWN AM COLLIN L HAGAN JJ MIDDLEMISS DN RILEY GJ THOMAS DR UPTON N
Citation: It. Forbes et al., (4-METHYL-PIPERIDIN-1-YL)PROPYL]BENZENESULFONAMIDE - THE FIRST SELECTIVE 5-HT7 RECEPTOR ANTAGONIST, Journal of medicinal chemistry, 41(5), 1998, pp. 655-657
NOVEL AND SELECTIVE 5-HT2C 2B RECEPTOR ANTAGONISTS AS POTENTIAL ANXIOLYTIC AGENTS - SYNTHESIS, QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS, AND MOLECULAR MODELING OF SUBSTITUTED 1-(3-PYRIDYLCARBAMOYL)INDOLINES/
Authors: BROMIDGE SM DABBS S DAVIES DT DUCKWORTH DM FORBES IT HAM P JONES GE KING FD SAUNDERS DV STARR S THEWLIS KM WYMAN PA BLANEY FE NAYLOR CB BAILEY F BLACKBURN TP HOLLAND V KENNETT GA RILEY GJ WOOD MD
Citation: Sm. Bromidge et al., NOVEL AND SELECTIVE 5-HT2C 2B RECEPTOR ANTAGONISTS AS POTENTIAL ANXIOLYTIC AGENTS - SYNTHESIS, QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS, AND MOLECULAR MODELING OF SUBSTITUTED 1-(3-PYRIDYLCARBAMOYL)INDOLINES/, Journal of medicinal chemistry, 41(10), 1998, pp. 1598-1612
FUNCTIONAL-CHARACTERIZATION OF THE HUMAN CLONED 5-HT7 RECEPTOR (LONG FORM) - ANTAGONIST PROFILE OF SB-258719
Authors: THOMAS DR GITTINS SA COLLIN LL MIDDLEMISS DN RILEY G HAGAN J GLOGER I ELLIS CE FORBES IT BROWN AM
Citation: Dr. Thomas et al., FUNCTIONAL-CHARACTERIZATION OF THE HUMAN CLONED 5-HT7 RECEPTOR (LONG FORM) - ANTAGONIST PROFILE OF SB-258719, British Journal of Pharmacology, 124(6), 1998, pp. 1300-1306
SB-242084, A SELECTIVE AND BRAIN PENETRANT 5-HT2C RECEPTOR ANTAGONIST
Authors: KENNETT GA WOOD MD BRIGHT F TRAIL B RILEY G HOLLAND V AVENELL KY STEAN T UPTON N BROMIDGE S FORBES IT BROWN AM MIDDLEMISS DN BLACKBURN TP
Citation: Ga. Kennett et al., SB-242084, A SELECTIVE AND BRAIN PENETRANT 5-HT2C RECEPTOR ANTAGONIST, Neuropharmacology, 36(4-5), 1997, pp. 609-620
ETHYL-3-PYRIDYL)OXY]-5-PYRIDYL]CARBAMOYL]-INDOLINE (SB-242084) - THE FIRST SELECTIVE AND BRAIN PENETRANT 5-HT2C RECEPTOR ANTAGONIST
Authors: BROMIDGE SM DUCKWORTH M FORBES IT HAM P KING FD THEWLIS KM BLANEY FE NAYLOR CB BLACKBURN TP KENNETT GA WOOD MD CLARKE SE
Citation: Sm. Bromidge et al., ETHYL-3-PYRIDYL)OXY]-5-PYRIDYL]CARBAMOYL]-INDOLINE (SB-242084) - THE FIRST SELECTIVE AND BRAIN PENETRANT 5-HT2C RECEPTOR ANTAGONIST, Journal of medicinal chemistry, 40(22), 1997, pp. 3494-3496
N-ALKENYL NITRONE DIPOLAR CYCLOADDITION ROUTES TO PIPERIDINES AND INDOLIZIDINES .8. THE SCOPE OF TANDEM REACTIONS INVOLVING HYDROXYLAMINE-ALKYNE CYCLIZATIONS
Authors: DAVISON EC FORBES IT HOLMES AB WARNER JA
Citation: Ec. Davison et al., N-ALKENYL NITRONE DIPOLAR CYCLOADDITION ROUTES TO PIPERIDINES AND INDOLIZIDINES .8. THE SCOPE OF TANDEM REACTIONS INVOLVING HYDROXYLAMINE-ALKYNE CYCLIZATIONS, Tetrahedron, 52(35), 1996, pp. 11601-11624
A SYNTHESIS OF NOVEL IH-IMIDAZO[1,2-ALPHA]INDOLE-3-CARBOXYLATES
Authors: FORBES IT MORGAN HKA THOMPSON M
Citation: It. Forbes et al., A SYNTHESIS OF NOVEL IH-IMIDAZO[1,2-ALPHA]INDOLE-3-CARBOXYLATES, Synthetic communications, 26(4), 1996, pp. 745-754
SYNTHESIS, BIOLOGICAL-ACTIVITY, AND MOLECULAR MODELING STUDIES OF SELECTIVE 5-HT2C 2B RECEPTOR ANTAGONISTS/
Authors: FORBES IT DABBS S DUCKWORTH DM HAM P JONES GE KING FD SAUNDERS DV BLANEY FE NAYLOR CB BAXTER GS BLACKBURN TP KENNETT GA WOOD MD
Citation: It. Forbes et al., SYNTHESIS, BIOLOGICAL-ACTIVITY, AND MOLECULAR MODELING STUDIES OF SELECTIVE 5-HT2C 2B RECEPTOR ANTAGONISTS/, Journal of medicinal chemistry, 39(25), 1996, pp. 4966-4977
IN-VITRO AND IN-VIVO PROFILE OF SB-206553, A POTENT 5-HT2C 5-HT2B RECEPTOR ANTAGONIST WITH ANXIOLYTIC-LIKE PROPERTIES/
Authors: KENNETT GA WOOD MD BRIGHT F CILIA J PIPER DC GAGER T THOMAS D BAXTER GS FORBES IT HAM P BLACKBURN TP
Citation: Ga. Kennett et al., IN-VITRO AND IN-VIVO PROFILE OF SB-206553, A POTENT 5-HT2C 5-HT2B RECEPTOR ANTAGONIST WITH ANXIOLYTIC-LIKE PROPERTIES/, British Journal of Pharmacology, 117(3), 1996, pp. 427-434
ISOSTERIC REPLACEMENT OF THE INDOLE NUCLEUS BY BENZOTHIOPHENE IN A SERIES OF PYRIDO[2,3-B]INDOLES WITH POTENTIAL ANXIOLYTIC ACTIVITY
Authors: BLACKBURN TP DAVIES DT FORBES IT HAYWARD CJ JOHNSON CN MARTIN RT PIPER DC THOMAS DR THOMPSON M UPTON N WARD RW
Citation: Tp. Blackburn et al., ISOSTERIC REPLACEMENT OF THE INDOLE NUCLEUS BY BENZOTHIOPHENE IN A SERIES OF PYRIDO[2,3-B]INDOLES WITH POTENTIAL ANXIOLYTIC ACTIVITY, Bioorganic & medicinal chemistry letters, 5(22), 1995, pp. 2589-2592
A TANDEM SYNTHESIS OF (+ -)-EUPHOCOCCININE AND (+/-)-ADALINE/
Authors: DAVISON EC HOLMES AB FORBES IT
Citation: Ec. Davison et al., A TANDEM SYNTHESIS OF (+ -)-EUPHOCOCCININE AND (+/-)-ADALINE/, Tetrahedron letters, 36(49), 1995, pp. 9047-9050
METHYL-5-INDOLYL)-N'-(3-METHYL-5-ISOTHIAZOLYL)UREA - A NOVEL, HIGH-AFFINITY 5-HT2B RECEPTOR ANTAGONIST
Authors: FORBES IT JONES GE MURPHY OE HOLLAND V BAXTER GS
Citation: It. Forbes et al., METHYL-5-INDOLYL)-N'-(3-METHYL-5-ISOTHIAZOLYL)UREA - A NOVEL, HIGH-AFFINITY 5-HT2B RECEPTOR ANTAGONIST, Journal of medicinal chemistry, 38(6), 1995, pp. 855-857
LCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO[2,3-F]INDOLE - A NOVEL 5-HT2C 5-HT2B RECEPTOR ANTAGONIST WITH IMPROVED AFFINITY, SELECTIVITY, AND ORAL ACTIVITY
Authors: FORBES IT HAM P BOOTH DH MARTIN RT THOMPSON M BAXTER GS BLACKBURN TP GLEN A KENNETT GA WOOD MD
Citation: It. Forbes et al., LCARBAMOYL)-1,2,3,5-TETRAHYDROPYRROLO[2,3-F]INDOLE - A NOVEL 5-HT2C 5-HT2B RECEPTOR ANTAGONIST WITH IMPROVED AFFINITY, SELECTIVITY, AND ORAL ACTIVITY, Journal of medicinal chemistry, 38(14), 1995, pp. 2524-2530
SB-204741 - A POTENT AND SELECTIVE ANTAGONIST AT 5-HT(2B) RECEPTORS
Authors: BAXTER GS ELLIS ES FORBES IT JONES GE KENNETT GA
Citation: Gs. Baxter et al., SB-204741 - A POTENT AND SELECTIVE ANTAGONIST AT 5-HT(2B) RECEPTORS, British Journal of Pharmacology, 114, 1995, pp. 157-157
-DIMETHYL-1,2,3,4-TETRAHYDRO-6H-QUININDOLIN-1-ONE, A NOVEL GABA(A) MODULATOR WITH POTENTIAL ANXIOLYTIC ACTIVITY
Authors: BLACKBURN TP BOLTON D FORBES IT JOHNSON CN MARTIN RT THOMAS DR THOMPSON M UPTON N
Citation: Tp. Blackburn et al., -DIMETHYL-1,2,3,4-TETRAHYDRO-6H-QUININDOLIN-1-ONE, A NOVEL GABA(A) MODULATOR WITH POTENTIAL ANXIOLYTIC ACTIVITY, Bioorganic & medicinal chemistry letters, 4(2), 1994, pp. 279-284
N-ALKENYL NITRONE DIPOLAR CYCLOADDITION ROUTES TO PIPERIDINES AND INDOLIZIDINES .7. HYDROXYLAMINE ALKYNE CYCLIZATIONS - FORMATION OF CYCLICNITRONES AND APPLICATION TO THE SYNTHESIS OF THE PROPOSED STRUCTURE FOR (+ -)-ACACIALACTAM/
Authors: FOX ME HOLMES AB FORBES IT THOMPSON M
Citation: Me. Fox et al., N-ALKENYL NITRONE DIPOLAR CYCLOADDITION ROUTES TO PIPERIDINES AND INDOLIZIDINES .7. HYDROXYLAMINE ALKYNE CYCLIZATIONS - FORMATION OF CYCLICNITRONES AND APPLICATION TO THE SYNTHESIS OF THE PROPOSED STRUCTURE FOR (+ -)-ACACIALACTAM/, Journal of the Chemical Society. Perkin transactions. I, (23), 1994, pp. 3379-3395
SYNTHESIS AND POTENTIAL ANXIOLYTIC ACTIVITY OF 4-AMINO-PYRIDO[2,3-B]INDOLES
Authors: BOLTON D FORBES IT HAYWARD CJ PIPER DC THOMAS DR THOMPSON M UPTON N
Citation: D. Bolton et al., SYNTHESIS AND POTENTIAL ANXIOLYTIC ACTIVITY OF 4-AMINO-PYRIDO[2,3-B]INDOLES, Bioorganic & medicinal chemistry letters, 3(10), 1993, pp. 1941-1946
N-(1-METHYL-5-INDOLYL)-N'-(3-PYRIDYL)UREA HYDROCHLORIDE - THE 1ST SELECTIVE 5-HT(1C) RECEPTOR ANTAGONIST
Authors: FORBES IT KENNETT GA GADRE A HAM P HAYWARD CJ MARTIN RT THOMPSON M WOOD MD BAXTER GS GLEN A MURPHY OE STEWART BA BLACKBURN TP
Citation: It. Forbes et al., N-(1-METHYL-5-INDOLYL)-N'-(3-PYRIDYL)UREA HYDROCHLORIDE - THE 1ST SELECTIVE 5-HT(1C) RECEPTOR ANTAGONIST, Journal of medicinal chemistry, 36(8), 1993, pp. 1104-1107
Risultati: 1-18 |