Authors:
GALANAKIS D
CALDER JAD
GANELLIN CR
OWEN CS
DUNN PM
Citation: D. Galanakis et al., SYNTHESIS AND QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS OF DEQUALINIUM ANALOGS AS K- INVESTIGATION INTO THE ROLE OF THE SUBSTITUENT AT POSITION-4 OF THE QUINOLINE RING( CHANNEL BLOCKERS ), Journal of medicinal chemistry, 38(18), 1995, pp. 3536-3546
Authors:
GANELLIN CR
HOSSEINI SK
KHALAF YS
TERTIUK W
ARRANG JM
GARBARG M
LIGNEAU X
SCHWARTZ JC
Citation: Cr. Ganellin et al., DESIGN OF POTENT NON-THIOUREA H-3 RECEPTOR HISTAMINE-ANTAGONISTS, Journal of medicinal chemistry, 38(17), 1995, pp. 3342-3350
Authors:
BANNISTER C
BURNS K
PROUT K
WATKIN DJ
COOPER DG
DURANT GJ
GANELLIN CR
IFE RJ
SACH GS
Citation: C. Bannister et al., STRUCTURES OF HISTAMINE H1-RECEPTOR ANTAGONISTS DERIVED FROM THE CIMETIDINE GROUP OF HISTAMINE-H2-RECEPTOR ANTAGONISTS, Acta crystallographica. Section B, Structural science, 50, 1994, pp. 221-243
Authors:
PARSONS ME
OWEN DAA
GANELLIN CR
DURANT GJ
Citation: Me. Parsons et al., DIMAPRIT - [S-[3-(N,N-DIMETHYLAMINO)PROPYL]ISOTHIOUREA] - A HIGHLY SPECIFIC HISTAMINE H-2-RECEPTOR AGONIST .1. PHARMACOLOGY, Agents and actions, 43(3-4), 1994, pp. 132-138
Citation: Gj. Durant et al., DIMAPRIT, [S-[3-(N,N-DIMETHYLAMINO)PROPYL]ISOTHIOUREA] - A HIGHLY SPECIFIC HISTAMINE H-2-RECEPTOR AGONIST .2. STRUCTURE-ACTIVITY CONSIDERATIONS, Agents and actions, 43(3-4), 1994, pp. 139-143
Authors:
DUNN PM
ROSA JC
BECKWITHHALL B
BENTON DC
AYALEW Y
GANELLIN CR
JENKINSON DH
Citation: Pm. Dunn et al., A NOVEL BIS-QUATERNARY CYCLOPHANE, UCL-1530, MAY DISCRIMINATE BETWEENSUBTYPES OF APAMIN-SENSITIVE K+ CHANNELS, British Journal of Pharmacology, 112, 1994, pp. 210000068-210000068
Authors:
BROWN TH
BLAKEMORE RC
DURANT GJ
GANELLIN CR
PARSONS ME
RASMUSSEN AC
RAWLINGS DA
Citation: Th. Brown et al., ISOCYTOSINE H(2)-RECEPTOR HISTAMINE-ANTAGONISTS .4. THE SYNTHESIS ANDBIOLOGICAL-ACTIVITY OF DONETIDINE (SK-AND-F-93574) AND RELATED-COMPOUNDS, European journal of medicinal chemistry, 28(7-8), 1993, pp. 601-608
Authors:
YOUNG RC
GANELLIN CR
GRIFFITHS R
MITCHELL RC
PARSONS ME
SAUNDERS D
SORE NE
Citation: Rc. Young et al., AN APPROACH TO THE DESIGN OF BRAIN-PENETRATING HISTAMINERGIC AGONISTS, European journal of medicinal chemistry, 28(3), 1993, pp. 201-211
Authors:
PROUT K
BURNS K
WATKIN DJ
COOPER DG
DURANT GJ
GANELLIN CR
SACH GS
Citation: K. Prout et al., STRUCTURES OF 9 HISTAMINE-H-2 ANTAGONISTS RELATED TO -CYANO-N'-METHYL-N''-[4-(2-PYRIDYL)BUTYL]GUANIDINE, Acta crystallographica. Section B, Structural science, 49, 1993, pp. 547-559