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Results: 1-25 | 26-27
Results: 1-25/27
Effects of two-carbon bridge region methoxylation of benztropine: Discovery of novel chiral ligands for the dopamine transporter
Authors: Simoni, D Roberti, M Rondanin, R Baruchello, R Rossi, M Invidiata, FP Merighi, S Varani, K Gessi, S Borea, PA Marino, S Cavallini, S Bianchi, C Siniscalchi, A
Citation: D. Simoni et al., Effects of two-carbon bridge region methoxylation of benztropine: Discovery of novel chiral ligands for the dopamine transporter, BIOORG MED, 11(6), 2001, pp. 823-827
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A(2B) adenosine receptor antagonists
Authors: Baraldi, PG Cacciari, B Romagnoli, R Klotz, KN Spalluto, G Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A(2B) adenosine receptor antagonists, DRUG DEV R, 53(2-3), 2001, pp. 225-235
Fluorosulfonyl- and bis-(beta-chloroethyl)amino-phenylamino functionalizedpyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: Irreversible antagonists at the human A(3) adenosine receptor and molecular modeling studies
Authors: Baraldi, PG Cacciari, B Moro, S Romagnoli, R Ji, XD Jacobson, KA Gessi, S Borea, PA Spalluto, G
Citation: Pg. Baraldi et al., Fluorosulfonyl- and bis-(beta-chloroethyl)amino-phenylamino functionalizedpyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: Irreversible antagonists at the human A(3) adenosine receptor and molecular modeling studies, J MED CHEM, 44(17), 2001, pp. 2735-2742
Pharmacological and biochemical characterization of adenosine receptors inthe human malignant melanoma A375 cell line
Authors: Merighi, S Varani, K Gessi, S Cattabriga, E Iannotta, V Ulouglu, C Leung, E Borea, PA
Citation: S. Merighi et al., Pharmacological and biochemical characterization of adenosine receptors inthe human malignant melanoma A375 cell line, BR J PHARM, 134(6), 2001, pp. 1215-1226
Pharmacological and biochemical characterization of A(3) adenosine receptors in Jurkat T cells
Authors: Gessi, S Varani, K Merighi, S Morelli, A Ferrari, D Leung, E Baraldi, PG Spalluto, G Borea, PA
Citation: S. Gessi et al., Pharmacological and biochemical characterization of A(3) adenosine receptors in Jurkat T cells, BR J PHARM, 134(1), 2001, pp. 116-126
Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors
Authors: Baraldi, PG Cacciari, B Romagnoli, R Varani, K Merighi, S Gessi, S Borea, PA Leung, E Hickey, SL Spalluto, G
Citation: Pg. Baraldi et al., Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors, BIOORG MED, 10(3), 2000, pp. 209-211
Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors (vol 10, pg 209, 2000)
Authors: Baraldi, PG Cacciari, B Romagnoli, R Varani, K Merighi, S Gessi, S Borea, PA Leung, E Hickey, SL Spalluto, G
Citation: Pg. Baraldi et al., Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors (vol 10, pg 209, 2000), BIOORG MED, 10(12), 2000, pp. 1403-1403
Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension are normalized after treatment with doxazosin but not propranolol
Authors: Portaluppi, F Manfredini, R Varani, K Gessi, S Caiazza, A Borea, PA
Citation: F. Portaluppi et al., Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension are normalized after treatment with doxazosin but not propranolol, J HYPERTENS, 18(2), 2000, pp. 217-221
[H-3]MRE 3008F20: A novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors
Authors: Varani, K Merighi, S Gessi, S Klotz, KN Leung, E Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Borea, PA
Citation: K. Varani et al., [H-3]MRE 3008F20: A novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors, MOLEC PHARM, 57(5), 2000, pp. 968-975
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: Influence of thechain at the N-8 pyrazole nitrogen
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Moro, S Klotz, KN Leung, E Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: Influence of thechain at the N-8 pyrazole nitrogen, J MED CHEM, 43(25), 2000, pp. 4768-4780
Further studies on nociceptin-related peptides: Discovery of a new chemical template with antagonist activity on the nociceptin receptor
Authors: Guerrini, R Calo, G Bigoni, R Rizzi, A Varani, K Toth, G Gessi, S Hashiba, E Hashimoto, Y Lambert, DG Borea, PA Tomatis, R Salvadori, S Regoli, D
Citation: R. Guerrini et al., Further studies on nociceptin-related peptides: Discovery of a new chemical template with antagonist activity on the nociceptin receptor, J MED CHEM, 43(15), 2000, pp. 2805-2813
Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes
Authors: Vianello, P Albinati, A Pinna, GA Lavecchia, A Marinelli, L Borea, PA Gessi, S Fadda, P Tronci, S Cignarella, G
Citation: P. Vianello et al., Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes, J MED CHEM, 43(11), 2000, pp. 2115-2123
Synthesis, modelling, and mu-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes
Authors: Pinna, GA Murineddu, G Curzu, MM Villa, S Vianello, P Borea, PA Gessi, S Toma, L Colombo, D Cignarella, G
Citation: Ga. Pinna et al., Synthesis, modelling, and mu-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes, FARMACO, 55(8), 2000, pp. 553-562
Dose and time effects of caffeine intake on human platelet adenosine A(2A)receptors - Functional and biochemical aspects
Authors: Varani, K Portaluppi, F Gessi, S Merighi, S Ongini, E Belardinelli, L Borea, PA
Citation: K. Varani et al., Dose and time effects of caffeine intake on human platelet adenosine A(2A)receptors - Functional and biochemical aspects, CIRCULATION, 102(3), 2000, pp. 285-289
A(2A) adenosine receptors in human peripheral blood cells
Authors: Gessi, S Varani, K Merighi, S Ongini, E Borea, PA
Citation: S. Gessi et al., A(2A) adenosine receptors in human peripheral blood cells, BR J PHARM, 129(1), 2000, pp. 2-11
Synthesis and preliminary biological evaluation of novel N-substituted 1-amino-3[1-methyl(phenyl)-1H-indazol-4-yloxy]-propan-2-ols interesting as potential antiarrhythmic, local anaesthetic and analgesic agents
Authors: Mosti, L Menozzi, G Fossa, P Filippelli, W Gessi, S Rinaldi, B Falcone, G
Citation: L. Mosti et al., Synthesis and preliminary biological evaluation of novel N-substituted 1-amino-3[1-methyl(phenyl)-1H-indazol-4-yloxy]-propan-2-ols interesting as potential antiarrhythmic, local anaesthetic and analgesic agents, ARZNEI-FOR, 50(11), 2000, pp. 963-972
Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension
Authors: Varani, K Gessi, S Caiazza, A Rastelli, G Portaluppi, F Borea, PA
Citation: K. Varani et al., Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension, BR J CL PH, 47(2), 1999, pp. 167-172
Changes in hippocampal and cortical B-1 bradykinin receptor biological activity in two experimental models of epilepsy
Authors: Bregola, G Varani, K Gessi, S Beani, L Bianchi, C Borea, PA Regoli, D Simonato, M
Citation: G. Bregola et al., Changes in hippocampal and cortical B-1 bradykinin receptor biological activity in two experimental models of epilepsy, NEUROSCIENC, 92(3), 1999, pp. 1043-1049
4-(4-fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors
Authors: Claudi, F Scoccia, L Giorgioni, G Accorroni, B Marucci, G Gessi, S Siniscalchi, A Borea, PA
Citation: F. Claudi et al., 4-(4-fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors, EUR J MED C, 34(10), 1999, pp. 843-852
Early changes in adenosine A(1) receptors in cerebral cortex slices submitted to in vitro ischemia
Authors: Siniscalchi, A Rodi, D Gessi, S Campi, F Borea, PA
Citation: A. Siniscalchi et al., Early changes in adenosine A(1) receptors in cerebral cortex slices submitted to in vitro ischemia, NEUROCHEM I, 34(6), 1999, pp. 517-522
Pharmacology of [Tyr(1)]nociceptin analogs: receptor binding and bioassay studies
Authors: Varani, K Rizzi, A Calo, G Bigoni, R Toth, G Guerrini, R Gessi, S Salvadori, S Borea, PA Regoli, D
Citation: K. Varani et al., Pharmacology of [Tyr(1)]nociceptin analogs: receptor binding and bioassay studies, N-S ARCH PH, 360(3), 1999, pp. 270-277
Comparison of CGS15943, ZM241385 and SCH58261 as antagonists at human adenosine receptors
Authors: Ongini, E Dionisotti, S Gessi, S Irenius, E Fredholm, BB
Citation: E. Ongini et al., Comparison of CGS15943, ZM241385 and SCH58261 as antagonists at human adenosine receptors, N-S ARCH PH, 359(1), 1999, pp. 7-10
Temperature dependence and GABA modulation of beta-carboline binding to rat cerebellum benzodiazepine receptors
Authors: Gessi, S Dalpiaz, A Varani, K Borea, PA
Citation: S. Gessi et al., Temperature dependence and GABA modulation of beta-carboline binding to rat cerebellum benzodiazepine receptors, LIFE SCI, 64(16), 1999, pp. PL185-PL192
alpha(2)-adrenergic agonist modulation of [S-35]GTP gamma S binding to guanine-nucleotide-binding-proteins in human platelet membranes
Authors: Gessi, S Campi, F Varani, K Borea, PA
Citation: S. Gessi et al., alpha(2)-adrenergic agonist modulation of [S-35]GTP gamma S binding to guanine-nucleotide-binding-proteins in human platelet membranes, LIFE SCI, 64(16), 1999, pp. 1403-1413
Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]-pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Klotz, KN Leung, E Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]-pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists, J MED CHEM, 42(22), 1999, pp. 4473-4478
Risultati: 1-25 | 26-27