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Results: 1-25 | 26-30
Results: 1-25/30
PYRAZOLO[1,5-A]PYRIMIDINE CRF-1 RECEPTOR ANTAGONISTS
Authors: WUSTROW DJ CAPIRIS T RUBIN R KNOBELSDORF JA AKUNNE H DAVIS MD MACKENZIE R PUGSLEY TA ZOSKI KT HEFFNER TG WISE LD
Citation: Dj. Wustrow et al., PYRAZOLO[1,5-A]PYRIMIDINE CRF-1 RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 8(16), 1998, pp. 2067-2070
ISOINDOLINONE ENANTIOMERS HAVING AFFINITY FOR THE DOPAMINE D-4 RECEPTOR
Authors: BELLIOTTI TR BRINK WA KESTEN SR RUBIN JR WUSTROW DJ ZOSKI KT WHETZEL SZ CORBIN AE PUGSLEY TA HEFFNER TG WISE LD
Citation: Tr. Belliotti et al., ISOINDOLINONE ENANTIOMERS HAVING AFFINITY FOR THE DOPAMINE D-4 RECEPTOR, Bioorganic & medicinal chemistry letters, 8(12), 1998, pp. 1499-1502
PHARMACOLOGICAL CHARACTERIZATION OF PD-152255, A NOVEL DIMERIC BENZIMIDAZOLE DOPAMINE D-3 ANTAGONIST
Authors: CORBIN AE PUGSLEY TA AKUNNE HC WHETZEL SZ ZOSKI KT GEORGIC LM NELSON CB WRIGHT JL WISE LD HEFFNER TG
Citation: Ae. Corbin et al., PHARMACOLOGICAL CHARACTERIZATION OF PD-152255, A NOVEL DIMERIC BENZIMIDAZOLE DOPAMINE D-3 ANTAGONIST, Pharmacology, biochemistry and behavior, 59(2), 1998, pp. 487-493
NOVEL SMALL-MOLECULE NEUROTENSIN ANTAGONISTS - 3-(1,5-DIARYL-1,5-DIOXOPENTAN-3-YL)BENZOIC ACIDS
Authors: JOHNSON SJ AKUNNE HC HEFFNER TG KESTEN SR PUGSLEY TA WISE LD WUSTROW DJ
Citation: Sj. Johnson et al., NOVEL SMALL-MOLECULE NEUROTENSIN ANTAGONISTS - 3-(1,5-DIARYL-1,5-DIOXOPENTAN-3-YL)BENZOIC ACIDS, Bioorganic & medicinal chemistry letters, 7(5), 1997, pp. 561-566
DISCOVERY OF SELECTIVE DOPAMINE D4 RECEPTOR ANTAGONISTS - 1-ARYLOXY-3-(4-ARYLOXYPIPERIDINYL)-2-PROPANOLS
Authors: WRIGHT JL GREGORY TF HEFFNER TG MACKENZIE RG PUGSLEY TA MEULEN SV WISE LD
Citation: Jl. Wright et al., DISCOVERY OF SELECTIVE DOPAMINE D4 RECEPTOR ANTAGONISTS - 1-ARYLOXY-3-(4-ARYLOXYPIPERIDINYL)-2-PROPANOLS, Bioorganic & medicinal chemistry letters, 7(11), 1997, pp. 1377-1380
PHARMACOKINETICS AND PHARMACODYNAMICS OF AN INVESTIGATIONAL ANTIPSYCHOTIC AGENT, CI-1007, IN RATS AND MONKEYS
Authors: FENG MR CORBIN AE WANG YF CHRISTOFFERSEN CL WILEY JN STRENKOSKI CA TUCKER EV NINTEMAN FW MELTZER LT HEFFNER TG WRIGHT DS
Citation: Mr. Feng et al., PHARMACOKINETICS AND PHARMACODYNAMICS OF AN INVESTIGATIONAL ANTIPSYCHOTIC AGENT, CI-1007, IN RATS AND MONKEYS, Pharmaceutical research, 14(3), 1997, pp. 329-336
THE PHARMACOLOGY OF THE NOVEL AND SELECTIVE SIGMA-LIGAND, PD-144418
Authors: AKUNNE HC WHETZEL SZ WILEY JN CORBIN AE NINTEMAN FW TECLE H PEI Y PUGSLEY TA HEFFNER TG
Citation: Hc. Akunne et al., THE PHARMACOLOGY OF THE NOVEL AND SELECTIVE SIGMA-LIGAND, PD-144418, Neuropharmacology, 36(1), 1997, pp. 51-62
DOPAMINE AGONIST-INDUCED INHIBITION OF NEUROTRANSMITTER RELEASE FROM THE AWAKE SQUIRREL-MONKEY PUTAMEN AS MEASURED BY MICRODIALYSIS
Authors: DAVIS MD HEFFNER TG COOKE LW
Citation: Md. Davis et al., DOPAMINE AGONIST-INDUCED INHIBITION OF NEUROTRANSMITTER RELEASE FROM THE AWAKE SQUIRREL-MONKEY PUTAMEN AS MEASURED BY MICRODIALYSIS, Journal of neurochemistry, 68(2), 1997, pp. 659-666
(ARYLOXY)ALKYLAMINES AS SELECTIVE HUMAN DOPAMINE D-4 RECEPTOR ANTAGONISTS - POTENTIAL ANTIPSYCHOTIC AGENTS
Authors: UNANGST PC CAPIRIS T CONNOR DT DOUBLEDAY R HEFFNER TG MACKENZIE RG MILLER SR PUGSLEY TA WISE LD
Citation: Pc. Unangst et al., (ARYLOXY)ALKYLAMINES AS SELECTIVE HUMAN DOPAMINE D-4 RECEPTOR ANTAGONISTS - POTENTIAL ANTIPSYCHOTIC AGENTS, Journal of medicinal chemistry, 40(25), 1997, pp. 4026-4029
(4-ARYL-1-PIPERAZINYL)ALKYL]CYCLOHEXYL]-1H-INDOLES AS DOPAMINE D2 PARTIAL AGONISTS AND AUTORECEPTOR AGONISTS
Authors: WUSTROW DJ SMITH WJ CORBIN AE DAVIS MD GEORGIC LM PUGSLEY TA WHETZEL SZ HEFFNER TG WISE LD
Citation: Dj. Wustrow et al., (4-ARYL-1-PIPERAZINYL)ALKYL]CYCLOHEXYL]-1H-INDOLES AS DOPAMINE D2 PARTIAL AGONISTS AND AUTORECEPTOR AGONISTS, Journal of medicinal chemistry, 40(2), 1997, pp. 250-259
CHROMENO[3,4-C]PYRIDIN-5-ONES - SELECTIVE HUMAN DOPAMINE D-4 RECEPTORANTAGONISTS AS POTENTIAL ANTIPSYCHOTIC AGENTS
Authors: UNANGST PC CAPIRIS T CONNOR DT HEFFNER TG MACKENZIE RG MILLER SR PUGSLEY TA WISE LD
Citation: Pc. Unangst et al., CHROMENO[3,4-C]PYRIDIN-5-ONES - SELECTIVE HUMAN DOPAMINE D-4 RECEPTORANTAGONISTS AS POTENTIAL ANTIPSYCHOTIC AGENTS, Journal of medicinal chemistry, 40(17), 1997, pp. 2688-2693
SUBSTITUTED [(4-PHENYLPIPERAZINYL)METHYL]BENZAMIDES - SELECTIVE DOPAMINE D-4 AGONISTS
Authors: GLASE SA AKUNNE HC GEORGIC LM HEFFNER TG MACKENZIE RG MANLEY PJ PUGSLEY TA WISE LD
Citation: Sa. Glase et al., SUBSTITUTED [(4-PHENYLPIPERAZINYL)METHYL]BENZAMIDES - SELECTIVE DOPAMINE D-4 AGONISTS, Journal of medicinal chemistry, 40(12), 1997, pp. 1771-1772
RYL-1-PIPERAZINYL)ETHYL]-2-NAPHTHALENECARBOXAMIDES - SELECTIVE DOPAMINE D-3 RECEPTOR PARTIAL AGONISTS
Authors: GLASE SA AKUNNE HC HEFFNER TG JOHNSON SJ KESTEN SR MACKENZIE RG MANLEY PJ PUGSLEY TA WRIGHT JL WISE LD
Citation: Sa. Glase et al., RYL-1-PIPERAZINYL)ETHYL]-2-NAPHTHALENECARBOXAMIDES - SELECTIVE DOPAMINE D-3 RECEPTOR PARTIAL AGONISTS, Bioorganic & medicinal chemistry letters, 6(12), 1996, pp. 1361-1366
AFFINITY FOR DOPAMINE D-2, D-3, AND D-4 RECEPTORS OF 8-AMINOTETRALINS- RELEVANCE OF D-2 AGONIST BINDING FOR DETERMINATION OF RECEPTOR SUBTYPE SELECTIVITY
Authors: VANVLIET LA TEPPER PG DIJKSTRA D DAMSMA G WIKSTROM H PUGSLEY TA AKUNNE HC HEFFNER TG GLASE SA WISE LD
Citation: La. Vanvliet et al., AFFINITY FOR DOPAMINE D-2, D-3, AND D-4 RECEPTORS OF 8-AMINOTETRALINS- RELEVANCE OF D-2 AGONIST BINDING FOR DETERMINATION OF RECEPTOR SUBTYPE SELECTIVITY, Journal of medicinal chemistry, 39(21), 1996, pp. 4233-4237
ARYL 1-BUT-3-YNYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINES AS POTENTIAL ANTIPSYCHOTIC AGENTS - SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS
Authors: GLASE SA AKUNNE HC HEFFNER TG JAEN JC MACKENZIE RG MELTZER LT PUGSLEY TA SMITH SJ WISE LD
Citation: Sa. Glase et al., ARYL 1-BUT-3-YNYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINES AS POTENTIAL ANTIPSYCHOTIC AGENTS - SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS, Journal of medicinal chemistry, 39(16), 1996, pp. 3179-3187
REDUCED AMIDE BOND NEUROTENSIN-8-13 MIMETICS WITH POTENT IN-VIVO ACTIVITY
Authors: WUSTROW DJ DAVIS MD AKUNNE HC CORBIN AE WILEY JN WISE LD HEFFNER TG
Citation: Dj. Wustrow et al., REDUCED AMIDE BOND NEUROTENSIN-8-13 MIMETICS WITH POTENT IN-VIVO ACTIVITY, Bioorganic & medicinal chemistry letters, 5(9), 1995, pp. 997-1002
DIFFERENTIAL-EFFECTS OF THE NONPEPTIDE NEUROTENSIN ANTAGONIST, SR-48692, ON THE PHARMACOLOGICAL EFFECTS OF NEUROTENSIN AGONISTS
Authors: PUGSLEY TA AKUNNE HC WHETZEL SZ DEMATTOS S CORBIN AE WILEY JN WUSTROW DJ WISE LD HEFFNER TG
Citation: Ta. Pugsley et al., DIFFERENTIAL-EFFECTS OF THE NONPEPTIDE NEUROTENSIN ANTAGONIST, SR-48692, ON THE PHARMACOLOGICAL EFFECTS OF NEUROTENSIN AGONISTS, Peptides, 16(1), 1995, pp. 37-44
CHARACTERIZATION OF BINDING OF [H-3]PD-128907, A SELECTIVE DOPAMINE D-3 RECEPTOR AGONIST LIGAND, TO CHO-K1 CELLS
Authors: AKUNNE HC TOWERS P ELLIS GJ DIJKSTRA D WIKSTROM H HEFFNER TG WISE LD PUGSLEY TA
Citation: Hc. Akunne et al., CHARACTERIZATION OF BINDING OF [H-3]PD-128907, A SELECTIVE DOPAMINE D-3 RECEPTOR AGONIST LIGAND, TO CHO-K1 CELLS, Life sciences, 57(15), 1995, pp. 1401-1410
NEUROCHEMICAL AND FUNCTIONAL-CHARACTERIZATION OF THE PREFERENTIALLY SELECTIVE DOPAMINE D3 AGONIST PD-128907
Authors: PUGSLEY TA DAVIS MD AKUNNE HC MACKENZIE RG SHIH YH DAMSMA G WIKSTROM H WHETZEL SZ GEORGIC LM COOKE LW DEMATTOS SB CORBIN AE GLASE SA WISE LD DIJKSTRA D HEFFNER TG
Citation: Ta. Pugsley et al., NEUROCHEMICAL AND FUNCTIONAL-CHARACTERIZATION OF THE PREFERENTIALLY SELECTIVE DOPAMINE D3 AGONIST PD-128907, The Journal of pharmacology and experimental therapeutics, 275(3), 1995, pp. 1355-1366
CI-1007, A DOPAMINE PARTIAL AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT.1. NEUROCHEMICAL EFFECTS
Authors: PUGSLEY TA DAVIS MD AKUNNE HC COOKE LW WHETZEL SZ MACKENZIE RG SHIH YH VANLEEUWEN DH DEMATTOS SB GEORGIC LM CAPRATHE BW WRIGHT JC JAEN JC WISE LD HEFFNER TG
Citation: Ta. Pugsley et al., CI-1007, A DOPAMINE PARTIAL AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT.1. NEUROCHEMICAL EFFECTS, The Journal of pharmacology and experimental therapeutics, 274(2), 1995, pp. 898-911
CI-1007, A DOPAMINE PARTIAL AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT.2. NEUROPHYSIOLOGICAL-EFFECTS AND BEHAVIORAL-EFFECTS
Authors: MELTZER LT CHRISTOFFERSEN CL CORBIN AE NINTEMAN FW SERPA KA WILEY JN WISE LD HEFFNER TG
Citation: Lt. Meltzer et al., CI-1007, A DOPAMINE PARTIAL AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT.2. NEUROPHYSIOLOGICAL-EFFECTS AND BEHAVIORAL-EFFECTS, The Journal of pharmacology and experimental therapeutics, 274(2), 1995, pp. 912-920
IDENTIFICATION, CHARACTERIZATION AND PHARMACOLOGICAL PROFILE OF 3 METABOLITES OF PHENYL-1-[(3-PHENYLCYCLOHEXEN-1-YL)METHYL]PYRIDINE (CI-1007), A DOPAMINE AUTORECEPTOR AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT())
Authors: WRIGHT JL DOWNING DM FENG MR HAYES RN HEFFNER TG MACKENZIE RG MELTZER LT PUGSLEY TA WISE LD
Citation: Jl. Wright et al., IDENTIFICATION, CHARACTERIZATION AND PHARMACOLOGICAL PROFILE OF 3 METABOLITES OF PHENYL-1-[(3-PHENYLCYCLOHEXEN-1-YL)METHYL]PYRIDINE (CI-1007), A DOPAMINE AUTORECEPTOR AGONIST AND POTENTIAL ANTIPSYCHOTIC AGENT()), Journal of medicinal chemistry, 38(26), 1995, pp. 5007-5014
SYNTHESIS AND DOPAMINERGIC ACTIVITY OF PYRIDINE ANALOGS OF 5-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN
Authors: GLASE SA CORBIN AE PUGSLEY TA HEFFNER TG WISE LD
Citation: Sa. Glase et al., SYNTHESIS AND DOPAMINERGIC ACTIVITY OF PYRIDINE ANALOGS OF 5-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN, Journal of medicinal chemistry, 38(16), 1995, pp. 3132-3137
AGONIST PROPERTIES OF A STABLE HEXAPEPTIDE ANALOG OF NEUROTENSIN, N(ALPHA)MEARG-LYS-PRO-TRP-TLEU-LEU (NT1)
Authors: AKUNNE HC DEMATTOS SB WHETZEL SZ WUSTROW DJ DAVIS DM WISE LD CODY WL PUGSLEY TA HEFFNER TG
Citation: Hc. Akunne et al., AGONIST PROPERTIES OF A STABLE HEXAPEPTIDE ANALOG OF NEUROTENSIN, N(ALPHA)MEARG-LYS-PRO-TRP-TLEU-LEU (NT1), Biochemical pharmacology, 49(8), 1995, pp. 1147-1154
STRUCTURE-ACTIVITY AND CONFORMATIONAL STUDIES OF A SERIES OF MODIFIEDC-TERMINAL HEXAPEPTIDE NEUROTENSIN ANALOGS
Authors: HEYL DL SEFLER AM HE JX SAWYER TK WUSTROW DJ AKUNNE HC DAVIS MD PUGSLEY TA HEFFNER TG CORBIN AE CODY WL
Citation: Dl. Heyl et al., STRUCTURE-ACTIVITY AND CONFORMATIONAL STUDIES OF A SERIES OF MODIFIEDC-TERMINAL HEXAPEPTIDE NEUROTENSIN ANALOGS, International journal of peptide & protein research, 44(3), 1994, pp. 233-238
Risultati: 1-25 | 26-30