Authors:
HAMILL TG
HUTCHINSON JH
HARTMAN GD
BURNS HD
Citation: Tg. Hamill et al., NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONISTS - 3 - THE SYNTHESIS OF [H-3]L-767,685 AND [H-3]L-767,679, Journal of labelled compounds & radiopharmaceuticals, 41(7), 1998, pp. 677-680
Authors:
PRUEKSARITANONT T
GORHAM LM
BRESLIN MJ
HUTCHINSON JH
HARTMAN GD
VYAS KP
BAILLIE TA
Citation: T. Prueksaritanont et al., IN-VITRO AND IN-VIVO EVALUATIONS OF THE METABOLISM, PHARMACOKINETICS,AND BIOAVAILABILITY OF ESTER PRODRUGS OF L-767,679, A POTENT FIBRINOGEN RECEPTOR ANTAGONIST - AN APPROACH FOR THE SELECTION OF A PRODRUG CANDIDATE, Drug metabolism and disposition, 25(8), 1997, pp. 978-984
Authors:
HUTCHINSON JH
COOK JJ
BRASHEAR KM
BRESLIN MJ
GLASS JD
GOULD RJ
HALCZENKO W
HOLAHAN MA
LYNCH RJ
SITKO GR
STRANIERI MT
HARTMAN GD
Citation: Jh. Hutchinson et al., NONPEPTIDE GLYCOPROTEIN IIB IIIA ANTAGONISTS .2. DESIGN AND IN-VIVO EVALUATION OF 3,4-DIHYDRO-1(1H)-ISOQUINOLINONE-BASED ANTAGONISTS AND ETHYL-ESTER PRODRUGS/, Journal of medicinal chemistry, 39(23), 1996, pp. 4583-4591
Authors:
HUTCHINSON JH
CHARLESON S
EVANS JF
FALGUEYRET JP
HOOGSTEEN K
JONES TR
KARGMAN S
MACDONALD D
MCFARLANE CS
NICHOLSON DW
PIECHUTA H
RIENDEAU D
SCHEIGETZ J
THERIEN M
GIRARD Y
Citation: Jh. Hutchinson et al., THIOPYRANOL[2,3,4-C,D] INDOLES AS INHIBITORS OF 5-LIPOXYGENASE, 5-LIPOXYGENASE-ACTIVATING PROTEIN, AND LEUKOTRIENE C-4 SYNTHASE, Journal of medicinal chemistry, 38(22), 1995, pp. 4538-4547
Authors:
FALGUEYRET JP
DENIS D
MACDONALD D
HUTCHINSON JH
RIENDEAU D
Citation: Jp. Falgueyret et al., CHARACTERIZATION OF THE ARACHIDONATE AND ATP BINDING-SITES OF HUMAN 5-LIPOXYGENASE USING PHOTOAFFINITY-LABELING AND ENZYME IMMOBILIZATION, Biochemistry, 34(41), 1995, pp. 13603-13611
Authors:
HUTCHINSON JH
RIENDEAU D
BRIDEAU C
CHAN C
FALGUEYRET JP
GUAY J
JONES TR
LEPINE C
MACDONALD D
MCFARLANE CS
PIECHUTA H
SCHEIGETZ J
TAGARI P
THERIEN M
GIRARD Y
Citation: Jh. Hutchinson et al., THIOPYRANO[2,3,4-CD]INDOLES AS 5-LIPOXYGENASE INHIBITORS - SYNTHESIS,BIOLOGICAL PROFILE, AND RESOLUTION OF RO-1H-THIOPYRANO[2,3,4-CD]INDOL-YL]ETHOXY]BUTANOIC ACID, Journal of medicinal chemistry, 37(8), 1994, pp. 1153-1164
Authors:
DUCHARME Y
BRIDEAU C
DUBE D
CHAN CC
FALGUEYRET JP
GILLARD JW
GUAY J
HUTCHINSON JH
MCFARLANE CS
RIENDEAU D
SCHEIGETZ J
GIRARD Y
Citation: Y. Ducharme et al., NAPHTHALENIC LIGNAN LACTONES AS SELECTIVE, NONREDOX 5-LIPOXYGENASE INHIBITORS - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF (METHOXYALKYL)THIAZOLEAND METHOXYTETRAHYDROPYRAN HYBRIDS, Journal of medicinal chemistry, 37(4), 1994, pp. 512-518
Authors:
YOUNG RN
GILLARD JW
HUTCHINSON JH
LEGER S
PRASIT P
Citation: Rn. Young et al., DISCOVERY OF INHIBITORS OF THE 5-LIPOXYGENASE ACTIVATING PROTEIN (FLAP), Journal of lipid mediators, 6(1-3), 1993, pp. 233-238
Authors:
PRASIT P
BELLEY M
BLOUIN M
BRIDEAU C
CHAN C
CHARLESON S
EVANS JF
FRENETTE R
GAUTHIER JY
GUAY J
GILLARD JW
GRIMM E
FORDHUTCHINSON AW
HUTCHINSON JH
FORTIN R
JONES TR
MANCINI J
LEGER S
MCFARLANE CS
PIECHUTA H
RIENDEAU D
ROY P
TAGARI P
VICKERS PJ
YOUNG RN
ZAMBONI R
Citation: P. Prasit et al., A NEW CLASS OF LEUKOTRIENE BIOSYNTHESIS INHIBITOR - THE DEVELOPMENT OF MK-0591, Journal of lipid mediators, 6(1-3), 1993, pp. 239-244
Authors:
BRIDEAU C
CHAN CC
GUEVREMONT D
HUTCHINSON JH
MCDONNELL J
MOORE V
Citation: C. Brideau et al., INHIBITION OF SYNOVIAL-LTB(4) PRODUCTION BY A SPECIFIC LEUKOTRIENE BIOSYNTHESIS INHIBITOR, MK-0591, IN A RABBIT MODEL OF JOINT INFLAMMATION, Drug development research, 29(3), 1993, pp. 188-194
Authors:
HUTCHINSON JH
RIENDEAU D
BRIDEAU C
CHAN C
DELORME D
DENIS D
FALGUEYRET JP
FORTIN R
GUAY J
HAMEL P
JONES TR
MACDONALD D
MCFARLANE CS
PIECHUTA H
SCHEIGETZ J
TAGARI P
THERIEN M
GIRARD Y
Citation: Jh. Hutchinson et al., SUBSTITUTED THIOPYRANO[2,3,4-C,D]INDOLES AS POTENT, SELECTIVE, AND ORALLY-ACTIVE INHIBITORS OF 5-LIPOXYGENASE - SYNTHESIS AND BIOLOGICAL EVALUATION OF L-691,816, Journal of medicinal chemistry, 36(19), 1993, pp. 2771-2787