Authors:
Lerner, C
Ruf, A
Gramlich, V
Masjost, B
Zurcher, G
Jakob-Roetne, R
Borroni, E
Diederich, F
Citation: C. Lerner et al., X-ray crystal structure of a bisubstrate inhibitor bound to the enzyme catechol-O-methyltransferase: A dramatic effect of inhibitor preorganization on binding affinity, ANGEW CHEM, 40(21), 2001, pp. 4040
Authors:
Masjost, B
Ballmer, P
Borroni, E
Zurcher, G
Winkler, FK
Jakob-Roetne, R
Diederich, F
Citation: B. Masjost et al., Structure-based design, synthesis, and in vitro evaluation of bisubstrate inhibitors for catechol O-methyltransferase (COMT), CHEM-EUR J, 6(6), 2000, pp. 971-982
Authors:
Kuner, P
Bohrmann, B
Tjernberg, LO
Naslund, J
Huber, G
Celenk, S
Gruninger-Leitch, F
Richards, JG
Jakob-Roetne, R
Kemp, JA
Nordstedt, C
Citation: P. Kuner et al., Controlling polymerization of beta-amyloid and prion-derived peptides withsynthetic small molecule ligands, J BIOL CHEM, 275(3), 2000, pp. 1673-1678