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Results: 1-25 | 26-49
Results: 1-25/49
The estrogen receptor: a structure-based approach to the design of new specific hormone-receptor combinations
Authors: Tedesco, R Thomas, JA Katzenellenbogen, BS Katzenellenbogen, JA
Citation: R. Tedesco et al., The estrogen receptor: a structure-based approach to the design of new specific hormone-receptor combinations, CHEM BIOL, 8(3), 2001, pp. 277-287
Fluorine-substituted ligands for the peroxisome proliferator-activated receptor gamma (PPAR gamma): potential imaging agents for metastatic tumors
Authors: Kim, SH Jonson, SD Welch, MJ Katzenellenbogen, JA
Citation: Sh. Kim et al., Fluorine-substituted ligands for the peroxisome proliferator-activated receptor gamma (PPAR gamma): potential imaging agents for metastatic tumors, BIOCONJ CHE, 12(3), 2001, pp. 439-450
Comparison of animal models for the evaluation of radiolabeled androgens
Authors: Downer, JD Jones, LA Engelbach, JA Lich, LL Mao, W Carlson, KE Katzenellenbogen, JA Welch, MJ
Citation: Jd. Downer et al., Comparison of animal models for the evaluation of radiolabeled androgens, NUCL MED BI, 28(6), 2001, pp. 613-626
Effect of administration route on FES uptake into MCF-7 tumors
Authors: Downer, JB Jones, LA Katzenellenbogen, JA Welch, MJ
Citation: Jb. Downer et al., Effect of administration route on FES uptake into MCF-7 tumors, NUCL MED BI, 28(4), 2001, pp. 397-399
Estrogen pyrazoles: Defining the pyrazole core structure and the orientation of substituents in the ligand binding pocket of the estrogen receptor
Authors: Stauffer, SR Huang, Y Coletta, CJ Tedesco, R Katzenellenbogen, JA
Citation: Sr. Stauffer et al., Estrogen pyrazoles: Defining the pyrazole core structure and the orientation of substituents in the ligand binding pocket of the estrogen receptor, BIO MED CH, 9(1), 2001, pp. 141-150
Triarylpyrazoles with basic side chains: Development of pyrazole-based estrogen receptor antagonists
Authors: Stauffer, SR Huang, YR Aron, ZD Coletta, CJ Sun, J Katzenellenbogen, BS Katzenellenbogen, JA
Citation: Sr. Stauffer et al., Triarylpyrazoles with basic side chains: Development of pyrazole-based estrogen receptor antagonists, BIO MED CH, 9(1), 2001, pp. 151-161
Furans with basic side chains: Synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha
Authors: Mortensen, DS Rodriguez, AL Sun, J Katzenellenbogen, BS Katzenellenbogen, JA
Citation: Ds. Mortensen et al., Furans with basic side chains: Synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha, BIOORG MED, 11(18), 2001, pp. 2521-2524
Synthesis and evaluation of hexahydrochrysene and tetrahydrobenzofluorene ligands for the estrogen receptor
Authors: Tedesco, R Youngman, MK Wilson, SR Katzenellenbogen, JA
Citation: R. Tedesco et al., Synthesis and evaluation of hexahydrochrysene and tetrahydrobenzofluorene ligands for the estrogen receptor, BIOORG MED, 11(10), 2001, pp. 1281-1284
Probing conformational changes in the estrogen receptor: Evidence for a partially unfolded intermediate facilitating ligand binding and release
Authors: Gee, AC Katzenellenbogen, JA
Citation: Ac. Gee et Ja. Katzenellenbogen, Probing conformational changes in the estrogen receptor: Evidence for a partially unfolded intermediate facilitating ligand binding and release, MOL ENDOCR, 15(3), 2001, pp. 421-428
Metabolic flare: Indicator of hormone responsiveness in advanced breast cancer
Authors: Mortimer, JE Dehdashti, F Siegel, BA Trinkaus, K Katzenellenbogen, JA Welch, MJ
Citation: Je. Mortimer et al., Metabolic flare: Indicator of hormone responsiveness in advanced breast cancer, J CL ONCOL, 19(11), 2001, pp. 2797-2803
Estrogen regulation of human osteoblast function is determined by the stage of differentiation and the estrogen receptor isoform
Authors: Waters, KM Rickard, DJ Riggs, BL Khosla, S Katzenellenbogen, JA Katzenellenbogen, BS Moore, J Spelsberg, TC
Citation: Km. Waters et al., Estrogen regulation of human osteoblast function is determined by the stage of differentiation and the estrogen receptor isoform, J CELL BIOC, 83(3), 2001, pp. 448-462
Nongenotropic, sex-nonspecific signaling through the estrogen or androgen receptors: Dissociation from transcriptional activity
Authors: Kousteni, S Bellido, T Plotkin, LI O'Brien, CA Bodenner, DL Han, L Han, K DiGregorio, GB Katzenellenbogen, JA Katzenellenbogen, BS Roberson, PK Weinstein, RS Jilka, RL Manolagas, SC
Citation: S. Kousteni et al., Nongenotropic, sex-nonspecific signaling through the estrogen or androgen receptors: Dissociation from transcriptional activity, CELL, 104(5), 2001, pp. 719-730
Estrogen receptor-beta potency-selective ligands: Structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues
Authors: Meyers, MJ Sun, J Carlson, KE Marriner, GA Katzenellenbogen, BS Katzenellenbogen, JA
Citation: Mj. Meyers et al., Estrogen receptor-beta potency-selective ligands: Structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues, J MED CHEM, 44(24), 2001, pp. 4230-4251
Salicylaldoxime moiety as a phenolic "A-ring" substitute in estrogen receptor ligands
Authors: Minutolo, F Bertini, S Papi, C Carlson, KE Katzenellenbogen, JA Macchia, M
Citation: F. Minutolo et al., Salicylaldoxime moiety as a phenolic "A-ring" substitute in estrogen receptor ligands, J MED CHEM, 44(24), 2001, pp. 4288-4291
Synthesis and biological evaluation of a novel series of furans: Ligands selective for estrogen receptor alpha
Authors: Mortensen, DS Rodriguez, AL Carlson, KE Sun, J Katzenellenbogen, BS Katzenellenbogen, JA
Citation: Ds. Mortensen et al., Synthesis and biological evaluation of a novel series of furans: Ligands selective for estrogen receptor alpha, J MED CHEM, 44(23), 2001, pp. 3838-3848
Steroids labeled with F-18 for imaging tumors by positron emission tomography
Authors: Katzenellenbogen, JA
Citation: Ja. Katzenellenbogen, Steroids labeled with F-18 for imaging tumors by positron emission tomography, J FLUORINE, 109(1), 2001, pp. 49-54
Activation of estrogen receptor beta is a prerequisite for estrogen-dependent upregulation of nitric oxide synthases in neonatal rat cardiac myocytes
Authors: Nuedling, S Karas, RH Mendelsohn, ME Katzenellenbogen, JA Katzenellenbogen, BS Meyer, R Vetter, H Grohe, C
Citation: S. Nuedling et al., Activation of estrogen receptor beta is a prerequisite for estrogen-dependent upregulation of nitric oxide synthases in neonatal rat cardiac myocytes, FEBS LETTER, 502(3), 2001, pp. 103-108
One-pot formation of substituted cyclopentadienyl and indenyltricarbonyl rhenium complexes through in situ generation of cyclopentadienyl- and indenyltributylstannanes
Authors: Cesati, RR Katzenellenbogen, JA
Citation: Rr. Cesati et Ja. Katzenellenbogen, One-pot formation of substituted cyclopentadienyl and indenyltricarbonyl rhenium complexes through in situ generation of cyclopentadienyl- and indenyltributylstannanes, J AM CHEM S, 123(17), 2001, pp. 4093-4094
Preparation of hexahydrobenzo[f]isoquinolines using a vinylogous Pictet-Spengler cyclization
Authors: Cesati, RR Katzenellenbogen, JA
Citation: Rr. Cesati et Ja. Katzenellenbogen, Preparation of hexahydrobenzo[f]isoquinolines using a vinylogous Pictet-Spengler cyclization, ORG LETT, 2(23), 2000, pp. 3635-3638
Regioselective synthesis of 1,3,5-triaryl-4-alkylpyrazoles: Novel ligands for the estrogen receptor
Authors: Huang, YR Katzenellenbogen, JA
Citation: Yr. Huang et Ja. Katzenellenbogen, Regioselective synthesis of 1,3,5-triaryl-4-alkylpyrazoles: Novel ligands for the estrogen receptor, ORG LETT, 2(18), 2000, pp. 2833-2836
Solid-phase synthesis of tetrasubstituted pyrazoles, novel ligands for theestrogen receptor
Authors: Stauffer, SR Katzenellenbogen, JA
Citation: Sr. Stauffer et Ja. Katzenellenbogen, Solid-phase synthesis of tetrasubstituted pyrazoles, novel ligands for theestrogen receptor, J COMB CHEM, 2(4), 2000, pp. 318-329
Estrogen receptor transcription and transactivation Estrogen receptor alpha and estrogen receptor beta: regulation by selective estrogen receptor modulators and importance in breast cancer
Authors: Katzenellenbogen, BS Katzenellenbogen, JA
Citation: Bs. Katzenellenbogen et Ja. Katzenellenbogen, Estrogen receptor transcription and transactivation Estrogen receptor alpha and estrogen receptor beta: regulation by selective estrogen receptor modulators and importance in breast cancer, BREAST CA R, 2(5), 2000, pp. 335-344
Radiochemical synthesis and tissue distribution of Tc-99m-labeled 7 alpha-substituted estradiol complexes
Authors: Skadden, MB Wust, FR Jonson, S Syhre, R Welch, MJ Spies, H Katzenellenbogen, JA
Citation: Mb. Skadden et al., Radiochemical synthesis and tissue distribution of Tc-99m-labeled 7 alpha-substituted estradiol complexes, NUCL MED BI, 27(3), 2000, pp. 269-278
Acyclic amides as estrogen receptor ligands: Synthesis, binding, activity and receptor interaction
Authors: Stauffer, SR Sun, J Katzenellenbogen, BS Katzenellenbogen, JA
Citation: Sr. Stauffer et al., Acyclic amides as estrogen receptor ligands: Synthesis, binding, activity and receptor interaction, BIO MED CH, 8(6), 2000, pp. 1293-1316
Triarylethylene bisphenols with a novel cycle are ligands for the estrogenreceptor
Authors: Kim, SH Katzenellenbogen, JA
Citation: Sh. Kim et Ja. Katzenellenbogen, Triarylethylene bisphenols with a novel cycle are ligands for the estrogenreceptor, BIO MED CH, 8(4), 2000, pp. 785-793
Risultati: 1-25 | 26-49