Authors:
ELLIOTT JM
CASCIERI MA
CHICCHI G
DAVIES S
KELLEHER FJ
KURTZ M
LADDUWAHETTY T
LEWIS RT
MACLEOD AM
MERCHANT KJ
SADOWSKI S
STEVENSON GI
Citation: Jm. Elliott et al., SERINE DERIVED NK1 ANTAGONISTS 1 - THE EFFECT OF MODIFICATIONS TO THESERINE SUBSTITUENTS, Bioorganic & medicinal chemistry letters, 8(14), 1998, pp. 1845-1850
Authors:
STEVENSON GI
HUSCROFT I
MACLEOD AM
SWAIN CJ
CASCIERI MA
CHICCHI GG
GRAHAM MI
HARRISON T
KELLEHER FJ
KURTZ M
LADDUWAHETTY T
MERCHANT KJ
METZGER JM
MACINTYRE DE
SADOWSKI S
SOHAL B
OWENS AP
Citation: Gi. Stevenson et al., 4,4-DISUBSTITUTED PIPERIDINE HIGH-AFFINITY NK1 ANTAGONISTS - STRUCTURE-ACTIVITY-RELATIONSHIPS AND IN-VIVO ACTIVITY, Journal of medicinal chemistry, 41(23), 1998, pp. 4623-4635
Authors:
SWAIN CJ
WILLIAMS BJ
BAKER R
CASCIERI MA
CHICCHI G
FORREST M
HERBERT R
KEOWN L
LADDUWAHETTY T
LUELL S
MACINTYRE DE
METZGER J
MORTON S
OWENS AP
SADOWSKI S
WATT AP
Citation: Cj. Swain et al., 3-BENZYLOXY-2-PHENYLPIPERIDINE NK1 ANTAGONISTS - THE INFLUENCE OF ALPHA-METHYL SUBSTITUTION, Bioorganic & medicinal chemistry letters, 7(23), 1997, pp. 2959-2962
Authors:
TATTERSALL FD
RYCROFT W
FRANCIS B
PEARCE D
MERCHANT K
MACLEOD AM
LADDUWAHETTY T
KEOWN L
SWAIN C
BAKER R
CASCIERI M
BER E
METZGER J
MACINTYRE DE
HILL RG
HARGREAVES RJ
Citation: Fd. Tattersall et al., TACHYKININ NK1 RECEPTOR ANTAGONISTS ACT CENTRALLY TO INHIBIT EMESIS INDUCED BY THE CHEMOTHERAPEUTIC AGENT CISPLATIN IN FERRETS, Neuropharmacology, 35(8), 1996, pp. 1121-1129
Authors:
LADDUWAHETTY T
BAKER R
CASCIERI MA
CHAMBERS MS
HAWORTH K
KEOWN LE
MACINTYRE DE
METZGER JM
OWEN S
RYCROFT W
SADOWSKI S
SEWARD EM
SHEPHEARD SL
SWAIN CJ
TATTERSALL FD
WATT AP
WILLIAMSON DW
HARGREAVES RJ
Citation: T. Ladduwahetty et al., N-HETEROARYL-2-PHENYL-3-(BENZYLOXY)PIPERIDINES - A NOVEL CLASS OF POTENT ORALLY-ACTIVE HUMAN NK1 ANTAGONISTS, Journal of medicinal chemistry, 39(15), 1996, pp. 2907-2914
Authors:
LADDUWAHETTY T
KEOWN L
CASCIERI MA
SADOWSKI S
Citation: T. Ladduwahetty et al., MORPHOLINE-BASED SUBSTANCE-P ANTAGONISTS - ASSESSMENT OF THE 3-POINT BINDING MODEL, Bioorganic & medicinal chemistry letters, 4(16), 1994, pp. 1917-1920