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BERAN M
CAO XB
ESTROV Z
JEHA S
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TALPAZ M
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LYDON NB
KANTARJIAN H
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REGENASS U
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Citation: E. Buchdunger et al., SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A PROTEIN-TYROSINE KINASE INHIBITOR OF THE 2-PHENYLAMINOPYRIMIDINE CLASS (VOL 92, PG 2558, 1995), Proceedings of the National Academy of Sciences of the United Statesof America, 95(20), 1998, pp. 12069-12069
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BUCHDUNGER E
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LYDON NB
Citation: E. Buchdunger et al., 4,5-DIANILINOPHTHALIMIDE - A PROTEIN-TYROSINE KINASE INHIBITOR WITH SELECTIVITY FOR THE EPIDERMAL GROWTH-FACTOR RECEPTOR SIGNAL-TRANSDUCTION PATHWAY AND POTENT IN-VIVO ANTITUMOR-ACTIVITY (VOL 91, PG 2334, 1994), Proceedings of the National Academy of Sciences of the United Statesof America, 95(20), 1998, pp. 12069-12069
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Citation: Nb. Lydon et al., A POTENT PROTEIN-TYROSINE KINASE INHIBITOR WHICH SELECTIVELY BLOCKS PROLIFERATION OF EPIDERMAL GROWTH-FACTOR RECEPTOR-EXPRESSING TUMOR-CELLS IN-VITRO AND IN-VIVO, International journal of cancer, 76(1), 1998, pp. 154-163
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MOLOGNI L
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MARCHESI E
DINICOLA M
BIONDI A
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BELOTTI D
POGLIANI E
LYDON NB
Citation: C. Gambacortipasserini et al., INHIBITION OF THE ABL KINASE-ACTIVITY BLOCKS THE PROLIFERATION OF BCRABL(+) LEUKEMIC-CELLS AND INDUCES APOPTOSIS/, Blood cells, molecules, & diseases, 23(19), 1997, pp. 380-394
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TAMURA S
BUCHDUNGER E
ZIMMERMANN J
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GILLILAND DG
DRUKER BJ
Citation: M. Carroll et al., CGP-57148, A TYROSINE KINASE INHIBITOR, INHIBITS THE GROWTH OF CELLS EXPRESSING BCR-ABL, TEL-ABL, AND TEL-PDGFR FUSION PROTEINS, Blood, 90(12), 1997, pp. 4947-4952
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CARROLL M
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TAMURA S
BUCHDUNGER E
LYDON NB
GILLILAND DG
Citation: Bj. Druker et al., CGP 57148, A TYROSINE KINASE INHIBITOR, INHIBITS THE GROWTH OF CELLS EXPRESSING BCR-ABL, TEL-ABL, AND TEL-PDGFR FUSION PROTEINS, Blood, 90(10), 1997, pp. 1091-1091
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LYDON NB
Citation: Bj. Druker et al., EFFECTS OF A SELECTIVE INHIBITOR OF THE ABL TYROSINE KINASE ON THE GROWTH OF BCR-ABL POSITIVE CELLS, Nature medicine, 2(5), 1996, pp. 561-566
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Authors:
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CHERINGTON V
TRAXLER PM
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ROBERTS TM
Citation: Mj. Corbley et al., A STRATEGY FOR SCREENING ANTITUMOR DRUGS UTILIZING ONCOGENES ENCODED IN RETROVIRAL VECTORS, International journal of cancer, 66(6), 1996, pp. 753-759
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ZIMMERMANN J
METT H
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MULLER M
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LYDON NB
Citation: E. Buchdunger et al., INHIBITION OF THE ABL PROTEIN-TYROSINE KINASE IN-VITRO AND IN-VIVO BYA 2-PHENYLAMINOPYRIMIDINE DERIVATIVE, Cancer research, 56(1), 1996, pp. 100-104
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MARCHESI E
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POGLIANI E
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Citation: C. Gambacortipasserini et al., INHIBITION OF THE ABELSON KINASE-ACTIVITY SELECTIVELY BLOCKS THE GROWTH OF BCR ABL LEUKEMIC-CELLS/, Blood, 88(10), 1996, pp. 924-924
Citation: M. Deininger et al., THE TYROSINE KINASE INHIBITOR CGP-57148 SELECTIVELY INHIBITS HEMATOPOIETIC COLONY FORMATION BY CML PROGENITOR CELLS OVER A 2-LOG DOSE RANGE, Blood, 88(10), 1996, pp. 1444-1444
Citation: M. Deininger et al., BCR-ABL POSITIVE CELL-LINES SHOW DIFFERENTIAL SENSITIVITY TO THE EFFECTS OF THE TYROSINE KINASE INHIBITOR CGP-57148, Blood, 88(10), 1996, pp. 1445-1445
Authors:
BUCHDUNGER E
METT H
TRINKS U
REGENASS U
MULLER M
MEYER T
BEILSTEIN P
WIRZ B
SCHNEIDER P
TRAXLER P
LYDON NB
Citation: E. Buchdunger et al., 4,5-BIS(4-FLUOROANILINO)PHTHALIMIDE - A SELECTIVE INHIBITOR OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR SIGNAL-TRANSDUCTION PATHWAY WITH POTENTIN-VIVO ANTITUMOR-ACTIVITY, Clinical cancer research, 1(8), 1995, pp. 813-821
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ZIMMERMANN J
METT H
MEYER T
MULLER M
REGENASS U
BUCHDUNGER E
Citation: Nb. Lydon et al., SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A NOVEL TYROSINE PROTEIN-KINASE INHIBITOR OF THE 2-PHENYLAMINO PYRIMIDINE CLASS, Journal of cellular biochemistry, 1995, pp. 69-69
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BUCHDUNGER E
ZIMMERMANN J
METT H
MEYER T
MULLER M
REGENASS U
LYDON NB
Citation: E. Buchdunger et al., SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A PROTEIN-TYROSINE KINASE INHIBITOR OF THE 2-PHENYLAMINOPYRIMIDINE CLASS, Proceedings of the National Academy of Sciences of the United Statesof America, 92(7), 1995, pp. 2558-2562
Authors:
WRIGHT JD
KEMP DM
LYDON NB
BLUM W
TRAXLER P
WOOLLEY A
TAYLOR PW
Citation: Jd. Wright et al., INHIBITION OF EPIDERMAL GROWTH-FACTOR RECEPTOR PROTEIN-TYROSINE KINASE - A POTENTIAL TREATMENT FOR PSORIASIS, Journal of investigative dermatology, 105(3), 1995, pp. 487-487
Citation: Dr. Stover et al., SRC PHOSPHORYLATION OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR AT NOVEL SITES MEDIATES RECEPTOR INTERACTION WITH SRC AND P85-ALPHA, The Journal of biological chemistry, 270(26), 1995, pp. 15591-15597