Authors:
Tagat, JR
McCombie, SW
Steensma, RW
Lin, SI
Nazareno, DV
Baroudy, B
Vantuno, N
Xu, S
Liu, J
Citation: Jr. Tagat et al., Piperazine-based CCR5 antagonists as HIV-1 inhibitors. I: 2(S)-methyl piperazine as a key pharmacophore element, BIOORG MED, 11(16), 2001, pp. 2143-2146
Authors:
Tagat, JR
Steensma, RW
McCombie, SW
Nazareno, DV
Lin, SI
Neustadt, BR
Cox, K
Xu, S
Wojcik, L
Murray, MG
Vantuno, N
Baroudy, BM
Strizki, JM
Citation: Jr. Tagat et al., Piperazine-based CCR5 antagonists as HIV-1 inhibitors. II. Discovery of 1-[(2,4-dimethyl-3-pyridinyl)carbonyl]-4-methyl-4-[3(S)-methyl-4-[1(S)-[4-(trifluoro-methyl)phenyl]ethyl]-1-piperazinyl]-piperidine N1-oxide (Sch-350634), an orally bioavailable, potent CCR5 antagonist, J MED CHEM, 44(21), 2001, pp. 3343-3346
Citation: Sw. Mccombie et al., New reactions of hydrazides. Part 1: Directed ortho- and lateral metalation of aromatic carbocyclic and heterocyclic systems, TETRAHEDR L, 40(50), 1999, pp. 8767-8770