Citation: Je. Macor et al., AN UNUSUAL BY-PRODUCT FROM A NONSYNCHRONOUS REACTION BETWEEN ETHYL 1,2,4-TRIAZINE-3-CARBOXYLATE AND AN ENAMINE, Chemical communications, (9), 1998, pp. 983-984
Citation: Jc. Blosser et al., CHALLENGES AND OPPORTUNITIES FOR DEVELOPING MUSCARINIC RECEPTOR SUBTYPE-BASED THERAPEUTIC AGENTS - INTRODUCTION, Drug development research, 40(2), 1997, pp. 101-103
Citation: Je. Macor et al., SYNTHESIS AND REACTIVITY OF PYRROLO[3,2-E]INDOLE - REMOVAL OF A N-BOMGROUP FROM AN UNACTIVATED INDOLE, Tetrahedron letters, 38(10), 1997, pp. 1673-1676
Citation: Je. Macor et al., A DIRECT SYNTHESIS OF 3-(PYRROLIDIN-3-YL)INDOLES FOR USE AS CONFORMATIONALLY RESTRICTED ANALOGS OF TRYPTAMINES, Synthesis, (4), 1997, pp. 443
Citation: Rs. Mansbach et al., CP-135,807, A SELECTIVE 5-HT1D AGONIST - EFFECTS IN DRUG DISCRIMINATION AND PUNISHMENT PROCEDURES IN THE PIGEON, Psychopharmacology, 128(3), 1996, pp. 313-319
Citation: Je. Macor et al., AN IMPROVED SYNTHESIS OF THE UNIQUE ANTIMIGRAINE AGENT CP-122,288 - ABROMINE ATOM PASSENGER IN AN INTRAMOLECULAR HECK REACTION, Tetrahedron letters, 37(25), 1996, pp. 4289-4292
Authors:
YU XJ
WAEBER C
CASTANON N
SCEARCE K
HEN R
MACOR JE
CHAUVEAU J
MOSKOWITZ MA
Citation: Xj. Yu et al., 5-CARBOXAMIDOTRYPTAMINE, CP-122,288, AND DIHYDROERGOTAMINE BUT NOT SUMATRIPTAN, CP-93,129, AND SEROTONIN-5-O-CARBOXYMETHYLGLYCYL-TYROSINAMIDE BLOCK DURAL PLASMA-PROTEIN EXTRAVASATION IN KNOCKOUT MICE THAT LACK5-HYDROXYTRYPTAMINE(1B) RECEPTORS (VOL 49, PG 761, 1996), Molecular pharmacology, 50(4), 1996, pp. 1055-1055
Authors:
YU XJ
WAEBER C
CASTANON N
SCEARCE K
HEN R
MACOR JE
CHAVEAU J
MOSKOWITZ MA
Citation: Xj. Yu et al., 5-CARBOXAMIDO-TRYPTAMINE, CP-122,288 AND DIHYDROERGOTAMINE BUT NOT SUMATRIPTAN, CP-93,129, AND SEROTONIN-5-O-CARBOXYMETHYL-GLYCYL-TYROSINAMIDE BLOCK DURAL PLASMA-PROTEIN EXTRAVASATION IN KNOCKOUT MICE THAT LACK 5-HYDROXYTRYPTAMINE(1B) RECEPTORS, Molecular pharmacology, 49(5), 1996, pp. 761-765
Authors:
MACOR JE
ORDWAY T
SMITH RL
VERHOEST PR
MACK RA
Citation: Je. Macor et al., SYNTHESIS AND USE OF 5-VINYL-1,2,4-OXADIAZOLES AS MICHAEL ACCEPTORS -A RAPID SYNTHESIS OF THE POTENT MUSCARINIC AGONIST L-670,548, Journal of organic chemistry, 61(10), 1996, pp. 3228-3229
Authors:
MACOR JE
BLAKE JF
DESAI K
POST RJ
SCHMIDT AW
Citation: Je. Macor et al., THE DISCOVERY OF A NOVEL AND POTENT BENZODIAZEPINE RECEPTOR PHARMACOPHORE, Bioorganic & medicinal chemistry letters, 5(20), 1995, pp. 2397-2402
Citation: Je. Macor, AN UNUSUAL BY-PRODUCT IN A CONCISE SYNTHESIS OF A ROTATIONALLY RESTRICTED PHENOLIC ANALOG OF SEROTONIN, Tetrahedron letters, 36(39), 1995, pp. 7019-7022
Authors:
GUPTA P
BROWN D
BUTLER P
ELLIS P
GRAYSON KL
LAND GC
MACOR JE
ROBSON SF
WYTHES MJ
SHEPPERSON NB
Citation: P. Gupta et al., THE IN-VIVO PHARMACOLOGICAL PROFILE OF A 5-HT1 RECEPTOR AGONIST, CP-122,288, A SELECTIVE INHIBITOR OF NEUROGENIC INFLAMMATION, British Journal of Pharmacology, 116(5), 1995, pp. 2385-2390
Authors:
GUPTA P
BUTLER P
ELLIS P
GRAYSON KL
LAND GC
MACOR JE
ROBSON SF
SHEPPERSON NB
WYTHES MJ
Citation: P. Gupta et al., THE IN-VIVO PHARMACOLOGICAL PROFILE OF CP-122,288, A SELECTIVE INHIBITOR OF NEUROGENIC INFLAMMATION, British Journal of Pharmacology, 115, 1995, pp. 7-7
Citation: Je. Macor et K. Ryan, A SHORT SYNTHESIS OF A CONFORMATIONALLY RESTRICTED ANALOG OF THE NEUROTRANSMITTER SEROTONIN WITH REDUCED BASICITY, Heterocycles, 37(3), 1994, pp. 1447-1450
Authors:
LEBEL LA
NOWAKOWSKI JT
MACOR JE
FOX CB
KOE BK
Citation: La. Lebel et al., DOPAMINE UPTAKE INHIBITORY ACTIVITY OF NOVEL TRYPTAMINE 5-HT, RECEPTOR LIGANDS, Drug development research, 33(4), 1994, pp. 413-421
Citation: Je. Macor et al., THE SYNTHESIS OF CONFORMATIONALLY ROTATIONALLY RESTRICTED ANALOGS OF THE NEUROTRANSMITTER SEROTONIN, Tetrahedron letters, 35(1), 1994, pp. 45-48
Citation: Je. Macor et al., USE OF 2,5-DIMETHYLPYRROLE AS AN AMINO-PROTECTING GROUP IN AN EFFICIENT SYNTHESIS OF MINO-3-[(N-METHYL-PYRROLIDIN-2(R)-YL)METHYL]INDOLE, Journal of organic chemistry, 59(24), 1994, pp. 7496-7498
Authors:
MACOR JE
BLANK DH
FOX CB
LEBEL LA
NEWMAN ME
POST RJ
RYAN K
SCHMIDT AW
SCHULZ DW
KOE BK
Citation: Je. Macor et al., 5-[(3-NITROPYRID-2-YL)AMINO]INDOLES - NOVEL SEROTONIN AGONISTS WITH SELECTIVITY FOR THE 5-HT1D RECEPTOR - VARIATION OF THE C3 SUBSTITUENT ON THE INDOLE TEMPLATE LEADS TO INCREASED 5-HT1D RECEPTOR SELECTIVITY, Journal of medicinal chemistry, 37(16), 1994, pp. 2509-2512