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Results: 1-23 |
Results: 23
EXPLORATION OF THE IMPORTANCE OF THE P-2-P-3 -NHCO-MOIETY IN A POTENTDIPEPTIDE OR TRIPEPTIDE INHIBITOR OF CALPAIN-I - INSIGHTS INTO THE DEVELOPMENT OF NONPEPTIDIC INHIBITORS OF CALPAIN-I
Authors: CHATTERJEE S IQBAL M MALLYA S SENADHI SE OKANE TM MCKENNA BA BOZYCZKOCOYNE D KAUER JC SIMAN R MALLAMO JP
Citation: S. Chatterjee et al., EXPLORATION OF THE IMPORTANCE OF THE P-2-P-3 -NHCO-MOIETY IN A POTENTDIPEPTIDE OR TRIPEPTIDE INHIBITOR OF CALPAIN-I - INSIGHTS INTO THE DEVELOPMENT OF NONPEPTIDIC INHIBITORS OF CALPAIN-I, Bioorganic & medicinal chemistry, 6(5), 1998, pp. 509-522
PRODRUG ESTERS OF THE INDOLOCARBAZOLE CEP-751 (KT-6587)
Authors: HUDKINS RL IQBAL M PARK CH GOLDSTEIN J HERMAN JL SHEK E MURAKATA C MALLAMO JP
Citation: Rl. Hudkins et al., PRODRUG ESTERS OF THE INDOLOCARBAZOLE CEP-751 (KT-6587), Bioorganic & medicinal chemistry letters, 8(14), 1998, pp. 1873-1876
NOVEL PEPTIDYL PHOSPHORUS DERIVATIVES AS INHIBITORS OF HUMAN CALPAIN I
Authors: TAO M BIHOVSKY R WELLS GJ MALLAMO JP
Citation: M. Tao et al., NOVEL PEPTIDYL PHOSPHORUS DERIVATIVES AS INHIBITORS OF HUMAN CALPAIN I, Journal of medicinal chemistry, 41(20), 1998, pp. 3912-3916
D-AMINO-ACID CONTAINING, HIGH-AFFINITY INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I
Authors: CHATTERJEE S GU ZQ DUNN D TAO M JOSEF K TRIPATHY R BIHOVSKY R SENADHI SE OKANE TM MCKENNA BA MALLYA S ATOR MA BOZYCZKOCOYNE D SIMAN R MALLAMO JP
Citation: S. Chatterjee et al., D-AMINO-ACID CONTAINING, HIGH-AFFINITY INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I, Journal of medicinal chemistry, 41(15), 1998, pp. 2663-2666
NONPEPTIDIC INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I
Authors: CHATTERJEE S SENADHI S BOZYCZKOCOYNE D SIMAN R MALLAMO JP
Citation: S. Chatterjee et al., NONPEPTIDIC INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I, Bioorganic & medicinal chemistry letters, 7(3), 1997, pp. 287-290
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A SERIES OF POTENT FLUOROMETHYL KETONE INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I
Authors: CHATTERJEE S ATOR MA BOZYCZKOCOYNE D JOSEF K WELLS G TRIPATHY R IQBAL M BIHOVSKY R SENADHI SE MALLYA S OKANE T MCKENNA BA SIMAN R MALLAMO JP
Citation: S. Chatterjee et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A SERIES OF POTENT FLUOROMETHYL KETONE INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I, Journal of medicinal chemistry, 40(23), 1997, pp. 3820-3828
NEUROTROPHIC 3,9-BIS[(ALKYLTHIO)METHYL]-K-252A AND 3,9-BIS(ALKOXYMETHYL)-K-252A DERIVATIVES
Authors: KANEKO M SAITO Y SAITO H MATSUMOTO T MATSUDA Y VAUGHT JL DIONNE CA ANGELES TS GLICKSMAN MA NEFF NT ROTELLA DP KAUER JC MALLAMO JP HUDKINS RL MURAKATA C
Citation: M. Kaneko et al., NEUROTROPHIC 3,9-BIS[(ALKYLTHIO)METHYL]-K-252A AND 3,9-BIS(ALKOXYMETHYL)-K-252A DERIVATIVES, Journal of medicinal chemistry, 40(12), 1997, pp. 1863-1869
POTENT ALPHA-KETOCARBONYL AND BORONIC ESTER DERIVED INHIBITORS OF PROTEASOME
Authors: IQBAL M CHATTERJEE S KAUER JC MALLAMO JP MESSINA PA REIBOLDT A SIMAN R
Citation: M. Iqbal et al., POTENT ALPHA-KETOCARBONYL AND BORONIC ESTER DERIVED INHIBITORS OF PROTEASOME, Bioorganic & medicinal chemistry letters, 6(3), 1996, pp. 287-290
XANTHENE DERIVED POTENT NONPEPTIDIC INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I
Authors: CHATERJEE S IQBAL M KAUER JC MALLAMO JP SENADHI S MALLYA S BOZYCZKOCOYNE D SIMAN R
Citation: S. Chaterjee et al., XANTHENE DERIVED POTENT NONPEPTIDIC INHIBITORS OF RECOMBINANT HUMAN CALPAIN-I, Bioorganic & medicinal chemistry letters, 6(13), 1996, pp. 1619-1622
POTENT FLUOROMETHYL KETONE INHIBITORS OF RECOMBINANT HUMAN CALPAIN I+
Authors: CHATTERJEE S JOSEF K WELLS G IQBAL M BIHOVSKY R MALLAMO JP ATOR MA BOZYCZKOCOYNE D MALLYA S SENADHI S SIMAN R
Citation: S. Chatterjee et al., POTENT FLUOROMETHYL KETONE INHIBITORS OF RECOMBINANT HUMAN CALPAIN I+, Bioorganic & medicinal chemistry letters, 6(11), 1996, pp. 1237-1240
A CONVENIENT SYNTHESIS OF 3-SUBSTITUTED PIPECOLIC ACID METHYL-ESTERS
Authors: SUBRAMANYAM C CHATTARJEE S MALLAMO JP
Citation: C. Subramanyam et al., A CONVENIENT SYNTHESIS OF 3-SUBSTITUTED PIPECOLIC ACID METHYL-ESTERS, Tetrahedron letters, 37(4), 1996, pp. 459-462
A CONVENIENT SYNTHESIS OF 3-SUBSTITUTED PIPECOLIC ACID METHYL-ESTERS (VOL 37, PG 459, 1996)
Authors: SUBRAMANYAM C CHATTERJEE S MALLAMO JP
Citation: C. Subramanyam et al., A CONVENIENT SYNTHESIS OF 3-SUBSTITUTED PIPECOLIC ACID METHYL-ESTERS (VOL 37, PG 459, 1996), Tetrahedron letters, 37(14), 1996, pp. 2315-2315
SYNTHESIS AND BINDING-AFFINITY OF ,9A-HEXAHYDRO-9,4-(IMINOMETHANO)-1H-BENZ[F]INDENES - LIGANDS FOR THE PCP SITE OF THE NMDA RECEPTOR
Authors: REUMAN M MALLAMO JP DEHAVENHUDKINS DL
Citation: M. Reuman et al., SYNTHESIS AND BINDING-AFFINITY OF ,9A-HEXAHYDRO-9,4-(IMINOMETHANO)-1H-BENZ[F]INDENES - LIGANDS FOR THE PCP SITE OF THE NMDA RECEPTOR, Bioorganic & medicinal chemistry letters, 5(4), 1995, pp. 371-376
REGIOCONTROLLED SYNTHESES OF BENZO[B]QUINOLIZINIUM AND HETEROISOQUINOLINIUM CATIONS
Authors: EARLEY WG DORITY JA KUMAR V MALLAMO JP
Citation: Wg. Earley et al., REGIOCONTROLLED SYNTHESES OF BENZO[B]QUINOLIZINIUM AND HETEROISOQUINOLINIUM CATIONS, Heterocycles, 41(2), 1995, pp. 309-314
WIN-63480, A HYDROPHILIC TCP-SITE LIGAND, HAS REDUCED AGONIST-INDEPENDENT NMDA ION-CHANNEL ACCESS COMPARED TO MK-801 AND PHENCYCLIDINE
Authors: AULT B MILLER MS KELLY MD HILDEBRAND LM EARLEY WG LUTTINGER D MALLAMO JP WARD SJ
Citation: B. Ault et al., WIN-63480, A HYDROPHILIC TCP-SITE LIGAND, HAS REDUCED AGONIST-INDEPENDENT NMDA ION-CHANNEL ACCESS COMPARED TO MK-801 AND PHENCYCLIDINE, Neuropharmacology, 34(12), 1995, pp. 1597-1606
AN EVALUATION OF THE ANTIRHINOVIRAL ACTIVITY OF ACYLFURAN REPLACEMENTS FOR 3-METHYLISOXZOLES - ARE 2-ACETYLFURANS BIOISOSTERES FOR 3-METHYLISOXAZOLES (VOL 37, PG 4179, 1994)
Authors: BAILEY TR DIANA GD MALLAMO JP VESCIO N DRAPER TL CARABATEAS PM LONG MA GIRANDA VL DUTKO FJ PEVEAR DC
Citation: Tr. Bailey et al., AN EVALUATION OF THE ANTIRHINOVIRAL ACTIVITY OF ACYLFURAN REPLACEMENTS FOR 3-METHYLISOXZOLES - ARE 2-ACETYLFURANS BIOISOSTERES FOR 3-METHYLISOXAZOLES (VOL 37, PG 4179, 1994), Journal of medicinal chemistry, 38(8), 1995, pp. 1416-1416
NOVEL BENZO[B]QUINOLIZINIUM CATIONS AS UNCOMPETITIVE N-METHYL-D-ASPARTIC ACID (NMDA) ANTAGONISTS - THE RELATIONSHIP BETWEEN LOG-D AND AGONIST INDEPENDENT (CLOSED) NMDA CHANNEL BLOCK
Authors: EARLEY WG KUMAR V MALLAMO JP SUBRAMANYAM C DORITY JA MILLER MS DEHAVENHUDKINS DL AIMONE LD KELLY MD AULT B
Citation: Wg. Earley et al., NOVEL BENZO[B]QUINOLIZINIUM CATIONS AS UNCOMPETITIVE N-METHYL-D-ASPARTIC ACID (NMDA) ANTAGONISTS - THE RELATIONSHIP BETWEEN LOG-D AND AGONIST INDEPENDENT (CLOSED) NMDA CHANNEL BLOCK, Journal of medicinal chemistry, 38(18), 1995, pp. 3586-3592
SYNTHESIS AND EVALUATION OF 6,11-ETHANOHEXAHYDROBENZO[B]QUINOLIZIDINES - A NEW CLASS OF NONCOMPETITIVE N-METHYL-D-ASPARTATE ANTAGONISTS
Authors: SUBRAMANYAM C MALLAMO JP PILLING GM EARLEY WG CARABATEAS PM WETZEL JR DEHAVENHUDKINS D ALLEN T KULLNIG RK
Citation: C. Subramanyam et al., SYNTHESIS AND EVALUATION OF 6,11-ETHANOHEXAHYDROBENZO[B]QUINOLIZIDINES - A NEW CLASS OF NONCOMPETITIVE N-METHYL-D-ASPARTATE ANTAGONISTS, Journal of medicinal chemistry, 38(13), 1995, pp. 2483-2489
NOVEL NMDA ANTAGONISTS - REPLACEMENT OF THE PYRIDINIUM RING OF 6,11-ETHANOBENZO[B]QUINOLIZINIUM CATIONS WITH HETEROISOQUINOLINIUM CATIONS
Authors: KUMAR V CARABATEAS PM DORITY JA EARLEY WG MALLAMO JP SUBRAMANYAM C AIMONE LD AULT B HUDKINS DLD MILLER MS
Citation: V. Kumar et al., NOVEL NMDA ANTAGONISTS - REPLACEMENT OF THE PYRIDINIUM RING OF 6,11-ETHANOBENZO[B]QUINOLIZINIUM CATIONS WITH HETEROISOQUINOLINIUM CATIONS, Journal of medicinal chemistry, 38(10), 1995, pp. 1826-1830
DISCOVERY OF ANO-12,12-DIARYL-6,11-DIHYDROBENZO[B]QUINOLIZINIUM CATIONS, A NOVEL CLASS OF N-METHYL-D-ASPARTATE ANTAGONISTS
Authors: SUBRAMANYAM C MALLAMO JP DORITY JA EARLEY WG KUMAR V AIMONE LD AULT B MILLER MS LUTTINGER DA DEHAVENHUDKINS DL
Citation: C. Subramanyam et al., DISCOVERY OF ANO-12,12-DIARYL-6,11-DIHYDROBENZO[B]QUINOLIZINIUM CATIONS, A NOVEL CLASS OF N-METHYL-D-ASPARTATE ANTAGONISTS, Journal of medicinal chemistry, 38(1), 1995, pp. 21-27
IDENTIFICATION, SYNTHESIS, AND CHARACTERIZATION OF A UNIQUE CLASS OF N-METHYL-D-ASPARTATE ANTAGONISTS - THE 6,11-ETHANOBENZO[B]QUINOLIZINIUM CATION
Authors: MALLAMO JP EARLEY WG KUMAR V SUBRAMANYAM C DORITY JA MILLER MS DEHAVENHUDKINS DL AULT B HERRMANN JL DUNG JS MCMULLEN LA JAEGER E KULLNIG R MAGEE LJ
Citation: Jp. Mallamo et al., IDENTIFICATION, SYNTHESIS, AND CHARACTERIZATION OF A UNIQUE CLASS OF N-METHYL-D-ASPARTATE ANTAGONISTS - THE 6,11-ETHANOBENZO[B]QUINOLIZINIUM CATION, Journal of medicinal chemistry, 37(26), 1994, pp. 4438-4448
AN EVALUATION OF THE ANTIRHINOVIRAL ACTIVITY OF ACYLFURAN REPLACEMENTS FOR 3-METHYLISOXAZOLES - ARE 2-ACETYLFURANS BIOISOSTERES FOR 3-METHYLISOXAZOLES
Authors: BAILEY TR DIANA GD MALLAMO JP VESCIO N DRAPER TL CARABATEAS PM LONG MA GIRANDA VL DUTKO FJ PEVEAR DC
Citation: Tr. Bailey et al., AN EVALUATION OF THE ANTIRHINOVIRAL ACTIVITY OF ACYLFURAN REPLACEMENTS FOR 3-METHYLISOXAZOLES - ARE 2-ACETYLFURANS BIOISOSTERES FOR 3-METHYLISOXAZOLES, Journal of medicinal chemistry, 37(24), 1994, pp. 4177-4184
ANTIPICORNAVIRUS ACTIVITY OF TETRAZOLE ANALOGS RELATED TO DISOXARIL
Authors: DIANA GD CUTCLIFFE D VOLKOTS DL MALLAMO JP BAILEY TR VESCIO N OGLESBY RC NITZ TJ WETZEL J GIRANDA V PEVEAR DC DUTKO FJ
Citation: Gd. Diana et al., ANTIPICORNAVIRUS ACTIVITY OF TETRAZOLE ANALOGS RELATED TO DISOXARIL, Journal of medicinal chemistry, 36(22), 1993, pp. 3240-3250
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