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Results: 1-22 |
Results: 22
3-[2-(PYRROLIDIN-1-YL)ETHYL]INDOLES AND 3-[3-(PIPERIDIN-1-YL)PROPYL]INDOLES - AGONISTS FOR THE H5-HT1D RECEPTOR WITH HIGH SELECTIVITY OVER THE H5-HT1B SUBTYPE
Authors: CASTRO JL STREET LJ GUIBLIN AR JELLEY RA RUSSELL MGN STERNFELD F BEER MS STANTON JA MATASSA VG
Citation: Jl. Castro et al., 3-[2-(PYRROLIDIN-1-YL)ETHYL]INDOLES AND 3-[3-(PIPERIDIN-1-YL)PROPYL]INDOLES - AGONISTS FOR THE H5-HT1D RECEPTOR WITH HIGH SELECTIVITY OVER THE H5-HT1B SUBTYPE, Journal of medicinal chemistry, 40(22), 1997, pp. 3497-3500
SELECTIVE, ORALLY-ACTIVE 5-HT1D RECEPTOR AGONISTS AS POTENTIAL ANTIMIGRAINE AGENTS
Authors: MACLEOD AM STREET LJ REEVE AJ JELLEY RA STERNFELD F BEER MS STANTON JA WATT AP RATHBONE D MATASSA VG
Citation: Am. Macleod et al., SELECTIVE, ORALLY-ACTIVE 5-HT1D RECEPTOR AGONISTS AS POTENTIAL ANTIMIGRAINE AGENTS, Journal of medicinal chemistry, 40(22), 1997, pp. 3501-3503
5-(PIPERIDIN-2-YL)-1,4-BENZODIAZEPINES AND 5-(HOMOPIPERIDIN-2-YL)-1,4-BENZODIAZEPINES - HIGH-AFFINITY, BASIC LIGANDS FOR THE CHOLECYSTOKININ-B RECEPTOR
Authors: CASTRO JL BROUGHTON HB RUSSELL MGN RATHBONE D WATT AP BALL RG CHAPMAN KL PATEL S SMITH AJ MARSHALL GR MATASSA VG
Citation: Jl. Castro et al., 5-(PIPERIDIN-2-YL)-1,4-BENZODIAZEPINES AND 5-(HOMOPIPERIDIN-2-YL)-1,4-BENZODIAZEPINES - HIGH-AFFINITY, BASIC LIGANDS FOR THE CHOLECYSTOKININ-B RECEPTOR, Journal of medicinal chemistry, 40(16), 1997, pp. 2491-2501
L-743,345 - THE C5-(3-AZABICYCLO[3.2.2.]NONAN-3-YL) ANALOG OF DEVAZEPIDE, A SELECTIVE, HIGH-AFFINITY ANTAGONIST FOR THE CHOLECYSTOKININ-A RECEPTOR
Authors: SHOWELL GA BOURRAIN S NEDUVELIL JG MATASSA VG MATHESON S PATEL S SMITH AJ CHAPMAN KL MARQUISOMER D BALL RG
Citation: Ga. Showell et al., L-743,345 - THE C5-(3-AZABICYCLO[3.2.2.]NONAN-3-YL) ANALOG OF DEVAZEPIDE, A SELECTIVE, HIGH-AFFINITY ANTAGONIST FOR THE CHOLECYSTOKININ-A RECEPTOR, Medicinal chemistry research, 6(5), 1996, pp. 312-317
THE CHEMICAL EVOLUTION OF 2-[5-(1,2,4-TRIAZOL-4-YL)-1H-INDOL-3-YL]ETHYLAMINE (L-741,604) AND ANALOGS - POTENT AND SELECTIVE AGONISTS FOR 5-HT1D RECEPTORS
Authors: STERNFELD F BAKER R BROUGHTON HB GUIBLIN AR JELLEY RA MATASSA VG REEVE AJ BEER MS STANTON JA HARGREAVES RJ SHEPHEARD SL LONGMORE J RAZZAQUE Z GRAHAM MI SOHAL B STREET LJ
Citation: F. Sternfeld et al., THE CHEMICAL EVOLUTION OF 2-[5-(1,2,4-TRIAZOL-4-YL)-1H-INDOL-3-YL]ETHYLAMINE (L-741,604) AND ANALOGS - POTENT AND SELECTIVE AGONISTS FOR 5-HT1D RECEPTORS, Bioorganic & medicinal chemistry letters, 6(15), 1996, pp. 1825-1830
CONTROLLED MODIFICATION OF ACIDITY IN CHOLECYSTOKININ B RECEPTOR ANTAGONISTS - ZEPIN-3-YL)-N'-[3-(TETRAZOL-5-YLAMINO)PHENYL]UREAS
Authors: CASTRO JL BALL RG BROUGHTON HB RUSSELL MGN RATHBONE D WATT AP BAKER R CHAPMAN KL FLETCHER AE PATEL S SMITH AJ MARSHALL GR RYECROFT W MATASSA VG
Citation: Jl. Castro et al., CONTROLLED MODIFICATION OF ACIDITY IN CHOLECYSTOKININ B RECEPTOR ANTAGONISTS - ZEPIN-3-YL)-N'-[3-(TETRAZOL-5-YLAMINO)PHENYL]UREAS, Journal of medicinal chemistry, 39(4), 1996, pp. 842-849
IN-VITRO PHARMACOLOGICAL EFFECTS OF 2 NOVEL 5-HT1D-RECEPTOR AGONISTS L-741,519 AND L-741,604 - COMPARISON WITH SUMATRIPTAN AND BW311C
Authors: RAZZAQUE Z BAKER R BEER MS HILL RG MATASSA VG STAGG AT STERNFELD F STREET L LONGMORE J
Citation: Z. Razzaque et al., IN-VITRO PHARMACOLOGICAL EFFECTS OF 2 NOVEL 5-HT1D-RECEPTOR AGONISTS L-741,519 AND L-741,604 - COMPARISON WITH SUMATRIPTAN AND BW311C, British Journal of Pharmacology, 117, 1996, pp. 119-119
C5-PIPERAZINYL-1,4-BENZODIAZEPINES, WATER-SOLUBLE, ORALLY BIOAVAILABLE CCKB GASTRIN RECEPTOR ANTAGONISTS
Authors: SHOWELL GA BOURRAIN S FLETCHER SR NEDUVELIL JG FLETCHER AE FREEDMAN SB PATEL S SMITH AJ MARSHALL GR GRAHAM MI SOHAL B MATASSA VG
Citation: Ga. Showell et al., C5-PIPERAZINYL-1,4-BENZODIAZEPINES, WATER-SOLUBLE, ORALLY BIOAVAILABLE CCKB GASTRIN RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 5(24), 1995, pp. 3023-3026
POTENT, SELECTIVE, WATER-SOLUBLE BENZODIAZEPINE-BASED CCKB RECEPTOR ANTAGONISTS THAT CONTAIN LIPOPHILIC CARBOXYLATE SURROGATES
Authors: CHAMBERS MS HOBBS SC GRAHAM MI WATT AP FLETCHER SR BAKER R FREEDMAN SB PATEL S SMITH AJ MATASSA VG
Citation: Ms. Chambers et al., POTENT, SELECTIVE, WATER-SOLUBLE BENZODIAZEPINE-BASED CCKB RECEPTOR ANTAGONISTS THAT CONTAIN LIPOPHILIC CARBOXYLATE SURROGATES, Bioorganic & medicinal chemistry letters, 5(20), 1995, pp. 2303-2308
CCKB SELECTIVE RECEPTOR LIGANDS - NOVEL 1,3,5-TRISUBSTITUTED BENZAZEPIN-2-ONES
Authors: VANNIEL MB FREEDMAN SB MATASSA VG PATEL S PENGILLEY RR SMITH AJ
Citation: Mb. Vanniel et al., CCKB SELECTIVE RECEPTOR LIGANDS - NOVEL 1,3,5-TRISUBSTITUTED BENZAZEPIN-2-ONES, Bioorganic & medicinal chemistry letters, 5(13), 1995, pp. 1421-1426
IN-VITRO STUDIES OF THE OXIDATIVE-METABOLISM OF L-737,415, A C5-CYCLOALKYLAMINE-1,4-BENZODIAZEPIN-2-ONE CCKB RECEPTOR ANTAGONIST
Authors: WATT AP OCONNOR D THOMAS S HERBERT RH MATASSA VG
Citation: Ap. Watt et al., IN-VITRO STUDIES OF THE OXIDATIVE-METABOLISM OF L-737,415, A C5-CYCLOALKYLAMINE-1,4-BENZODIAZEPIN-2-ONE CCKB RECEPTOR ANTAGONIST, Journal of liquid chromatography, 18(11), 1995, pp. 2271-2282
SYNTHESIS AND SEROTONERGIC ACTIVITY OF HYL-2-[5-(1,2,4-TRIAZOL-1-YLMETHYL)-1H-INDOL-3-YL] ETHYLAMINE AND ANALOGS - POTENT AGONISTS FOR 5-HT1D RECEPTORS
Authors: STREET LJ BAKER R DAVEY WB GUIBLIN AR JELLEY RA REEVE AJ ROUTLEDGE H STERNFELD F WATT AP BEER MS MIDDLEMISS DN NOBLE AJ STANTON JA SCHOLEY K HARGREAVES RJ SOHAL B GRAHAM MI MATASSA VG
Citation: Lj. Street et al., SYNTHESIS AND SEROTONERGIC ACTIVITY OF HYL-2-[5-(1,2,4-TRIAZOL-1-YLMETHYL)-1H-INDOL-3-YL] ETHYLAMINE AND ANALOGS - POTENT AGONISTS FOR 5-HT1D RECEPTORS, Journal of medicinal chemistry, 38(10), 1995, pp. 1799-1810
SYNTHESIS AND SEROTONERGIC ACTIVITY OF BENZOFURAN AND DIHYDROBENZOFURAN ANALOGS OF 5-CARBOXAMIDOTRYPTAMINE
Authors: RUSSELL MGN CASTRO JL MATASSA VG BEER MS HEALD A SCHOLEY K STANTON JA BROUGHTON HB
Citation: Mgn. Russell et al., SYNTHESIS AND SEROTONERGIC ACTIVITY OF BENZOFURAN AND DIHYDROBENZOFURAN ANALOGS OF 5-CARBOXAMIDOTRYPTAMINE, Bioorganic & medicinal chemistry letters, 4(10), 1994, pp. 1207-1212
BIOLOGICAL PROPERTIES OF THE BENZODIAZEPINE AMIDINE DERIVATIVE L-740,093, A CHOLECYSTOKININ-B GASTRIN RECEPTOR ANTAGONIST WITH HIGH-AFFINITY IN-VITRO AND HIGH POTENCY IN-VIVO
Authors: PATEL S SMITH AJ CHAPMAN KL FLETCHER AE KEMP JA MARSHALL GR HARGREAVES RJ RYECROFT W IVERSEN LL IVERSEN SD BAKER R SHOWELL GA BOURRAIN S NEDUVELIL JG MATASSA VG FREEDMAN SB
Citation: S. Patel et al., BIOLOGICAL PROPERTIES OF THE BENZODIAZEPINE AMIDINE DERIVATIVE L-740,093, A CHOLECYSTOKININ-B GASTRIN RECEPTOR ANTAGONIST WITH HIGH-AFFINITY IN-VITRO AND HIGH POTENCY IN-VIVO, Molecular pharmacology, 46(5), 1994, pp. 943-948
MITSUNOBU-LIKE PROCESSES WITH A NOVEL TRIPHENYLPHOSPHINE-CYCLIC SULFAMIDE BETAINE
Authors: CASTRO JL MATASSA VG BALL RG
Citation: Jl. Castro et al., MITSUNOBU-LIKE PROCESSES WITH A NOVEL TRIPHENYLPHOSPHINE-CYCLIC SULFAMIDE BETAINE, Journal of organic chemistry, 59(9), 1994, pp. 2289-2291
HIGH-AFFINITY AND POTENT, WATER-SOLUBLE 5-AMINO-1,4-BENZODIAZEPINE CCK(B) GASTRIN RECEPTOR ANTAGONISTS CONTAINING A CATIONIC SOLUBILIZING GROUP
Authors: SHOWELL GA BOURRAIN S NEDUVELIL JG FLETCHER SR BAKER R WATT AP FLETCHER AE FREEDMAN SB KEMP JA MARSHALL GR PATEL S SMITH AJ MATASSA VG
Citation: Ga. Showell et al., HIGH-AFFINITY AND POTENT, WATER-SOLUBLE 5-AMINO-1,4-BENZODIAZEPINE CCK(B) GASTRIN RECEPTOR ANTAGONISTS CONTAINING A CATIONIC SOLUBILIZING GROUP, Journal of medicinal chemistry, 37(6), 1994, pp. 719-721
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF ETHYL-1,2,5-THIADIAZOLIDIN-2-YL)-METHYL]-1H-INDOLE AND ANALOGS - AGONISTS FOR THE 5-HT1D RECEPTOR
Authors: CASTRO JL BAKER R GUIBLIN AR HOBBS SC JENKINS MR RUSSELL MGN BEER MS STANTON JA SCHOLEY K HARGREAVES RJ GRAHAM MI MATASSA VG
Citation: Jl. Castro et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF ETHYL-1,2,5-THIADIAZOLIDIN-2-YL)-METHYL]-1H-INDOLE AND ANALOGS - AGONISTS FOR THE 5-HT1D RECEPTOR, Journal of medicinal chemistry, 37(19), 1994, pp. 3023-3032
SYNTHESIS, BIOLOGICAL-ACTIVITY AND ELECTROSTATIC PROPERTIES OF [(3-AMINO-1,2,4-THIADIAZOL-5-YL)METHYL]-1H-INDOLE, A NOVEL 5-HT1D RECEPTOR AGONIST
Authors: CASTRO JL MATASSA VG BROUGHTON HB MOSLEY RT STREET LJ BAKER R
Citation: Jl. Castro et al., SYNTHESIS, BIOLOGICAL-ACTIVITY AND ELECTROSTATIC PROPERTIES OF [(3-AMINO-1,2,4-THIADIAZOL-5-YL)METHYL]-1H-INDOLE, A NOVEL 5-HT1D RECEPTOR AGONIST, Bioorganic & medicinal chemistry letters, 3(6), 1993, pp. 993-997
L-708,474 - THE C5-CYCLOHEXYL ANALOG OF L-365,260, A SELECTIVE HIGH-AFFINITY LIGAND FOR THE CCK(B) GASTRIN RECEPTOR/
Authors: CHAMBERS MS HOBBS SC FLETCHER SR MATASSA VG MITCHELL PJ WATT AP BAKER R FREEDMAN SB PATEL S SMITH AJ
Citation: Ms. Chambers et al., L-708,474 - THE C5-CYCLOHEXYL ANALOG OF L-365,260, A SELECTIVE HIGH-AFFINITY LIGAND FOR THE CCK(B) GASTRIN RECEPTOR/, Bioorganic & medicinal chemistry letters, 3(10), 1993, pp. 1919-1924
METHIODIDE APPROACH TO THE SYNTHESIS OF METHYL-1,2,5-THIADIAZOLIDIN-2-YL)METHYL]-1H-INDOLE AND ANALOGS
Authors: CASTRO JL MATASSA VG
Citation: Jl. Castro et Vg. Matassa, METHIODIDE APPROACH TO THE SYNTHESIS OF METHYL-1,2,5-THIADIAZOLIDIN-2-YL)METHYL]-1H-INDOLE AND ANALOGS, Tetrahedron letters, 34(29), 1993, pp. 4705-4708
SYNTHESIS AND SEROTONERGIC ACTIVITY OF 5-(OXADIAZOLYL)TRYPTAMINES - POTENT AGONISTS FOR 5-HT(1D) RECEPTORS
Authors: STREET LJ BAKER R CASTRO JL CHAMBERS MS GUIBLIN AR HOBBS SC MATASSA VG REEVE AJ BEER MS MIDDLEMISS DN NOBLE AJ STANTON JA SCHOLEY K HARGREAVES RJ
Citation: Lj. Street et al., SYNTHESIS AND SEROTONERGIC ACTIVITY OF 5-(OXADIAZOLYL)TRYPTAMINES - POTENT AGONISTS FOR 5-HT(1D) RECEPTORS, Journal of medicinal chemistry, 36(11), 1993, pp. 1529-1538
L-694,247 - A POTENT 5-HT(1D) RECEPTOR AGONIST
Authors: BEER MS STANTON JA BEVAN Y HEALD A REEVE AJ STREET LJ MATASSA VG HARGREAVES RJ MIDDLEMISS DN
Citation: Ms. Beer et al., L-694,247 - A POTENT 5-HT(1D) RECEPTOR AGONIST, British Journal of Pharmacology, 110(3), 1993, pp. 1196-1200
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