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Results: 1-25/26
Authors:
MINARINI A
BUDRIESI R
CHIARINI A
LEONARDI A
MELCHIORRE C
Citation: A. Minarini et al., SEARCH FOR ALPHA(1)-ADRENOCEPTOR SUBTYPES SELECTIVE ANTAGONISTS - DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CYSTAZOSIN, AN ALPHA(1D)-ADRENOCEPTOR ANTAGONIST, Bioorganic & medicinal chemistry letters, 8(11), 1998, pp. 1353-1358
Authors:
BOLOGNESI ML
BUDRIESI R
CHIARINI A
POGGESI E
LEONARDI A
MELCHIORRE C
Citation: Ml. Bolognesi et al., DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF PRAZOSIN-RELATED ANTAGONISTS - ROLE OF THE PIPERAZINE AND FURAN UNITS OF PRAZOSIN ON THE SELECTIVITY FOR ALPHA(1)-ADRENORECEPTOR SUBTYPES, Journal of medicinal chemistry, 41(24), 1998, pp. 4844-4853
Authors:
MELCHIORRE C
ANDRISANO V
BOLOGNESI ML
BUDRIESI R
CAVALLI A
CAVRINI V
ROSINI M
TUMIATTI V
RECANATINI M
Citation: C. Melchiorre et al., ACETYLCHOLINESTERASE NONCOVALENT INHIBITORS BASED ON A POLYAMINE BACKBONE FOR POTENTIAL USE AGAINST ALZHEIMERS-DISEASE, Journal of medicinal chemistry, 41(22), 1998, pp. 4186-4189
UNIVERSAL TEMPLATE APPROACH TO DRUG DESIGN - POLYAMINES AS SELECTIVE MUSCARINIC RECEPTOR ANTAGONISTS
Authors:
BOLOGNESI ML
MINARINI A
BUDRIESI R
CACCIAGUERRA S
CHIARINI A
SPAMPINATO S
TUMIATTI V
MELCHIORRE C
Citation: Ml. Bolognesi et al., UNIVERSAL TEMPLATE APPROACH TO DRUG DESIGN - POLYAMINES AS SELECTIVE MUSCARINIC RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 41(21), 1998, pp. 4150-4160
Authors:
QUAGLIA W
GIANNELLA M
PIERGENTILI A
PIGINI M
BRASILI L
DITORO R
ROSSETTI L
SPAMPINATO S
MELCHIORRE C
Citation: W. Quaglia et al., -DIHYDROSPIRO[2H-1-BENZOTHIOPYRAN-2,4'-PIPERIDINE] (SPIPETHIANE), A POTENT AND HIGHLY SELECTIVE SIGMA(1) LIGAND, Journal of medicinal chemistry, 41(10), 1998, pp. 1557-1560
Authors:
MELCHIORRE C
BOLOGNESI ML
BUDRIESI R
CHIARINI A
GIARDINA D
MINARINI A
QUAGLIA W
LEONARDI A
Citation: C. Melchiorre et al., SEARCH FOR SELECTIVE ANTAGONISTS AT ALPHA(1)-ADRENORECEPTORS - NEUTRAL OR NEGATIVE ANTAGONISM, Il Farmaco, 53(4), 1998, pp. 278-286
Authors:
BARBIER P
COLELLI A
BOLOGNESI ML
MINARINI A
TUMIATTI V
CORSINI GU
MELCHIORRE C
MAGGIO R
Citation: P. Barbier et al., ANTAGONIST BINDING PROFILE OF THE SPLIT CHIMERIC MUSCARINIC M2-TRUNC M3-TAIL RECEPTOR/, European journal of pharmacology, 355(2-3), 1998, pp. 267-274
Authors:
GIARDINA D
CRUCIANELLI M
MARUCCI G
ANGELI P
MELCHIORRE C
ANTOLINI L
Citation: D. Giardina et al., SYNTHESIS AND ALPHA-ADRENOCEPTOR BLOCKING ACTIVITY OF THE ENANTIOMERSOF ROETHYL)-[2-(2-METHOXYPHENOXY)-1-METHYLETHYL]AMINE HYDROCHLORIDE, Bioorganic & medicinal chemistry, 5(9), 1997, pp. 1775-1782
Authors:
GIARDINA D
CRUCIANELLI M
GULINI U
MARUCCI G
MELCHIORRE C
SPAMPINATO S
Citation: D. Giardina et al., SYNTHESIS AND ALPHA(1)-ANTAGONIST ACTIVITY OF NEW PRAZOSIN-RELATED AND BENEXTRAMINE-RELATED TETRAAMINE DISULFIDES, European journal of medicinal chemistry, 32(1), 1997, pp. 9-20
Authors:
GIARDINA D
CRUCIANELLI M
ROMANELLI R
LEONARDI A
POGGESI E
MELCHIORRE C
Citation: D. Giardina et al., SYNTHESIS AND BIOLOGICAL PROFILE OF THE ENANTIOMERS OF HOXYQUINAZOLIN-2-YL)-CIS-OCTAHYDROQUINOXALIN-1-YL] FURAN-2-YLMETHANONE (CYCLAZOSIN),A POTENT COMPETITIVE ALPHA(1B)-ADRENOCEPTOR ANTAGONIST, Journal of medicinal chemistry, 39(23), 1996, pp. 4602-4607
Authors:
QUAGLIA W
PIGINI M
TAYEBATI SK
PIERGENTILI A
GIANNELLA M
LEONARDI A
TADDEI C
MELCHIORRE C
Citation: W. Quaglia et al., SYNTHESIS, ABSOLUTE-CONFIGURATION, AND BIOLOGICAL PROFILE OF THE ENANTIOMERS OF OLYL-2,3-DIHYDRO-1,4-BENZODIOXIN-2-YL)METHYL]AMINE (MEPHENDIOXAN), A POTENT COMPETITIVE ALPHA(1A)-ADRENOCEPTOR ANTAGONIST, Journal of medicinal chemistry, 39(11), 1996, pp. 2253-2258
Authors:
QUAGLIA W
GIANNELLA M
MARUCCI G
PIERGENTILI A
PIGINI M
TAYEBATI SK
MELCHIORRE C
Citation: W. Quaglia et al., STRUCTURE-ACTIVITY-RELATIONSHIPS IN 1,4-BENZODIOXAN-RELATED COMPOUNDS.5. EFFECTS OF MODIFICATION OF THE SIDE-CHAIN ON ALPHA-ADRENOCEPTOR BLOCKING ACTIVITY, Il Farmaco, 51(1), 1996, pp. 27-32
Authors:
GIARDINA D
CRUCIANELLI M
MARUCCI G
MELCHIORRE C
POLIDORI C
POMPEI P
MASSI M
Citation: D. Giardina et al., PHARMACOLOGICAL EVALUATION OF PRAZOSIN-RELATED AND DOXAZOSIN-RELATED COMPOUNDS WITH MODIFIED PIPERAZINE RING, Arzneimittel-Forschung, 46(11), 1996, pp. 1054-1059
Authors:
MELCHIORRE C
MINARINI A
SPAMPINATO S
TUMIATTI V
Citation: C. Melchiorre et al., DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME TETRAAMINES RELATEDTO METHOCTRAMINE AND 4-DAMP, Bioorganic & medicinal chemistry letters, 5(8), 1995, pp. 785-790
Authors:
TUMIATTI V
SPAMPINATO S
RECANATINI M
MINARINI A
MELCHIORRE C
CHIARINI A
BUDRIESI R
Citation: V. Tumiatti et al., DESIGN, SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME 4-DAMP-RELATED COMPOUNDS, Bioorganic & medicinal chemistry letters, 5(20), 1995, pp. 2325-2330
Authors:
ANGELI P
CANTALAMESSA F
GULINI U
MELCHIORRE C
Citation: P. Angeli et al., SELECTIVE BLOCKADE OF MUSCARINIC M(2) RECEPTORS IN-VIVO BY THE NEW ANTAGONIST TRIPITRAMINE, Naunyn-Schmiedeberg's archives of pharmacology, 352(3), 1995, pp. 304-307
Authors:
MELCHIORRE C
MINARINI A
BUDRIESI R
CHIARINI A
SPAMPINATO S
TUMIATTI V
Citation: C. Melchiorre et al., THE DESIGN OF NOVEL METHOCTRAMINE-RELATED TETRAAMINES AS MUSCARINIC RECEPTOR SUBTYPE-SELECTIVE ANTAGONISTS, Life sciences, 56(11-12), 1995, pp. 837-844
Authors:
CANTALAMESSA F
ANGELI P
MELCHIORRE C
Citation: F. Cantalamessa et al., TRIPITRAMINE - FURTHER PHARMACOLOGICAL EVALUATION IN PITHED RAT, Life sciences, 56(11-12), 1995, pp. 1012-1012
Authors:
GIARDINA D
CRUCIANELLI M
MELCHIORRE C
TADDEI C
TESTA R
Citation: D. Giardina et al., RECEPTOR-BINDING PROFILE OF CYCLAZOSIN, A NEW ALPHA(1B)-ADRENOCEPTOR ANTAGONIST, European journal of pharmacology, 287(1), 1995, pp. 13-16
Authors:
CHIARINI A
BUDRIESI R
BOLOGNESI ML
MINARINI A
MELCHIORRE C
Citation: A. Chiarini et al., IN-VITRO CHARACTERIZATION OF TRIPITRAMINE, A POLYMETHYLENE TETRAAMINEDISPLAYING HIGH SELECTIVITY AND AFFINITY FOR MUSCARINIC M(2) RECEPTORS, British Journal of Pharmacology, 114(7), 1995, pp. 1507-1517
Authors:
MAGGIO R
BARBIER P
BOLOGNESI ML
MINARINI A
TEDESCHI D
MELCHIORRE C
Citation: R. Maggio et al., BINDING PROFILE OF THE SELECTIVE MUSCARINIC RECEPTOR ANTAGONIST TRIPITRAMINE, European journal of pharmacology. Molecular pharmacology section, 268(3), 1994, pp. 459-462
Authors:
SABATINO P
RECANATINI M
TUMIATTI V
MELCHIORRE C
Citation: P. Sabatino et al., STRUCTURAL STUDIES ON THE ANTIMUSCARINIC AGENTS SPIRO-DAMP AND HYDROXY-DAMP, AND COMPARISON WITH RELATED-COMPOUNDS, Acta crystallographica. Section C, Crystal structure communications, 50, 1994, pp. 640-645
Authors:
MINARINI A
BOLOGNESI ML
BUDRIESI R
CANOSSA M
CHIARINI A
SPAMPINATO S
MELCHIORRE C
Citation: A. Minarini et al., DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF METHOCTRAMINE-RELATED TETRAAMINES BEARING AN 1-DIHYDRO-6H-PYRIDO[2,3-B][1,4]BENZODIAZEPIN-6-ONE MOIETY - STRUCTURAL REQUIREMENTS FOR OPTIMUM OCCUPANCY OF MUSCARINIC RECEPTOR SUBTYPES AS REVEALED BY SYMMETRICAL AND UNSYMMETRICAL POLYAMINES, Journal of medicinal chemistry, 37(20), 1994, pp. 3363-3372
Authors:
MELCHIORRE C
ROMUALDI P
BOLOGNESI ML
DONATINI A
FERRI S
Citation: C. Melchiorre et al., BINDING PROFILE OF BENEXTRAMINE AT NEUROPEPTIDE-Y RECEPTOR SUBTYPES IN RAT-BRAIN AREAS, European journal of pharmacology, 265(1-2), 1994, pp. 93-98
Authors:
MELCHIORRE C
BOLOGNESI ML
CHIARINI A
MINARINI A
SPAMPINATO S
Citation: C. Melchiorre et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SOME METHOCTRAMINE-RELATED TETRAAMINES BEARING A -DIHYDRO-6H-PYRIDO[2,3-B][1,4]-BENZODIAZEPIN-6-ONE MOIETY AS ANTIMUSCARINICS - A 2ND-GENERATION OF HIGHLY SELECTIVE M(2)-MUSCARINIC RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 36(23), 1993, pp. 3734-3737