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Results: 1-11 |
Results: 11
Synthesis and progesterone receptor antagonist activities of 6-aryl benzimidazolones and benzothiazolones
Authors: Zhang, PW Terefenko, EA Wrobel, J Zhang, ZM Zhu, Y Cohen, J Marschke, KB Mais, D
Citation: Pw. Zhang et al., Synthesis and progesterone receptor antagonist activities of 6-aryl benzimidazolones and benzothiazolones, BIOORG MED, 11(20), 2001, pp. 2747-2750
Effects of isosteric pyridone replacements in androgen receptor antagonists based on 1,2-dihydro- and 1,2,3,4-tetrahydro-2,2-dimethyl-6-trifluoromethyl-8-pyridono[5,6-g]quinolines
Authors: Kong, JW Hamann, LG Ruppar, DA Edwards, JP Marschke, KB Jones, TK
Citation: Jw. Kong et al., Effects of isosteric pyridone replacements in androgen receptor antagonists based on 1,2-dihydro- and 1,2,3,4-tetrahydro-2,2-dimethyl-6-trifluoromethyl-8-pyridono[5,6-g]quinolines, BIOORG MED, 10(5), 2000, pp. 411-414
Nonsteroidal progesterone receptor antagonists based on 6-thiophenehydroquinolines
Authors: Zhi, L Tegley, CM Pio, B West, SJ Marschke, KB Mais, DE Jones, TK
Citation: L. Zhi et al., Nonsteroidal progesterone receptor antagonists based on 6-thiophenehydroquinolines, BIOORG MED, 10(5), 2000, pp. 415-418
Novel class of non-steroidal progesterone receptor antagonists
Authors: Zhi, L Marschke, KB
Citation: L. Zhi et Kb. Marschke, Novel class of non-steroidal progesterone receptor antagonists, EXPERT OP T, 9(6), 1999, pp. 695-700
4-alkyl- and 3,4-dialkyl-1,2,3,4-tetrahydro-8-pyridono [5,6-g]quinolines: Potent, nonsteroidal androgen receptor agonists
Authors: Higuchi, RI Edwards, JP Caferro, TR Ringgenberg, JD Kong, JW Hamann, LG Arienti, KL Marschke, KB Davis, RL Farmer, LJ Jones, TK
Citation: Ri. Higuchi et al., 4-alkyl- and 3,4-dialkyl-1,2,3,4-tetrahydro-8-pyridono [5,6-g]quinolines: Potent, nonsteroidal androgen receptor agonists, BIOORG MED, 9(9), 1999, pp. 1335-1340
Nonsteroidal androgen receptor agonists based on 4-(trifluoromethyl)-2H-pyrano[3,2-g]quinolin-2-one
Authors: Edwards, JP Higuchi, RI Winn, DT Pooley, CLF Caferro, TR Hamann, LG Zhi, L Marschke, KB Goldman, ME Jones, TK
Citation: Jp. Edwards et al., Nonsteroidal androgen receptor agonists based on 4-(trifluoromethyl)-2H-pyrano[3,2-g]quinolin-2-one, BIOORG MED, 9(7), 1999, pp. 1003-1008
Switching androgen receptor antagonists to agonists by modifying C-ring substituents on piperidino[3,2-g]quinolinone
Authors: Zhi, L Tegley, CM Marschke, KB Jones, TK
Citation: L. Zhi et al., Switching androgen receptor antagonists to agonists by modifying C-ring substituents on piperidino[3,2-g]quinolinone, BIOORG MED, 9(7), 1999, pp. 1009-1012
Estrogen receptor beta activates the human retinoic acid receptor alpha-1 promoter in response to tamoxifen and other estrogen receptor antagonists, but not in response to estrogen
Authors: Zou, AH Marschke, KB Arnold, KE Berger, EM Fitzgerald, P Mais, DE Allegretto, EA
Citation: Ah. Zou et al., Estrogen receptor beta activates the human retinoic acid receptor alpha-1 promoter in response to tamoxifen and other estrogen receptor antagonists, but not in response to estrogen, MOL ENDOCR, 13(3), 1999, pp. 418-430
5-aryl-1,2,3,4-tetrahydrochromeno[3,4-f]quinolin-3-ones as a novel class of nonsteroidal progesterone receptor agonists: Effect of A-ring modification
Authors: Zhi, L Tegley, CM Marschke, KB Mais, DE Jones, TK
Citation: L. Zhi et al., 5-aryl-1,2,3,4-tetrahydrochromeno[3,4-f]quinolin-3-ones as a novel class of nonsteroidal progesterone receptor agonists: Effect of A-ring modification, J MED CHEM, 42(8), 1999, pp. 1466-1472
Discovery of a potent, orally active, nonsteroidal androgen receptor agonist: 4-ethyl-1,2,3,4-tetrahydro-6(trifluoromethyl)-8-pyridono[5,6-g]-quinoline (LG121071)
Authors: Hamann, LG Mani, NS Davis, RL Wang, XN Marschke, KB Jones, TK
Citation: Lg. Hamann et al., Discovery of a potent, orally active, nonsteroidal androgen receptor agonist: 4-ethyl-1,2,3,4-tetrahydro-6(trifluoromethyl)-8-pyridono[5,6-g]-quinoline (LG121071), J MED CHEM, 42(2), 1999, pp. 210-212
5-alkyl 1,2-dihydrochromeno[3,4-f]quinolines: A novel class of nonsteroidal progesterone receptor modulators
Authors: Zhi, L Tegley, CM Edwards, JP West, SJ Marschke, KB Gottardis, MM Mais, DE Jones, TK
Citation: L. Zhi et al., 5-alkyl 1,2-dihydrochromeno[3,4-f]quinolines: A novel class of nonsteroidal progesterone receptor modulators, BIOORG MED, 8(23), 1998, pp. 3365-3370
Risultati: 1-11 |