AAAAAA

   
Results: 1-14 |
Results: 14
Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selectiveinhibitors of human 5 alpha-reductase 1
Authors: Guarna, A Occhiato, EG Machetti, F Trabocchi, A Scarpi, D Danza, G Mancina, R Comerci, A Serio, M
Citation: A. Guarna et al., Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selectiveinhibitors of human 5 alpha-reductase 1, BIO MED CH, 9(6), 2001, pp. 1385-1393
Introduction of the new dipeptide isostere 7-endo-BtA as reverse turn inducer in a Bowman-Birk proteinase inhibitor: Synthesis and conformational analysis
Authors: Scarpi, D Occhiato, EG Trabocchi, A Leatherbarrow, RJ Brauer, ABE Nievo, M Guarna, A
Citation: D. Scarpi et al., Introduction of the new dipeptide isostere 7-endo-BtA as reverse turn inducer in a Bowman-Birk proteinase inhibitor: Synthesis and conformational analysis, BIO MED CH, 9(6), 2001, pp. 1625-1632
Suzuki reaction of vinyl triflates from six- and seven-membered N-alkoxycarbonyl lactams with boronic acids and esters
Authors: Occhiato, EG Trabocchi, A Guarna, A
Citation: Eg. Occhiato et al., Suzuki reaction of vinyl triflates from six- and seven-membered N-alkoxycarbonyl lactams with boronic acids and esters, J ORG CHEM, 66(7), 2001, pp. 2459-2465
Pd(0)-catalyzed cross-coupling reactions of boron derivatives with a lactam-derived N-Boc enol triflate
Authors: Occhiato, EG Trabocchi, A Guama, A
Citation: Eg. Occhiato et al., Pd(0)-catalyzed cross-coupling reactions of boron derivatives with a lactam-derived N-Boc enol triflate, ORG LETT, 2(9), 2000, pp. 1241-1242
Oligomers of enantiopure bicyclic gamma/delta-amino acids (BTAa). 1. Synthesis and conformational analysis of 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid oligomers (PolyBTG)
Authors: Machetti, F Ferrali, A Menchi, G Occhiato, EG Guarna, A
Citation: F. Machetti et al., Oligomers of enantiopure bicyclic gamma/delta-amino acids (BTAa). 1. Synthesis and conformational analysis of 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid oligomers (PolyBTG), ORG LETT, 2(25), 2000, pp. 3987-3990
Synthesis of 8-chloro-benzo[c]quinolizin-3-ones as potent and selective inhibitors of human steroid 5 alpha-reductase 1
Authors: Guarna, A Occhiato, EG Scarpi, D Zorn, C Danza, G Comerci, A Mancina, R Serio, M
Citation: A. Guarna et al., Synthesis of 8-chloro-benzo[c]quinolizin-3-ones as potent and selective inhibitors of human steroid 5 alpha-reductase 1, BIOORG MED, 10(4), 2000, pp. 353-356
Stereoselective Meisenheimer rearrangement using BTAa's as chiral auxiliaries
Authors: Guarna, A Occhiato, EG Pizzetti, M Scarpi, D Sisi, S van Sterkenburg, M
Citation: A. Guarna et al., Stereoselective Meisenheimer rearrangement using BTAa's as chiral auxiliaries, TETRAHEDR-A, 11(20), 2000, pp. 4227-4238
Modification of the aza-Robinson annulation for the synthesis of 4-methyl-benzo[c]quinolizin-3-ones, potent inhibitors of steroid 5 alpha-reductase 1
Authors: Guarna, A Lombardi, E Machetti, F Occhiato, EG Scarpi, D
Citation: A. Guarna et al., Modification of the aza-Robinson annulation for the synthesis of 4-methyl-benzo[c]quinolizin-3-ones, potent inhibitors of steroid 5 alpha-reductase 1, J ORG CHEM, 65(23), 2000, pp. 8093-8095
Synthesis and reactivity of bicycles derived from tartaric acid and alpha-amino acids: A novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylicacid. (vol 64, pg 7358, 1995)
Authors: Guarna, A Guidi, A Machetti, F Menchi, G Occhiato, EG Scarpi, D Sisi, S Trabocch, A
Citation: A. Guarna et al., Synthesis and reactivity of bicycles derived from tartaric acid and alpha-amino acids: A novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylicacid. (vol 64, pg 7358, 1995), J ORG CHEM, 65(15), 2000, pp. 4782-4782
Benzo[c]quinolizin-3-ones: A novel class of potent and selective nonsteroidal inhibitors of human steroid 5 alpha-reductase
Authors: Guarna, A Machetti, G Occhiato, EG Scarpi, D Comerci, A Danza, G Mancina, R Serio, M Hardy, K
Citation: A. Guarna et al., Benzo[c]quinolizin-3-ones: A novel class of potent and selective nonsteroidal inhibitors of human steroid 5 alpha-reductase, J MED CHEM, 43(20), 2000, pp. 3718-3735
Lyophilised yeasts: easy-to-handle biocatalysts for stereoselective reduction of ketones
Authors: Molinari, F Gandolfi, R Villa, R Occhiato, EG
Citation: F. Molinari et al., Lyophilised yeasts: easy-to-handle biocatalysts for stereoselective reduction of ketones, TETRAHEDR-A, 10(18), 1999, pp. 3515-3520
A short and efficient route to enantiopure 3,5-diarylpyrrolizidines
Authors: Scarpi, D Occhiato, EG Guarna, A
Citation: D. Scarpi et al., A short and efficient route to enantiopure 3,5-diarylpyrrolizidines, J ORG CHEM, 64(5), 1999, pp. 1727-1732
Synthesis and reactivity of bicycles derived from tartaric acid and alpha-amino acids: A novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylicacid
Authors: Guarna, A Guidi, A Machetti, F Menchi, G Occhiato, EG Scarpi, D Sisi, S Trabocchi, A
Citation: A. Guarna et al., Synthesis and reactivity of bicycles derived from tartaric acid and alpha-amino acids: A novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylicacid, J ORG CHEM, 64(20), 1999, pp. 7347-7364
19-nor-10-azasteroids. 5. A synthetic strategy for the preparation of (+)-17-(3-pyridyl)-(5 beta)-10-azaestra-1,16-dien-3-one, a novel potential inhibitor for human cytochrome P450(17 alpha) (17 alpha-hydroxylase/C-17,C-20-lyase)
Authors: Guarna, A Occhiato, EG Machetti, F Giacomelli, V
Citation: A. Guarna et al., 19-nor-10-azasteroids. 5. A synthetic strategy for the preparation of (+)-17-(3-pyridyl)-(5 beta)-10-azaestra-1,16-dien-3-one, a novel potential inhibitor for human cytochrome P450(17 alpha) (17 alpha-hydroxylase/C-17,C-20-lyase), J ORG CHEM, 64(13), 1999, pp. 4985-4989
Risultati: 1-14 |