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Results: 1-25 |
Results: 25
A SIMPLE METHOD FOR COUPLING ALDEHYDES TO SOLID SUPPORT
Authors: METZ WA JONES WD CISKE FL PEET NP
Citation: Wa. Metz et al., A SIMPLE METHOD FOR COUPLING ALDEHYDES TO SOLID SUPPORT, Bioorganic & medicinal chemistry letters, 8(17), 1998, pp. 2399-2402
PREPARATION OF ALPHA-KETO ESTER ENOL ACETATES AS POTENTIAL PRODRUGS OF HUMAN NEUTROPHIL ELASTASE INHIBITORS
Authors: BURKHART JP MEHDI S KOEHL JR ANGELASTRO MR BEY P PEET NP
Citation: Jp. Burkhart et al., PREPARATION OF ALPHA-KETO ESTER ENOL ACETATES AS POTENTIAL PRODRUGS OF HUMAN NEUTROPHIL ELASTASE INHIBITORS, Bioorganic & medicinal chemistry letters, 8(1), 1998, pp. 63-64
INHIBITION OF HUMAN NEUTROPHIL ELASTASE - 4 - DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF P-2-MODIFIED, ORALLY-ACTIVE PEPTIDYL PENTAFLUOROETHYL KETONES
Authors: CREGGE RJ DURHAM SL FARR RA GALLION SL HARE CM HOFFMAN RV JANUSZ MJ KIM HO KOEHL JR MEHDI S METZ WA PEET NP PELTON JT SCHREUDER HA SUNDER S TARDIF C
Citation: Rj. Cregge et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE - 4 - DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF P-2-MODIFIED, ORALLY-ACTIVE PEPTIDYL PENTAFLUOROETHYL KETONES, Journal of medicinal chemistry, 41(14), 1998, pp. 2461-2480
ISOQUINOLINE ALKALOIDS - 3 - SYNTHESIS OF THE 6-ETHYL AND 6-BUTYL ANALOGS OF O-1,2,9,10-TETRAMETHOXY-4H-DIBENZO[DE,G]-QUINOLINE 1.5 PHOSPHATE (D,L-GLAUCINE 1.5 PHOSPHATE)
Authors: GORALSKI CT HASHA DL HENTON DR PEET NP
Citation: Ct. Goralski et al., ISOQUINOLINE ALKALOIDS - 3 - SYNTHESIS OF THE 6-ETHYL AND 6-BUTYL ANALOGS OF O-1,2,9,10-TETRAMETHOXY-4H-DIBENZO[DE,G]-QUINOLINE 1.5 PHOSPHATE (D,L-GLAUCINE 1.5 PHOSPHATE), Organic process research & development, 1(4), 1997, pp. 280-286
PREPARATION OF N-ARYL-2-HYDROXYPROPIONAMIDES FROM HYDROXY AROMATIC-COMPOUNDS USING A ONE-POT SMILES REARRANGEMENT PROCEDURE
Authors: WEIDNER JJ WEINTRAUB PM SCHNETTLER RA PEET NP
Citation: Jj. Weidner et al., PREPARATION OF N-ARYL-2-HYDROXYPROPIONAMIDES FROM HYDROXY AROMATIC-COMPOUNDS USING A ONE-POT SMILES REARRANGEMENT PROCEDURE, Tetrahedron, 53(18), 1997, pp. 6303-6312
DIRECT CONVERSION OF HYDROXY AROMATIC-COMPOUNDS TO HETEROARYLAMINES VIA A ONE-POT SMILES REARRANGEMENT PROCEDURE
Authors: WEIDNER JJ PEET NP
Citation: Jj. Weidner et Np. Peet, DIRECT CONVERSION OF HYDROXY AROMATIC-COMPOUNDS TO HETEROARYLAMINES VIA A ONE-POT SMILES REARRANGEMENT PROCEDURE, Journal of heterocyclic chemistry, 34(6), 1997, pp. 1857-1860
MOLECULAR DESIGN AND CHARACTERIZATION OF AN ALPHA-THROMBIN INHIBITOR CONTAINING A NOVEL PI MOIETY
Authors: MALIKAYIL JA BURKHART JP SCHREUDER HA BROERSMA RJ TARDIF C KUTCHER LW MEHDI S SCHATZMAN GL NEISES B PEET NP
Citation: Ja. Malikayil et al., MOLECULAR DESIGN AND CHARACTERIZATION OF AN ALPHA-THROMBIN INHIBITOR CONTAINING A NOVEL PI MOIETY, Biochemistry, 36(5), 1997, pp. 1034-1040
TIME-DEPENDENT INACTIVATION OF STEROID C-17(20)LYASE BY 17-BETA-CYCLOPROPYL ETHER-SUBSTITUTED STEROIDS
Authors: ANGELASTRO MR MARQUART AL WEINTRAUB PM GATES CA LAUGHLIN ME BLOHM TR PEET NP
Citation: Mr. Angelastro et al., TIME-DEPENDENT INACTIVATION OF STEROID C-17(20)LYASE BY 17-BETA-CYCLOPROPYL ETHER-SUBSTITUTED STEROIDS, Bioorganic & medicinal chemistry letters, 6(1), 1996, pp. 97-100
PREPARATION AND REACTIONS OF OPTICALLY-ACTIVE 4-HYDROXY-1,3-DIOXOLANES - 2-HYDROXY ALDEHYDE EQUIVALENTS
Authors: KIM HO FRIEDRICH D HUBER E PEET NP
Citation: Ho. Kim et al., PREPARATION AND REACTIONS OF OPTICALLY-ACTIVE 4-HYDROXY-1,3-DIOXOLANES - 2-HYDROXY ALDEHYDE EQUIVALENTS, Synthetic communications, 26(18), 1996, pp. 3453-3469
CARBOCYCLIC NUCLEOSIDES AS INHIBITORS OF HUMAN TUMOR-NECROSIS-FACTOR-ALPHA PRODUCTION - EFFECTS OF THE STEREOISOMERS OF (3-HYDROXYCYCLOPENTYL)ADENINES
Authors: BORCHERDING DR PEET NP MUNSON HR ZHANG H HOFFMAN PF BOWLIN TL EDWARDS CK
Citation: Dr. Borcherding et al., CARBOCYCLIC NUCLEOSIDES AS INHIBITORS OF HUMAN TUMOR-NECROSIS-FACTOR-ALPHA PRODUCTION - EFFECTS OF THE STEREOISOMERS OF (3-HYDROXYCYCLOPENTYL)ADENINES, Journal of medicinal chemistry, 39(13), 1996, pp. 2615-2620
ACTIVATION OF ADENOSINE A(3) RECEPTORS ON MACROPHAGES INHIBITS TUMOR-NECROSIS-FACTOR-ALPHA
Authors: MCWHINNEY CD DUDLEY MW BOWLIN TL PEET NP SCHOOK L BRADSHAW M DE M BORCHERDING DR EDWARDS CK
Citation: Cd. Mcwhinney et al., ACTIVATION OF ADENOSINE A(3) RECEPTORS ON MACROPHAGES INHIBITS TUMOR-NECROSIS-FACTOR-ALPHA, European journal of pharmacology, 310(2-3), 1996, pp. 209-216
PHARMACOLOGICAL EVALUATION OF SELECTED, ORALLY-ACTIVE, PEPTIDYL INHIBITORS OF HUMAN NEUTROPHIL ELASTASE
Authors: JANUSZ MJ DURHAM SL HARE CM GEARY JL MANDAGERE AK POOLE JC THOMPSON TN XU D ANGELASTRO MR BURKHART JP CHEN TM MARQUART AL PEET NP HWANG KK
Citation: Mj. Janusz et al., PHARMACOLOGICAL EVALUATION OF SELECTED, ORALLY-ACTIVE, PEPTIDYL INHIBITORS OF HUMAN NEUTROPHIL ELASTASE, The Journal of pharmacology and experimental therapeutics, 275(3), 1995, pp. 1233-1238
INHIBITION OF HUMAN NEUTROPHIL ELASTASE .3. AN ORALLY-ACTIVE ENOL ACETATE PRODRUG
Authors: BURKHART JP KOEHL JR MEHDI S DURHAM SL JANUSZ MJ HUBER EW ANGELASTRO MR SUNDER S METZ WA SHUM PW CHEN TM BEY P CREGGE RJ PEET NP
Citation: Jp. Burkhart et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE .3. AN ORALLY-ACTIVE ENOL ACETATE PRODRUG, Journal of medicinal chemistry, 38(2), 1995, pp. 223-233
REACTION OF NINHYDRIN WITH BETA-DICARBONYL COMPOUNDS
Authors: PEET NP HUBER EW HUFFMAN JC
Citation: Np. Peet et al., REACTION OF NINHYDRIN WITH BETA-DICARBONYL COMPOUNDS, Journal of heterocyclic chemistry, 32(1), 1995, pp. 33-41
INHIBITION OF OXIDOSQUALENE CYCLASE BY SUBSTITUTED QUINOLIZIDINES
Authors: MARQUART AL SCHATZMAN GL PEET NP MOORE WR HUBER EW GALLION SL ANGELASTRO MR
Citation: Al. Marquart et al., INHIBITION OF OXIDOSQUALENE CYCLASE BY SUBSTITUTED QUINOLIZIDINES, Bioorganic & medicinal chemistry letters, 4(11), 1994, pp. 1317-1318
PYRROLIDINE AND HEXAHYDRO-1H-AZEPINE MIMICS OF THE FLAP UP MANNOSYL CATION
Authors: FARR RA HOLLAND AK HUBER EW PEET NP WEINTRAUB PM
Citation: Ra. Farr et al., PYRROLIDINE AND HEXAHYDRO-1H-AZEPINE MIMICS OF THE FLAP UP MANNOSYL CATION, Tetrahedron, 50(4), 1994, pp. 1033-1044
REINVESTIGATION OF SYNTHETIC ROUTES TO 1,3,4-BENZOXADIAZEPIN-5-ONES AND 1,3-BENZOXAZEPINES
Authors: KIM HO HUBER EW FRIEDRICH D PEET NP
Citation: Ho. Kim et al., REINVESTIGATION OF SYNTHETIC ROUTES TO 1,3,4-BENZOXADIAZEPIN-5-ONES AND 1,3-BENZOXAZEPINES, Synthesis, (12), 1994, pp. 1406-1408
PHARMACOLOGY OF FLUORO-1-(1-METHYLETHYL)-2-OXOBUTYL]-L-PROLINAMIDE (MDL-101,146) - A POTENT ORALLY-ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE (VOL 270, PG 185, 1994)
Authors: DURHAM SL HARE CM ANGELASTRO MR BURKHART JP KOEHL JR MARQUART AL MEHDI S PEET NP JANUSZ MJ
Citation: Sl. Durham et al., PHARMACOLOGY OF FLUORO-1-(1-METHYLETHYL)-2-OXOBUTYL]-L-PROLINAMIDE (MDL-101,146) - A POTENT ORALLY-ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE (VOL 270, PG 185, 1994), The Journal of pharmacology and experimental therapeutics, 271(3), 1994, pp. 1720-1720
SYNTHESIS OF CHIRAL HYDROXYLATED QUINOLIZIDINES VIA VINYLOGOUS BISCHLER-NAPIERALSKI NITRILIUM ION CYCLIZATIONS
Authors: MARQUART AL PODLOGAR BL HUBER EW DEMETER DA PEET NP WEINTRAUB HJR ANGELASTRO MR
Citation: Al. Marquart et al., SYNTHESIS OF CHIRAL HYDROXYLATED QUINOLIZIDINES VIA VINYLOGOUS BISCHLER-NAPIERALSKI NITRILIUM ION CYCLIZATIONS, Journal of organic chemistry, 59(8), 1994, pp. 2092-2100
INHIBITION OF HUMAN NEUTROPHIL ELASTASE WITH PEPTIDYL ELECTROPHILIC KETONES .2. ORALLY-ACTIVE P-G-VAL-PRO-VAL PENTAFLUOROETHYL KETONES
Authors: ANGELASTRO MR BAUGH LE BEY P BURKHART JP CHEN TM DURHAM SL HARE CM HUBER EW JANUSZ MJ KOEHL JR MARQUART AL MEHDI S PEET NP
Citation: Mr. Angelastro et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE WITH PEPTIDYL ELECTROPHILIC KETONES .2. ORALLY-ACTIVE P-G-VAL-PRO-VAL PENTAFLUOROETHYL KETONES, Journal of medicinal chemistry, 37(26), 1994, pp. 4538-4553
SYNTHESIS OF A 2,5-DIARYLOXAZOLINE AS A POTENTIAL PLATELET-ACTIVATING-FACTOR ANTAGONIST
Authors: PEET NP BURKHART JP BROERSMA RJ HEMINGER EF
Citation: Np. Peet et al., SYNTHESIS OF A 2,5-DIARYLOXAZOLINE AS A POTENTIAL PLATELET-ACTIVATING-FACTOR ANTAGONIST, Journal of heterocyclic chemistry, 31(2), 1994, pp. 419-423
A-RING BRIDGED STEROIDS AS POTENT INHIBITORS OF AROMATASE
Authors: PEET NP JOHNSTON JO BURKHART JP WRIGHT CL
Citation: Np. Peet et al., A-RING BRIDGED STEROIDS AS POTENT INHIBITORS OF AROMATASE, Journal of steroid biochemistry and molecular biology, 44(4-6), 1993, pp. 409-420
BIOLOGICAL CHARACTERIZATION OF A-RING STEROIDS
Authors: JOHNSTON JO WRIGHT CL BURKHART JP PEET NP
Citation: Jo. Johnston et al., BIOLOGICAL CHARACTERIZATION OF A-RING STEROIDS, Journal of steroid biochemistry and molecular biology, 44(4-6), 1993, pp. 623-631
XANTHINES WITH C-8 CHIRAL SUBSTITUENTS AS POTENT AND SELECTIVE ADENOSINE A(1) ANTAGONISTS
Authors: PEET NP LENTZ NL DUDLEY MW OGDEN AML MCCARTY DR RACKE MM
Citation: Np. Peet et al., XANTHINES WITH C-8 CHIRAL SUBSTITUENTS AS POTENT AND SELECTIVE ADENOSINE A(1) ANTAGONISTS, Journal of medicinal chemistry, 36(25), 1993, pp. 4015-4020
MDL 101,146, A POTENT ORALLY ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE INDUCED ACUTE PULMONARY HEMORRHAGE IN RATS AND HAMSTERS
Authors: DURHAM SL HARE CM ANGELASTRO MR BURKHART JP KOEHL JR MARQUART AL MEHDI S PEET NP JANUSZ MJ
Citation: Sl. Durham et al., MDL 101,146, A POTENT ORALLY ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE INDUCED ACUTE PULMONARY HEMORRHAGE IN RATS AND HAMSTERS, The American review of respiratory disease, 147(4), 1993, pp. 675-675
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