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Results: 1-10 |
Results: 10
5,5-TRANS LACTONE-CONTAINING INHIBITORS OF SERINE PROTEASES - IDENTIFICATION OF A NOVEL, ACYLATING THROMBIN INHIBITOR
Authors: FINCH H PEGG NA MCLAREN J LOWDON A BOLTON R COOTE SJ DYER U MONTANA JG OWEN MR DOWLE M BUCKLEY D ROSE BC CAMPBELL C DIX C MOONEY C MANTANG C PATEL C
Citation: H. Finch et al., 5,5-TRANS LACTONE-CONTAINING INHIBITORS OF SERINE PROTEASES - IDENTIFICATION OF A NOVEL, ACYLATING THROMBIN INHIBITOR, Bioorganic & medicinal chemistry letters, 8(21), 1998, pp. 2955-2960
SYNTHESIS OF TRANS-FUSED[5,5]BICYCLIC LACTONES LACTAMS AS TEMPLATES FOR SERINE-PROTEASE INHIBITION/
Authors: KELLY HA BOLTON R BROWN SA COOTE SJ DOWLE M DYER U FINCH H GOLDING D LOWDON A MCLAREN J MONTANA JG OWEN MR PEGG NA ROSS BC THOMAS R WALKER DA
Citation: Ha. Kelly et al., SYNTHESIS OF TRANS-FUSED[5,5]BICYCLIC LACTONES LACTAMS AS TEMPLATES FOR SERINE-PROTEASE INHIBITION/, Tetrahedron letters, 39(38), 1998, pp. 6979-6982
REACTION OF ALPHA-AMINO ESTERS AND ALPHA-AMINO ESTER IMINES WITH THIIRANIUM ION INTERMEDIATES - APPLICATION TO THE SYNTHESIS OF NEW POTENTIAL AMINOPEPTIDASE INHIBITORS AND MECHANISTIC IMPLICATIONS
Authors: GILL DM PEGG NA RAYNER CM
Citation: Dm. Gill et al., REACTION OF ALPHA-AMINO ESTERS AND ALPHA-AMINO ESTER IMINES WITH THIIRANIUM ION INTERMEDIATES - APPLICATION TO THE SYNTHESIS OF NEW POTENTIAL AMINOPEPTIDASE INHIBITORS AND MECHANISTIC IMPLICATIONS, Tetrahedron, 53(9), 1997, pp. 3383-3394
TETRAZOLE NK1 RECEPTOR ANTAGONISTS - THE IDENTIFICATION OF AN EXCEPTIONALLY POTENT ORALLY-ACTIVE ANTIEMETIC COMPOUND
Authors: ARMOUR DR CHUNG KML CONGREVE M EVANS B GUNTRIP S HUBBARD T KAY C MIDDLEMISS D MORDAUNT JE PEGG NA VINADER MV WARD P WATSON SP
Citation: Dr. Armour et al., TETRAZOLE NK1 RECEPTOR ANTAGONISTS - THE IDENTIFICATION OF AN EXCEPTIONALLY POTENT ORALLY-ACTIVE ANTIEMETIC COMPOUND, Bioorganic & medicinal chemistry letters, 6(9), 1996, pp. 1015-1020
LEWIS-ACID INDUCED REARRANGEMENT OF 2,3-EPOXY SULFIDES - REGIOSPECIFIC TRAPPING OF THIIRANIUM ION INTERMEDIATES WITH NITROGEN-HETEROCYCLES AND AMIDES - USE OF IMINES AS NUCLEOPHILIC EQUIVALENTS FOR THE SELECTIVE MONOALKYLATION OF PRIMARY AMINES
Authors: GILL DM PEGG NA RAYNER CM
Citation: Dm. Gill et al., LEWIS-ACID INDUCED REARRANGEMENT OF 2,3-EPOXY SULFIDES - REGIOSPECIFIC TRAPPING OF THIIRANIUM ION INTERMEDIATES WITH NITROGEN-HETEROCYCLES AND AMIDES - USE OF IMINES AS NUCLEOPHILIC EQUIVALENTS FOR THE SELECTIVE MONOALKYLATION OF PRIMARY AMINES, Tetrahedron, 52(10), 1996, pp. 3609-3630
SPIRO-PIPERIDINE NONPEPTIDE NEUROKININ-1 RECEPTOR ANTAGONISTS
Authors: ARMOUR DR WATSON SP PEGG NA HERON NM MIDDLEMISS D CHAN C CHOLERTON TJ HUBBARD T VINADER MV DAVIES HG COCKER JD BAYS DE WARD P
Citation: Dr. Armour et al., SPIRO-PIPERIDINE NONPEPTIDE NEUROKININ-1 RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 5(22), 1995, pp. 2671-2676
IMINES AS SYNTHETIC EQUIVALENTS OF PRIMARY AMINES FOR THE NUCLEOPHILIC TRAPPING OF THIIRANIUM ION INTERMEDIATES
Authors: GILL DM PEGG NA RAYNER CM
Citation: Dm. Gill et al., IMINES AS SYNTHETIC EQUIVALENTS OF PRIMARY AMINES FOR THE NUCLEOPHILIC TRAPPING OF THIIRANIUM ION INTERMEDIATES, Synlett, (12), 1995, pp. 1275
ADDITION OF AMINO ESTERS TO THIIRANIUM ION INTERMEDIATES - A NOVEL-APPROACH TO THE SYNTHESIS OF NEW POTENTIAL AMINOPEPTIDASE INHIBITORS
Authors: GILL DM PEGG NA RAYNER CM
Citation: Dm. Gill et al., ADDITION OF AMINO ESTERS TO THIIRANIUM ION INTERMEDIATES - A NOVEL-APPROACH TO THE SYNTHESIS OF NEW POTENTIAL AMINOPEPTIDASE INHIBITORS, Tetrahedron letters, 36(45), 1995, pp. 8327-8330
DISCOVERY OF AN ORALLY BIOAVAILABLE NK1 RECEPTOR ANTAGONIST, -TETRAZOL-1-YLBENZYL)(2-PHENYLPIPERIDIN-3-YL)AMINE (GR203040), WITH POTENT ANTIEMETIC ACTIVITY
Authors: WARD P ARMOUR DR BAYS DE EVANS B GIBLIN GMP HERON N HUBBARD T LIANG K MIDDLEMISS D MORDAUNT J NAYLOR A PEGG NA VINADER MV WATSON SP BOUNTRA C EVANS DC
Citation: P. Ward et al., DISCOVERY OF AN ORALLY BIOAVAILABLE NK1 RECEPTOR ANTAGONIST, -TETRAZOL-1-YLBENZYL)(2-PHENYLPIPERIDIN-3-YL)AMINE (GR203040), WITH POTENT ANTIEMETIC ACTIVITY, Journal of medicinal chemistry, 38(26), 1995, pp. 4985-4992
THE SYNTHESIS OF A CONFORMATIONALLY RESTRAINED, COMBINED THROMBOXANE ANTAGONIST SYNTHASE INHIBITOR USING AN INTRAMOLECULAR STILLE-PALLADIUM-CATALYZED OR GRIGG-PALLADIUM-CATALYZED CYCLIZATION STRATEGY/
Authors: FINCH H PEGG NA EVANS B
Citation: H. Finch et al., THE SYNTHESIS OF A CONFORMATIONALLY RESTRAINED, COMBINED THROMBOXANE ANTAGONIST SYNTHASE INHIBITOR USING AN INTRAMOLECULAR STILLE-PALLADIUM-CATALYZED OR GRIGG-PALLADIUM-CATALYZED CYCLIZATION STRATEGY/, Tetrahedron letters, 34(51), 1993, pp. 8353-8356
Risultati: 1-10 |