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Results: 1-13 |
Results: 13
NEW THROMBIN INHIBITORS IN CARDIOVASCULAR-DISEASE
Authors: RIPKA WC
Citation: Wc. Ripka, NEW THROMBIN INHIBITORS IN CARDIOVASCULAR-DISEASE, CURRENT OPINION IN CHEMICAL BIOLOGY, 1(2), 1997, pp. 242-253
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF P-2-P-4 AZAPEPTIDOMIMETIC P-1-ARGININAL AND P-1-KETOARGININAMIDE DERIVATIVES - A NOVEL CLASS OF SERINE-PROTEASE INHIBITORS
Authors: SEMPLE JE ROWLEY DC BRUNCK TK RIPKA WC
Citation: Je. Semple et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF P-2-P-4 AZAPEPTIDOMIMETIC P-1-ARGININAL AND P-1-KETOARGININAMIDE DERIVATIVES - A NOVEL CLASS OF SERINE-PROTEASE INHIBITORS, Bioorganic & medicinal chemistry letters, 7(3), 1997, pp. 315-320
RATIONAL DESIGN, SYNTHESIS, AND SERINE-PROTEASE INHIBITORY ACTIVITY OF A NOVEL P-1-ARGININAL DERIVATIVE FEATURING A CONFORMATIONALLY CONSTRAINED P-2-P-3-BICYCLIC LACTAM MOIETY
Authors: TAMURA SY GOLDMAN EA BRUNCK TK RIPKA WC SEMPLE JE
Citation: Sy. Tamura et al., RATIONAL DESIGN, SYNTHESIS, AND SERINE-PROTEASE INHIBITORY ACTIVITY OF A NOVEL P-1-ARGININAL DERIVATIVE FEATURING A CONFORMATIONALLY CONSTRAINED P-2-P-3-BICYCLIC LACTAM MOIETY, Bioorganic & medicinal chemistry letters, 7(3), 1997, pp. 331-336
RATIONAL DESIGN AND SYNTHESIS OF A NOVEL, SELECTIVE CLASS OF THROMBININHIBITORS - P-1-ARGININAL DERIVATIVES INCORPORATING P-3-P-4 QUATERNARY LACTAM DIPEPTIDE SURROGATES
Authors: SEMPLE JE MINAMI NK TAMURA SY BRUNCK TK NUTT RF RIPKA WC
Citation: Je. Semple et al., RATIONAL DESIGN AND SYNTHESIS OF A NOVEL, SELECTIVE CLASS OF THROMBININHIBITORS - P-1-ARGININAL DERIVATIVES INCORPORATING P-3-P-4 QUATERNARY LACTAM DIPEPTIDE SURROGATES, Bioorganic & medicinal chemistry letters, 7(18), 1997, pp. 2421-2426
DESIGN AND SYNTHESIS OF A NOVEL CLASS OF THROMBIN INHIBITORS INCORPORATING HETEROCYCLIC DIPEPTIDE SURROGATES
Authors: TAMURA SY SEMPLE JE REINER JE GOLDMAN EA BRUNCK TK LIMWILBY MS CARPENTER SH ROTE WE OLDESHULTE GL RICHARD BM NUTT RF RIPKA WC
Citation: Sy. Tamura et al., DESIGN AND SYNTHESIS OF A NOVEL CLASS OF THROMBIN INHIBITORS INCORPORATING HETEROCYCLIC DIPEPTIDE SURROGATES, Bioorganic & medicinal chemistry letters, 7(12), 1997, pp. 1543-1548
RATIONAL DESIGN, SYNTHESIS, AND SERINE-PROTEASE INHIBITORY ACTIVITY OF NOVEL P-1-ARGININOYL HETEROCYCLES
Authors: TAMURA SY SHAMBLIN BM BRUNCK TK RIPKA WC
Citation: Sy. Tamura et al., RATIONAL DESIGN, SYNTHESIS, AND SERINE-PROTEASE INHIBITORY ACTIVITY OF NOVEL P-1-ARGININOYL HETEROCYCLES, Bioorganic & medicinal chemistry letters, 7(10), 1997, pp. 1359-1364
SYNTHESIS, STRUCTURE, AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF DIVALENT THROMBIN INHIBITORS CONTA AN ALPHA-KETO-AMIDE TRANSITION-STATE MIMETIC
Authors: KRISHNAN R TULINSKY A VLASUK GP PEARSON D VALLAR P BERGUM P BRUNCK TK RIPKA WC
Citation: R. Krishnan et al., SYNTHESIS, STRUCTURE, AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF DIVALENT THROMBIN INHIBITORS CONTA AN ALPHA-KETO-AMIDE TRANSITION-STATE MIMETIC, Protein science, 5(3), 1996, pp. 422-433
POTENT AND SELECTIVE THROMBIN INHIBITORS INCORPORATING THE CONSTRAINED ARGININE MIMIC L-3-PIPERIDYL(N-GUANIDINO)ALANINE AT P-1
Authors: LEVY OE SEMPLE JE LIM ML REINER J ROTE WE DEMPSEY E RICHARD BM ZHANG E TULINSKY A RIPKA WC NUTT RF
Citation: Oe. Levy et al., POTENT AND SELECTIVE THROMBIN INHIBITORS INCORPORATING THE CONSTRAINED ARGININE MIMIC L-3-PIPERIDYL(N-GUANIDINO)ALANINE AT P-1, Journal of medicinal chemistry, 39(23), 1996, pp. 4527-4530
DESIGN, SYNTHESIS, AND EVOLUTION OF A NOVEL, SELECTIVE, AND ORALLY BIOAVAILABLE CLASS OF THROMBIN INHIBITORS - P1-ARGININAL DERIVATIVES INCORPORATING P3-P4 LACTAM SULFONAMIDE MOIETIES
Authors: SEMPLE JE ROWLEY DC BRUNCK TK HAUONG T MINAMI NK OWENS TD TAMURA SY GOLDMAN EA SIEV DV ARDECKY RJ CARPENTER SH GE Y RICHARD BM NOLAN TG HAKANSON K TULINSKY A NUTT RF RIPKA WC
Citation: Je. Semple et al., DESIGN, SYNTHESIS, AND EVOLUTION OF A NOVEL, SELECTIVE, AND ORALLY BIOAVAILABLE CLASS OF THROMBIN INHIBITORS - P1-ARGININAL DERIVATIVES INCORPORATING P3-P4 LACTAM SULFONAMIDE MOIETIES, Journal of medicinal chemistry, 39(23), 1996, pp. 4531-4536
DESIGN STRATEGIES FOR SERINE-PROTEASE INHIBITORS
Authors: RIPKA WC
Citation: Wc. Ripka, DESIGN STRATEGIES FOR SERINE-PROTEASE INHIBITORS, The FASEB journal, 9(6), 1995, pp. 1253-1253
CHARACTERIZATION OF A NOVEL SERIES OF APROTININ-DERIVED ANTICOAGULANTS .1. IN-VITRO AND PHARMACOLOGICAL PROPERTIES
Authors: STASSEN JM LAMBEIR AM MATTHYSSENS G RIPKA WC NYSTROM A SIXMA JJ VERMYLEN J
Citation: Jm. Stassen et al., CHARACTERIZATION OF A NOVEL SERIES OF APROTININ-DERIVED ANTICOAGULANTS .1. IN-VITRO AND PHARMACOLOGICAL PROPERTIES, Thrombosis and haemostasis, 74(2), 1995, pp. 646-654
PROTEIN BETA-TURN MIMETICS .1. DESIGN, SYNTHESIS, AND EVALUATION IN MODEL CYCLIC-PEPTIDES
Authors: RIPKA WC DELUCCA GV BACH AC POTTORF RS BLANEY JM
Citation: Wc. Ripka et al., PROTEIN BETA-TURN MIMETICS .1. DESIGN, SYNTHESIS, AND EVALUATION IN MODEL CYCLIC-PEPTIDES, Tetrahedron, 49(17), 1993, pp. 3593-3608
PROTEIN BETA-TURN MIMETICS .2. DESIGN, SYNTHESIS, AND EVALUATION IN THE CYCLIC PEPTIDE GRAMICIDIN-S
Authors: RIPKA WC DELUCCA GV BACH AC POTTORF RS BLANEY JM
Citation: Wc. Ripka et al., PROTEIN BETA-TURN MIMETICS .2. DESIGN, SYNTHESIS, AND EVALUATION IN THE CYCLIC PEPTIDE GRAMICIDIN-S, Tetrahedron, 49(17), 1993, pp. 3609-3628
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