AAAAAA

   
Results: 1-19 |
Results: 19
DEPLETION OF GLUTATHIONE BY BENZO(A)PYRENE METABOLITES, IONOMYCIN, THAPSIGARGIN, AND PHORBOL-MYRISTATE IN HUMAN PERIPHERAL-BLOOD MONONUCLEAR-CELLS
Authors: ROMERO DL MOUNHO BJ LAUER FT BORN JL BURCHIEL SW
Citation: Dl. Romero et al., DEPLETION OF GLUTATHIONE BY BENZO(A)PYRENE METABOLITES, IONOMYCIN, THAPSIGARGIN, AND PHORBOL-MYRISTATE IN HUMAN PERIPHERAL-BLOOD MONONUCLEAR-CELLS, Toxicology and applied pharmacology, 144(1), 1997, pp. 62-69
THE PALLADIUM-CATALYZED ALLYLIC ALKYLATION OF BIS(TRIMETHYLSILYL) SUBSTITUTED PROPENYL ACETATES OR CARBONATES IN THE PRESENCE OF CHIRAL LIGANDS
Authors: ROMERO DL FRITZEN EL
Citation: Dl. Romero et El. Fritzen, THE PALLADIUM-CATALYZED ALLYLIC ALKYLATION OF BIS(TRIMETHYLSILYL) SUBSTITUTED PROPENYL ACETATES OR CARBONATES IN THE PRESENCE OF CHIRAL LIGANDS, Tetrahedron letters, 38(50), 1997, pp. 8659-8662
HUMAN T-CELLS ARE HIGHLY SENSITIVE TO SUPPRESSION OF MITOGENESIS BY POLYCYCLIC AROMATIC-HYDROCARBONS AND THIS EFFECT IS DIFFERENTIALLY REVERSED BY ALPHA-NAPHTHOFLAVONE
Authors: DAVILA DR ROMERO DL BURCHIEL SW
Citation: Dr. Davila et al., HUMAN T-CELLS ARE HIGHLY SENSITIVE TO SUPPRESSION OF MITOGENESIS BY POLYCYCLIC AROMATIC-HYDROCARBONS AND THIS EFFECT IS DIFFERENTIALLY REVERSED BY ALPHA-NAPHTHOFLAVONE, Toxicology and applied pharmacology, 139(2), 1996, pp. 333-341
(ALKYLAMINO)PIPERIDINE BIS(HETEROARYL)PIPERIZINE ANALOGS ARE POTENT, BROAD-SPECTRUM NONNUCLEOSIDE REVERSE-TRANSCRIPTASE INHIBITORS OF DRUG-RESISTANT ISOLATES OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 (HIV-1) AND SELECT FOR DRUG-RESISTANT VARIANTS OF HIV-1(IIIB) WITH REDUCED REPLICATION PHENOTYPES
Authors: OLMSTED RA SLADE DE KOPTA LA POPPE SM POEL TJ NEWPORT SW RANK KB BILES C MORGE RA DUEWEKE TJ YAGI Y ROMERO DL THOMAS RC SHARMA SK TARPLEY WG
Citation: Ra. Olmsted et al., (ALKYLAMINO)PIPERIDINE BIS(HETEROARYL)PIPERIZINE ANALOGS ARE POTENT, BROAD-SPECTRUM NONNUCLEOSIDE REVERSE-TRANSCRIPTASE INHIBITORS OF DRUG-RESISTANT ISOLATES OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 (HIV-1) AND SELECT FOR DRUG-RESISTANT VARIANTS OF HIV-1(IIIB) WITH REDUCED REPLICATION PHENOTYPES, Journal of virology, 70(6), 1996, pp. 3698-3705
SYNTHESIS AND BIOACTIVITY OF NOVEL BIS (HETEROARYL)PIPERAZINE (BHAP) REVERSE-TRANSCRIPTASE INHIBITORS - STRUCTURE-ACTIVITY-RELATIONSHIPS AND INCREASED METABOLIC STABILITY OF NOVEL SUBSTITUTED PYRIDINE ANALOGS
Authors: GENIN MJ POEL TJ YAGI Y BILES C ALTHAUS I KEISER BJ KOPTA LA FRIIS JM REUSSER F ADAMS WJ OLMSTED RA VOORMAN RL THOMAS RC ROMERO DL
Citation: Mj. Genin et al., SYNTHESIS AND BIOACTIVITY OF NOVEL BIS (HETEROARYL)PIPERAZINE (BHAP) REVERSE-TRANSCRIPTASE INHIBITORS - STRUCTURE-ACTIVITY-RELATIONSHIPS AND INCREASED METABOLIC STABILITY OF NOVEL SUBSTITUTED PYRIDINE ANALOGS, Journal of medicinal chemistry, 39(26), 1996, pp. 5267-5275
STRUCTURE-BASED DESIGN OF HIV PROTEASE INHIBITORS - 5,6-DIHYDRO-4-HYDROXY-2-PYRONES AS EFFECTIVE, NONPEPTIDIC INHIBITORS
Authors: THAISRIVONGS S ROMERO DL TOMMASI RA JANAKIRAMAN MN STROHBACH JW TURNER SR BILES C MORGE RR JOHNSON PD ARISTOFF PA TOMICH PK LYNN JC HORNG MM CHONG KT HINSHAW RR HOWE WJ FINZEL BC WATENPAUGH KD
Citation: S. Thaisrivongs et al., STRUCTURE-BASED DESIGN OF HIV PROTEASE INHIBITORS - 5,6-DIHYDRO-4-HYDROXY-2-PYRONES AS EFFECTIVE, NONPEPTIDIC INHIBITORS, Journal of medicinal chemistry, 39(23), 1996, pp. 4630-4642
TARGETING DELAVIRDINE ATEVIRDINE RESISTANT HIV-1 - IDENTIFICATION OF (ALKYLAMINO)PIPERIDINE-CONTAINING BIS(HETEROARYL)PIPERAZINES AS BROAD-SPECTRUM HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS/
Authors: ROMERO DL OLMSTED RA POEL TJ MORGE RA BILES C KEISER BJ KOPTA LA FRIIS JM HOSLEY JD STEFANSKI KJ WISHKA DG EVANS DB MORRIS J STEHLE RG SHARMA SK YAGI Y VOORMAN RL ADAMS WJ TARPLEY WG THOMAS RC
Citation: Dl. Romero et al., TARGETING DELAVIRDINE ATEVIRDINE RESISTANT HIV-1 - IDENTIFICATION OF (ALKYLAMINO)PIPERIDINE-CONTAINING BIS(HETEROARYL)PIPERAZINES AS BROAD-SPECTRUM HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS/, Journal of medicinal chemistry, 39(19), 1996, pp. 3769-3789
SPECTROSCOPIC STUDIES OF DELAVIRDINE MESYLATE (U-90,152T) A BIS(HETEROARYL)PIPERAZINE (BHAP) HIV REVERSE-TRANSCRIPTASE INHIBITOR
Authors: FARLEY KA WALKER GS ROBINS RH KUPSTASGUIDO JE DUHOLKE WK ROMERO DL MORGE RA MEULMAN PA CHAO RS HAVENS JL GAGE JR LYSTER MA FAGERNESS PE MARTIN GE
Citation: Ka. Farley et al., SPECTROSCOPIC STUDIES OF DELAVIRDINE MESYLATE (U-90,152T) A BIS(HETEROARYL)PIPERAZINE (BHAP) HIV REVERSE-TRANSCRIPTASE INHIBITOR, Journal of heterocyclic chemistry, 33(2), 1996, pp. 493-496
THE BENZYLTHIO-PYRIMIDINE U-31,355, A POTENT INHIBITOR OF HIV-1 REVERSE-TRANSCRIPTASE
Authors: ALTHAUS IW CHOU KC LEMAY RJ FRANKS KM DEIBEL MR KEZDY FJ RESNICK L BUSSO ME SO AG DOWNEY KM ROMERO DL THOMAS RC ARISTOFF PA TARPLEY WG REUSSER F
Citation: Iw. Althaus et al., THE BENZYLTHIO-PYRIMIDINE U-31,355, A POTENT INHIBITOR OF HIV-1 REVERSE-TRANSCRIPTASE, Biochemical pharmacology, 51(6), 1996, pp. 743-750
DESIGN AND SYNTHESIS OF A CONFORMATIONALLY CONSTRAINED ANALOG OF THE BIS(HETEROARYL)PIPERAZINE (BHAP) HIV-1 REVERSE-TRANSCRIPTASE INHIBITORATEVIRDINE
Authors: GENIN MJ CHIDESTER CG ROHRER DC ROMERO DL
Citation: Mj. Genin et al., DESIGN AND SYNTHESIS OF A CONFORMATIONALLY CONSTRAINED ANALOG OF THE BIS(HETEROARYL)PIPERAZINE (BHAP) HIV-1 REVERSE-TRANSCRIPTASE INHIBITORATEVIRDINE, Bioorganic & medicinal chemistry letters, 5(16), 1995, pp. 1875-1880
DISCOVERY, SYNTHESIS, AND BIOACTIVITY OF BIS(HETEROARYL)PIPERAZINES .1. A NOVEL CLASS OF NONNUCLEOSIDE HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS
Authors: ROMERO DL MORGE RA BILES C BERRIOSPENA TN MAY PD PALMER JR JOHNSON PD SMITH HW BUSSO M TAN CK VOORMAN RL REUSSER F ALTHAUS IW DOWNEY KM SO AG RESNICK L TARPLEY WG ARISTOFF PA
Citation: Dl. Romero et al., DISCOVERY, SYNTHESIS, AND BIOACTIVITY OF BIS(HETEROARYL)PIPERAZINES .1. A NOVEL CLASS OF NONNUCLEOSIDE HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS, Journal of medicinal chemistry, 37(7), 1994, pp. 999-1014
STEADY-STATE KINETIC-STUDIES WITH THE POLYSULFONATE U-9843, AN HIV REVERSE-TRANSCRIPTASE INHIBITOR
Authors: ALTHAUS IW CHOU JJ GONZALES AJ LEMAY RJ DEIBEL MR CHOU KC KEZDY FJ ROMERO DL THOMAS RC ARISTOFF PA TARPLEY WG REUSSER F
Citation: Iw. Althaus et al., STEADY-STATE KINETIC-STUDIES WITH THE POLYSULFONATE U-9843, AN HIV REVERSE-TRANSCRIPTASE INHIBITOR, Experientia, 50(1), 1994, pp. 23-28
KINETIC-STUDIES WITH THE NONNUCLEOSIDE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE INHIBITOR U-90152E
Authors: ALTHAUS IW CHOU JJ GONZALES AJ DEIBEL MR CHOU KC KEZDY FJ ROMERO DL THOMAS RC ARISTOFF PA TARPLEY WG REUSSER F
Citation: Iw. Althaus et al., KINETIC-STUDIES WITH THE NONNUCLEOSIDE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE INHIBITOR U-90152E, Biochemical pharmacology, 47(11), 1994, pp. 2017-2028
PD-CATALYZED CYCLOISOMERIZATION TO 1,2-DIALKYLIDENECYCLOALKANES .2. ALTERNATIVE CATALYST SYSTEM
Authors: TROST BM ROMERO DL RISE F
Citation: Bm. Trost et al., PD-CATALYZED CYCLOISOMERIZATION TO 1,2-DIALKYLIDENECYCLOALKANES .2. ALTERNATIVE CATALYST SYSTEM, Journal of the American Chemical Society, 116(10), 1994, pp. 4268-4278
U-90152, A POTENT INHIBITOR OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REPLICATION
Authors: DUEWEKE TJ POPPE SM ROMERO DL SWANEY SM SO AG DOWNEY KM ALTHAUS IW REUSSER F BUSSO M RESNICK L MAYERS DI LANE J ARISTOFF PA THOMAS RC TARPLEY WG
Citation: Tj. Dueweke et al., U-90152, A POTENT INHIBITOR OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REPLICATION, Antimicrobial agents and chemotherapy, 37(5), 1993, pp. 1127-1131
A NOVEL METHOD FOR THE T-BUTYLATION OF AROMATIC-AMINES
Authors: GENIN MJ BILES C ROMERO DL
Citation: Mj. Genin et al., A NOVEL METHOD FOR THE T-BUTYLATION OF AROMATIC-AMINES, Tetrahedron letters, 34(27), 1993, pp. 4301-4304
BIS(HETEROARYL)PIPERAZINE (BHAP) REVERSE-TRANSCRIPTASE INHIBITORS - STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL SUBSTITUTED INDOLE ANALOGS AND THE IDENTIFICATION OF ]-4-[3-[(1-METHYLETHYL)AMINO]-PYRIDINYL]PIPERAZINE MONOMETHANESULFONATE (U-90152S), A 2ND-GENERATION CLINICAL CANDIDATE
Authors: ROMERO DL MORGE RA GENIN MJ BILES C BUSSO M RESNICK L ALTHAUS IW REUSSER F THOMAS RC TARPLEY WG
Citation: Dl. Romero et al., BIS(HETEROARYL)PIPERAZINE (BHAP) REVERSE-TRANSCRIPTASE INHIBITORS - STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL SUBSTITUTED INDOLE ANALOGS AND THE IDENTIFICATION OF ]-4-[3-[(1-METHYLETHYL)AMINO]-PYRIDINYL]PIPERAZINE MONOMETHANESULFONATE (U-90152S), A 2ND-GENERATION CLINICAL CANDIDATE, Journal of medicinal chemistry, 36(10), 1993, pp. 1505-1508
THE QUINOLINE U-78036 IS A POTENT INHIBITOR OF HIV-1 REVERSE-TRANSCRIPTASE
Authors: ALTHAUS IW GONZALES AJ CHOU JJ ROMERO DL DEIBEL MR CHOU KC KEZDY FJ RESNICK L BUSSO ME SO AG DOWNEY KM THOMAS RC ARISTOFF PA TARPLEY WG REUSSER F
Citation: Iw. Althaus et al., THE QUINOLINE U-78036 IS A POTENT INHIBITOR OF HIV-1 REVERSE-TRANSCRIPTASE, The Journal of biological chemistry, 268(20), 1993, pp. 4875-4880
KINETIC-STUDIES WITH THE NONNUCLEOSIDE HIV-1 REVERSE-TRANSCRIPTASE INHIBITOR-U-88204E
Authors: ALTHAUS IW CHOU JJ GONZALES AJ DEIBEL MR CHOU KC KEZDY FJ ROMERO DL PALMER JR THOMAS RC ARISTOFF PA TARPLEY WG REUSSER F
Citation: Iw. Althaus et al., KINETIC-STUDIES WITH THE NONNUCLEOSIDE HIV-1 REVERSE-TRANSCRIPTASE INHIBITOR-U-88204E, Biochemistry, 32(26), 1993, pp. 6548-6554
Risultati: 1-19 |