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Results: 1-15 |
Results: 15
Three-dimensional model of the cyclin-dependent kinase 1 (CDK1): Ab initioactive site parameters for molecular dynamics studies of CDKs
Authors: Cavalli, A Dezi, C Folkers, G Scapozza, L Recanatini, M
Citation: A. Cavalli et al., Three-dimensional model of the cyclin-dependent kinase 1 (CDK1): Ab initioactive site parameters for molecular dynamics studies of CDKs, PROTEINS, 45(4), 2001, pp. 478-485
A new class of nonsteroidal aromatase inhibitors: Design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17 alpha-hydroxylase/C17,20-lyase
Authors: Recanatini, M Bisi, A Cavalli, A Belluti, F Gobbi, S Rampa, A Valenti, P Palzer, M Palusczak, A Hartmann, RW
Citation: M. Recanatini et al., A new class of nonsteroidal aromatase inhibitors: Design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17 alpha-hydroxylase/C17,20-lyase, J MED CHEM, 44(5), 2001, pp. 672-680
Acetylcholinesterase inhibitors: SAR and kinetic studies on omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)methyl]aminoalkoxyaryl derivatives
Authors: Rampa, A Piazzi, L Belluti, F Gobbi, S Bisi, A Bartolini, M Andrisano, V Cavrini, V Cavalli, A Recanatini, M Valenti, P
Citation: A. Rampa et al., Acetylcholinesterase inhibitors: SAR and kinetic studies on omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)methyl]aminoalkoxyaryl derivatives, J MED CHEM, 44(23), 2001, pp. 3810-3820
Synthesis and screening for antiacetylcholinesterase activity of (1-benzyl-4-oxopiperidin-3-ylidene)methylindoles and -pyrroles related to donepezil
Authors: Andreani, A Cavalli, A Granaiola, M Guardigli, M Leoni, A Locatelli, A Morigi, R Rambaldi, M Recanatini, M Roda, A
Citation: A. Andreani et al., Synthesis and screening for antiacetylcholinesterase activity of (1-benzyl-4-oxopiperidin-3-ylidene)methylindoles and -pyrroles related to donepezil, J MED CHEM, 44(23), 2001, pp. 4011-4014
Stereoselective binding of 2,3-substituted 3-hydroxypropionic acids on an immobilised human serum albumin chiral stationary phase: stereochemical characterisation and quantitative structure-retention relationship study
Authors: Andrisano, V Bertucci, C Cavrini, V Recanatini, M Cavalli, A Varoli, L Felix, G Wainer, IW
Citation: V. Andrisano et al., Stereoselective binding of 2,3-substituted 3-hydroxypropionic acids on an immobilised human serum albumin chiral stationary phase: stereochemical characterisation and quantitative structure-retention relationship study, J CHROMAT A, 876(1-2), 2000, pp. 75-86
Potential antitumor agents. Part 29: Synthesis and potential coanthracyclinic activity of imidazo[2,1-b]thiazole guanylhydrazones
Authors: Andreani, A Leoni, A Locatelli, A Morigi, R Rambaldi, M Recanatini, M Garaliene, V
Citation: A. Andreani et al., Potential antitumor agents. Part 29: Synthesis and potential coanthracyclinic activity of imidazo[2,1-b]thiazole guanylhydrazones, BIO MED CH, 8(9), 2000, pp. 2359-2366
Design, synthesis and binding at cloned muscarinic receptors of N-[5-(1 '-substituted-acetoxymethyl)-3-oxadiazolyl] and N-[4-(1 '-substituted-acetoxymethyl)-2-dioxolanyl] dialkyl amines
Authors: Manfredini, S Lampronti, I Vertuani, S Solaroli, N Recanatini, M Bryan, D McKinney, M
Citation: S. Manfredini et al., Design, synthesis and binding at cloned muscarinic receptors of N-[5-(1 '-substituted-acetoxymethyl)-3-oxadiazolyl] and N-[4-(1 '-substituted-acetoxymethyl)-2-dioxolanyl] dialkyl amines, BIO MED CH, 8(7), 2000, pp. 1559-1566
[4-[[N-(3-Chlorophenyl)carbamoyl]oxy]-2-butynyl]-trimethylammonium (McN-A-343)-related compounds. Effect of the butynyl chain inclusion into an aromatic unit on the potency for muscarinic receptors
Authors: Tumiatti, V Angeli, P Andrisano, V Bolognesi, ML Cavalli, A Marucci, G Minarini, A Recanatini, M Rosini, M Melchiorre, C
Citation: V. Tumiatti et al., [4-[[N-(3-Chlorophenyl)carbamoyl]oxy]-2-butynyl]-trimethylammonium (McN-A-343)-related compounds. Effect of the butynyl chain inclusion into an aromatic unit on the potency for muscarinic receptors, BIO MED CH, 8(4), 2000, pp. 681-689
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives
Authors: Rampa, A Bisi, A Belluti, F Gobbi, S Valenti, P Andrisano, V Cavrini, V Cavalli, A Recanatini, M
Citation: A. Rampa et al., Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: Molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives, BIO MED CH, 8(3), 2000, pp. 497-506
Linking CoMFA and protein homology models of enzyme-inhibitor interactions: an application to non-steroidal aromatase inhibitors
Authors: Cavalli, A Greco, G Novellino, E Recanatini, M
Citation: A. Cavalli et al., Linking CoMFA and protein homology models of enzyme-inhibitor interactions: an application to non-steroidal aromatase inhibitors, BIO MED CH, 8(12), 2000, pp. 2771-2780
Imidazo[2,1-b]thiazolylmethylene- and indolylmethylene-2-indolinones: a new class of cyclin-dependent kinase inhibitors. Design, synthesis, and CDK1/cyclin B inhibition
Authors: Andreani, A Cavalli, A Granaiola, M Leoni, A Locatelli, A Morigi, R Rambaldi, M Recanatini, M Garnier, M Meijer, L
Citation: A. Andreani et al., Imidazo[2,1-b]thiazolylmethylene- and indolylmethylene-2-indolinones: a new class of cyclin-dependent kinase inhibitors. Design, synthesis, and CDK1/cyclin B inhibition, ANTI-CAN DR, 15(6), 2000, pp. 447-452
SAR of 9-amino-1,2,3,4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues
Authors: Recanatini, M Cavalli, A Belluti, F Piazzi, L Rampa, A Bisi, A Gobbi, S Valenti, P Andrisano, V Bartolini, M Cavrini, V
Citation: M. Recanatini et al., SAR of 9-amino-1,2,3,4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues, J MED CHEM, 43(10), 2000, pp. 2007-2018
Synthesis and antagonistic activity at muscarinic receptor subtypes of some 2-carbonyl derivatives of diphenidol
Authors: Varoli, L Angeli, P Burnelli, S Marucci, G Recanatini, M
Citation: L. Varoli et al., Synthesis and antagonistic activity at muscarinic receptor subtypes of some 2-carbonyl derivatives of diphenidol, BIO MED CH, 7(9), 1999, pp. 1837-1844
Comparative molecular field analysis (CoMFA) of a series of selective adenosine receptor A(2A) antagonists
Authors: Baraldi, PG Borea, PA Bergonzoni, M Cacciari, B Ongini, E Recanatini, M Spalluto, G
Citation: Pg. Baraldi et al., Comparative molecular field analysis (CoMFA) of a series of selective adenosine receptor A(2A) antagonists, DRUG DEV R, 46(2), 1999, pp. 126-133
WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for alpha(1)-adrenoreceptor subtypes and 5-HT1A receptors
Authors: Bolognesi, ML Budriesi, R Cavalli, A Chiarini, A Gotti, R Leonardi, A Minarini, A Poggesi, E Recanatini, M Rosini, M Tumiatti, V Melchiorre, C
Citation: Ml. Bolognesi et al., WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for alpha(1)-adrenoreceptor subtypes and 5-HT1A receptors, J MED CHEM, 42(20), 1999, pp. 4214-4224
Risultati: 1-15 |