Authors:
Takeuchi, K
Kohn, TJ
Harper, RW
Lin, HS
Gifford-Moore, DS
Richett, ME
Sall, DJ
Smith, GF
Zhang, MS
Citation: K. Takeuchi et al., Diamino benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors. Part 6: Further focus on the contracted C4 '-sidechain analogues, BIOORG MED, 10(11), 2000, pp. 1199-1202
Authors:
Sall, DJ
Bailey, DL
Bastian, JA
Buben, JA
Chirgadze, NY
Clemens-Smith, AC
Denney, ML
Fisher, MJ
Giera, DD
Gifford-Moore, DS
Harper, RW
Johnson, LM
Klimkowski, VJ
Kohn, TJ
Lin, HS
McCowan, JR
Palkowitz, AD
Richett, ME
Smith, GF
Snyder, DW
Takeuchi, K
Toth, JE
Zhang, MS
Citation: Dj. Sall et al., Diamino benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors. 5. Potency, efficacy, and pharmacokinetic properties of modified C-3 side chain derivatives, J MED CHEM, 43(4), 2000, pp. 649-663
Authors:
Zhang, MS
Bailey, DL
Bastian, JA
Briggs, SL
Chirgadze, NY
Clawson, DK
Denney, ML
Gifford-Moore, DS
Harper, RW
Johnson, LM
Klimkowski, VJ
Kohn, TJ
Lin, HS
McCowan, JR
Richett, ME
Sall, DJ
Smith, AJ
Smith, GF
Snyder, DW
Takeuchi, K
Utterback, BG
Yan, SCB
Citation: Ms. Zhang et al., Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 2. Sidechain optimization and demonstration of invivo efficacy, BIOORG MED, 9(5), 1999, pp. 775-780
Authors:
Lin, HS
Rampersaud, AA
Richett, ME
Harper, RW
Beavers, LS
McClure, DB
Gardner, AJ
Eacho, PI
Foxworthy, PS
Gadski, RA
Citation: Hs. Lin et al., Synthesis and in vitro biological activity of 4 alpha-(2-propenyl)-5 alpha-cholest-24-en-3 alpha-ol: A 24,25-dehydro analog of the hypocholesterolemic agent 4 alpha-(2-propenyl)-5 alpha-cholestan-3 alpha-ol, STEROIDS, 64(3), 1999, pp. 217-227