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Results: 1-12 |
Results: 12
DESIGN AND SYNTHESIS OF N-ALKYLATED SACCHARINS AS SELECTIVE ALPHA-1A ADRENERGIC-RECEPTOR ANTAGONISTS
Authors: NERENBERG JB ERB JM THOMPSON WJ LEE HY GUARE JP MUNSON PM BERGMAN JM HUFF JR BROTEN TP CHANG RSL CHEN TB OMALLEY S SCHORN TW SCOTT AL
Citation: Jb. Nerenberg et al., DESIGN AND SYNTHESIS OF N-ALKYLATED SACCHARINS AS SELECTIVE ALPHA-1A ADRENERGIC-RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 8(18), 1998, pp. 2467-2472
IN-VIVO PHARMACOLOGY OF L-159,913, A NEW HIGHLY POTENT AND SELECTIVE NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONIST
Authors: GABEL RA KIVLIGHN SD ZINGARO GJ SCHORN TW SCHAFFER LW ASHTON WT CHANG LL FLANAGAN K GREENLEE WJ SIEGL PKS
Citation: Ra. Gabel et al., IN-VIVO PHARMACOLOGY OF L-159,913, A NEW HIGHLY POTENT AND SELECTIVE NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONIST, Clinical and experimental hypertension, 17(6), 1995, pp. 931-953
THE SAR OF -2-PROPYL-3-[(2'-TETRAZOL-5-YL)BIPHEN-4-YL)METHYL] QUINAZOLINONES AS BALANCED AFFINITY ANTAGONISTS OF THE HUMAN AT(1) AND AT(2) RECEPTORS
Authors: DELASZLO SE CHANG RS CHEN TB FAUST KA GREENLEE WJ KIVLIGHN SD LOTTI VJ OMALLEY SS SCHORN TW SIEGL PK TRAN J ZINGARO GJ
Citation: Se. Delaszlo et al., THE SAR OF -2-PROPYL-3-[(2'-TETRAZOL-5-YL)BIPHEN-4-YL)METHYL] QUINAZOLINONES AS BALANCED AFFINITY ANTAGONISTS OF THE HUMAN AT(1) AND AT(2) RECEPTORS, Bioorganic & medicinal chemistry letters, 5(13), 1995, pp. 1359-1364
IN-VIVO PHARMACOLOGY OF A NOVEL AT(1) SELECTIVE ANGIOTENSIN-II RECEPTOR ANTAGONIST, MK-996
Authors: KIVLIGHN SD ZINGARO GJ GABEL RA BROTEN TP SCHORN TW SCHAFFER LW NAYLOR EM CHAKRAVARTY PK PATCHETT AA GREENLEE WJ SIEGL PKS
Citation: Sd. Kivlighn et al., IN-VIVO PHARMACOLOGY OF A NOVEL AT(1) SELECTIVE ANGIOTENSIN-II RECEPTOR ANTAGONIST, MK-996, American journal of hypertension, 8(1), 1995, pp. 58-66
DISCOVERY OF L-162,313 - A NONPEPTIDE THAT MIMICS THE BIOLOGICAL ACTIONS OF ANGIOTENSIN-II
Authors: KIVLIGHN SD HUCKLE WR ZINGARO GJ RIVERO RA LOTTI VJ CHANG RSL SCHORN TW KEVIN N JOHNSON RG GREENLEE WJ SIEGL PKS
Citation: Sd. Kivlighn et al., DISCOVERY OF L-162,313 - A NONPEPTIDE THAT MIMICS THE BIOLOGICAL ACTIONS OF ANGIOTENSIN-II, American journal of physiology. Regulatory, integrative and comparative physiology, 37(3), 1995, pp. 820-823
QUINAZOLINONE BIPHENYL ACYLSULFONAMIDES - A POTENT NEW CLASS OF ANGIOTENSIN-II RECEPTOR ANTAGONISTS
Authors: CHAKRAVARTY PK STRELITZ RA CHEN TB CHANG RSL LOTTI VJ ZINGARO GJ SCHORN TW KIVLIGHN SD SIEGL PKS PATCHETT AA GREENLEE WJ
Citation: Pk. Chakravarty et al., QUINAZOLINONE BIPHENYL ACYLSULFONAMIDES - A POTENT NEW CLASS OF ANGIOTENSIN-II RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 75-80
TRIAZOLINONES AS NONPEPTIDE ANGIOTENSIN-II ANTAGONISTS .2. DISCOVERY OF A POTENT AND ORALLY-ACTIVE TRIAZOLINONE ACYLSULFONAMIDE
Authors: CHANG LL ASHTON WT FLANAGAN KL NAYLOR EM CHAKRAVARTY PK PATCHETT AA GREENLEE WJ BENDESKY RJ CHEN TB FAUST KA KLING PJ SCHAFFER LW SCHORN TW ZINGARO GJ CHANG RSL LOTTI VJ KIVLIGHN SD SIEGL PKS
Citation: Ll. Chang et al., TRIAZOLINONES AS NONPEPTIDE ANGIOTENSIN-II ANTAGONISTS .2. DISCOVERY OF A POTENT AND ORALLY-ACTIVE TRIAZOLINONE ACYLSULFONAMIDE, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 115-120
L-162,313, A NONPEPTIDE THAT MIMICS THE ACTION OF ANGIOTENSIN-II IN-VIVO
Authors: KIVLIGHN SD ZINGARO GJ RIVERO RA SCHORN TW CHANG RL LOTTI VJ KEVIN N GREENLEE WJ SIEGL PKS
Citation: Sd. Kivlighn et al., L-162,313, A NONPEPTIDE THAT MIMICS THE ACTION OF ANGIOTENSIN-II IN-VIVO, The FASEB journal, 8(5), 1994, pp. 10000879-10000879
A HIGHLY POTENT, ORALLY-ACTIVE IMIDAZO[4,5-B]PYRIDINE BIPHENYLACYLSULFONAMIDE (MK-996-L-159,282) - A NEW ANGIOTENSIN-II RECEPTOR ANTAGONIST
Authors: CHAKRAVARTY PK NAYLOR EM CHEN A CHANG RSL CHEN TB FAUST KA LOTTI VJ KIVLIGHN SD GABLE RA ZINGARO GJ SCHORN TW SCHAFFER LW BROTEN TP SIEGL PKS PATCHETT AA GREENLEE WJ
Citation: Pk. Chakravarty et al., A HIGHLY POTENT, ORALLY-ACTIVE IMIDAZO[4,5-B]PYRIDINE BIPHENYLACYLSULFONAMIDE (MK-996-L-159,282) - A NEW ANGIOTENSIN-II RECEPTOR ANTAGONIST, Journal of medicinal chemistry, 37(24), 1994, pp. 4068-4072
TRIAZOLINONE BIPHENYLSULFONAMIDE DERIVATIVES AS ORALLY-ACTIVE ANGIOTENSIN-II ANTAGONISTS WITH POTENT AT(1) RECEPTOR AFFINITY AND ENHANCED AT(2) AFFINITY
Authors: ASHTON WT CHANG LL FLANAGAN KL HUTCHINS SM NAYLOR EM CHAKRAVARTY PK PATCHETT AA GREENLEE WJ CHEN TB FAUST KA CHANG RSL LOTTI VJ ZINGARO GJ SCHORN TW SIEGL PKS KIVLIGHN SD
Citation: Wt. Ashton et al., TRIAZOLINONE BIPHENYLSULFONAMIDE DERIVATIVES AS ORALLY-ACTIVE ANGIOTENSIN-II ANTAGONISTS WITH POTENT AT(1) RECEPTOR AFFINITY AND ENHANCED AT(2) AFFINITY, Journal of medicinal chemistry, 37(17), 1994, pp. 2808-2824
L-368,899, A POTENT ORALLY-ACTIVE OXYTOCIN ANTAGONIST FOR POTENTIAL USE IN PRETERM LABOR
Authors: PETTIBONE DJ CLINESCHMIDT BV GUIDOTTI MT LIS EV REISS DR WOYDEN CJ BOCK MG EVANS BE FREIDINGER RM HOBBS DW VEBER DF WILLIAMS PD CHIU SHL THOMPSON KL SCHORN TW SIEGL PKS KAUFMAN MJ CUKIERSKI MA HALUSKA GJ COOK MJ NOVY MJ
Citation: Dj. Pettibone et al., L-368,899, A POTENT ORALLY-ACTIVE OXYTOCIN ANTAGONIST FOR POTENTIAL USE IN PRETERM LABOR, Drug development research, 30(3), 1993, pp. 129-142
BIOTRANSFORMATION OF 5-CHLORO-3-PHENYLTHIOINDOLE-2-CARBOXAMIDE (L-734,005) IN RHESUS-MONKEYS AND RAT-LIVER MICROSOMES TO A POTENT HIV-1 REVERSE-TRANSCRIPTASE INHIBITOR
Authors: BALANI SK GOLDMAN ME KAUFFMAN LR VARGA SL OBRIEN JA SMITH SJ OLAH TV RAMJIT HG SCHORN TW PITZENBERGER SM WILLIAMS TM ROONEY CS THEOHARIDES AD
Citation: Sk. Balani et al., BIOTRANSFORMATION OF 5-CHLORO-3-PHENYLTHIOINDOLE-2-CARBOXAMIDE (L-734,005) IN RHESUS-MONKEYS AND RAT-LIVER MICROSOMES TO A POTENT HIV-1 REVERSE-TRANSCRIPTASE INHIBITOR, Drug metabolism and disposition, 21(4), 1993, pp. 598-604
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