AAAAAA

   
Results: 1-21 |
Results: 21
Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists
Authors: Santagada, V Caliendo, G Severino, B Perissutti, E Ceccarelli, F Giusti, L Mazzoni, MR Salvadori, S Temussi, PA
Citation: V. Santagada et al., Probing the shape of a hydrophobic pocket in the active site of delta-opioid antagonists, J PEPT SCI, 7(7), 2001, pp. 374-385
Peptide T revisited: Conformational mimicry of epitopes of anti-HIV proteins
Authors: Picone, D Rivieccio, A Crescenzi, O Caliendo, G Santagada, V Perissutti, E Spisani, S Traniello, S Temussi, PA
Citation: D. Picone et al., Peptide T revisited: Conformational mimicry of epitopes of anti-HIV proteins, J PEPT SCI, 7(4), 2001, pp. 197-207
Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage
Authors: Caliendo, G Santagada, V Perissutti, E Severino, B Fiorino, F Warner, TD Wallace, JL Ifa, DR Antunes, E Cirino, G de Nucci, G
Citation: G. Caliendo et al., Synthesis of substituted benzamides as anti-inflammatory agents that inhibit preferentially cyclooxygenase 1 but do not cause gastric damage, EUR J MED C, 36(6), 2001, pp. 517-530
Synthesis and hydrolysis by cathepsin B of fluorogenic substrates with thegeneral structure benzoyl-X-ARG-MCA containing non-natural basic amino acids at position X
Authors: Melo, RL Pozzo, RCB Alves, LC Perissutti, E Caliendo, G Santagada, V Juliano, L Juliano, MA
Citation: Rl. Melo et al., Synthesis and hydrolysis by cathepsin B of fluorogenic substrates with thegeneral structure benzoyl-X-ARG-MCA containing non-natural basic amino acids at position X, BBA-PROT ST, 1547(1), 2001, pp. 82-94
Microwave-enhanced solution coupling of the alpha,alpha-dialkyl amino acid, Aib
Authors: Santagada, V Fiorino, F Perissutti, E Severino, B De Filippis, V Vivenzio, B Caliendo, G
Citation: V. Santagada et al., Microwave-enhanced solution coupling of the alpha,alpha-dialkyl amino acid, Aib, TETRAHEDR L, 42(31), 2001, pp. 5171-5173
A convenient synthesis of N-Fmoc-N,N '-bis-Boc-7-guanyl-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (Fmoc-N,N '-bis-Boc-7-guanyl-Tic-OH, GTIC)
Authors: Santagada, V Fiorino, F Severino, B Salvadori, S Lazarus, LH Bryant, SD Caliendo, G
Citation: V. Santagada et al., A convenient synthesis of N-Fmoc-N,N '-bis-Boc-7-guanyl-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (Fmoc-N,N '-bis-Boc-7-guanyl-Tic-OH, GTIC), TETRAHEDR L, 42(20), 2001, pp. 3507-3509
Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones
Authors: Santagada, V Perissutti, E Fiorino, F Vivenzio, B Caliendo, C
Citation: V. Santagada et al., Microwave enhanced solution synthesis of 1,4-benzodiazepin-5-ones, TETRAHEDR L, 42(12), 2001, pp. 2397-2400
S-1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids
Authors: Alves, LC Melo, RL Sanderson, SJ Mottram, JC Coombs, GH Caliendo, G Santagada, V Juliano, L Juliano, MA
Citation: Lc. Alves et al., S-1 subsite specificity of a recombinant cysteine proteinase, CPB, of Leishmania mexicana compared with cruzain, human cathepsin L and papain using substrates containing non-natural basic amino acids, EUR J BIOCH, 268(5), 2001, pp. 1206-1212
Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV
Authors: Ialenti, A Santagada, V Caliendo, G Severino, B Fiorino, F Maffia, P Ianaro, A Morelli, F Di Micco, B Carteni, M Stiuso, P Metafora, V Metafora, S
Citation: A. Ialenti et al., Synthesis of novel anti-inflammatory peptides derived from the amino-acid sequence of the bioactive protein SV-IV, EUR J BIOCH, 268(12), 2001, pp. 3399-3406
Human tissue kallikrein S-1 subsite recognition of non-natural basic aminoacids
Authors: Melo, RL Pozzo, RCB Pimenta, DC Perissutti, E Caliendo, G Santagada, V Juliano, L Juliano, MA
Citation: Rl. Melo et al., Human tissue kallikrein S-1 subsite recognition of non-natural basic aminoacids, BIOCHEM, 40(17), 2001, pp. 5226-5232
Determination of 21-hydroxydeflazacort in human plasma by high-performanceliquid chromatography/atmospheric pressure chemical ionization tandem massspectrometry. Application to bioequivalence study
Authors: Ifa, DR Moraes, ME Moraes, MO Santagada, V Caliendo, G de Nucci, G
Citation: Dr. Ifa et al., Determination of 21-hydroxydeflazacort in human plasma by high-performanceliquid chromatography/atmospheric pressure chemical ionization tandem massspectrometry. Application to bioequivalence study, J MASS SPEC, 35(3), 2000, pp. 440-445
Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands
Authors: Caliendo, G Fiorino, F Grieco, P Perissutti, E Santagada, V Severino, B Bruni, G Romeo, MR
Citation: G. Caliendo et al., Synthesis of new 1,2,3-benzotriazin-4-one-arylpiperazine derivatives as 5-HT1A serotonin receptor ligands, BIO MED CH, 8(3), 2000, pp. 533-538
Assessment of substitution in the second pharmacophore of Dmt-Tic analogues
Authors: Santagada, V Balboni, G Caliendo, G Guerrini, R Salvadori, S Bianchi, C Bryant, SD Lazarus, LH
Citation: V. Santagada et al., Assessment of substitution in the second pharmacophore of Dmt-Tic analogues, BIOORG MED, 10(24), 2000, pp. 2745-2748
Clarithromycin bioequivalence study of two oral formulations in healthy human volunteers
Authors: Lerner, FE Caliendo, G Santagada, V Santana, GSM Moraes, MEA De Nucci, G
Citation: Fe. Lerner et al., Clarithromycin bioequivalence study of two oral formulations in healthy human volunteers, INT J CL PH, 38(7), 2000, pp. 345-354
Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase
Authors: Sautebin, L Rombola, L Di Rosa, M Caliendo, G Perissutti, E Grieco, P Severino, B Santagada, V
Citation: L. Sautebin et al., Synthesis and structure-activity of antisense peptides corresponding to the region for CaM-binding domain of the inducible nitric oxide synthase, EUR J MED C, 35(7-8), 2000, pp. 727-732
Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei
Authors: Balboni, G Salvadori, S Guerrini, R Bianchi, C Santagada, V Calliendo, G Bryant, SD Lazarus, LH
Citation: G. Balboni et al., Opioid pseudopeptides containing heteroaromatic or heteroaliphatic nuclei, PEPTIDES, 21(11), 2000, pp. 1663-1671
Protease-activated receptor-2 modulates myocardial ischemia-reperfusion injury in the rat heart
Authors: Napoli, C Cicala, C Wallace, JL de Nigris, F Santagada, V Caliendo, C Franconi, F Ignarro, LJ Cirino, G
Citation: C. Napoli et al., Protease-activated receptor-2 modulates myocardial ischemia-reperfusion injury in the rat heart, P NAS US, 97(7), 2000, pp. 3678-3683
Synthesis and binding affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1-and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives
Authors: Caliendo, G Fiorino, F Grieco, P Perissutti, E Santagada, V Albrizio, S Spadola, L Bruni, G Romeo, MR
Citation: G. Caliendo et al., Synthesis and binding affinities for 5-HT1A, 5-HT2A and 5-HT2C receptors of a series of 1-and 2-(4-arylpiperazinylalkyl)-4-(benzoyl)-1,2,3-triazole derivatives, EUR J MED C, 34(9), 1999, pp. 719-727
Preparation and local anaesthetic activity of benzotriazinone and benzoyltriazole derivatives
Authors: Caliendo, G Fiorino, F Grieco, P Perissutti, E Santagada, V Meli, R Raso, GM Zanesco, A De Nucci, G
Citation: G. Caliendo et al., Preparation and local anaesthetic activity of benzotriazinone and benzoyltriazole derivatives, EUR J MED C, 34(12), 1999, pp. 1043-1051
Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids
Authors: Caliendo, G Fiorino, F Grieco, P Perissutti, E De Luca, S Giuliano, A Santelli, G Califano, D Severino, B Santagada, V
Citation: G. Caliendo et al., Synthesis and biological activity of pseudopeptides inhibitors of Ras farnesyl transferase containing unconventional amino acids, FARMACO, 54(11-12), 1999, pp. 785-790
Synthesis, biological activity and conformational study of 1,4-benzoxazinederivatives as potassium channel modulators
Authors: Caliendo, G Grieco, P Perissutti, E Santagada, V Santini, A Albrizio, S Fattorusso, C Pinto, A Sorrentino, R
Citation: G. Caliendo et al., Synthesis, biological activity and conformational study of 1,4-benzoxazinederivatives as potassium channel modulators, EUR J MED C, 33(12), 1998, pp. 957-967
Risultati: 1-21 |