ACNP - Italian Periodicals Catalogue

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Results: 1-22 |

Results: 22

Discovery of human CCR5 antagonists containing hydantoins for the treatment of HIV-1 infection

Authors: Kim, D Wang, LP Caldwell, CG Chen, P Finke, PE Oates, B MacCoss, M Mills, SG Malkowitz, L Gould, SL DeMartino, JA Springer, MS Hazuda, D Miller, M Kessler, J Danzeisen, R Carver, G Carella, A Holmes, K Lineberger, J Schleif, WA Emini, EA

Citation: D. Kim et al., Discovery of human CCR5 antagonists containing hydantoins for the treatment of HIV-1 infection, BIOORG MED, 11(24), 2001, pp. 3099-3102

Design, synthesis, and SAR of heterocycle-containing antagonists of the human CCR5 receptor for the treatment of HIV-1 infection

Citation: D. Kim et al., Design, synthesis, and SAR of heterocycle-containing antagonists of the human CCR5 receptor for the treatment of HIV-1 infection, BIOORG MED, 11(24), 2001, pp. 3103-3106

Combinatorial synthesis of CCR5 antagonists

Authors: Willoughby, CA Berk, SC Rosauer, KG Degrado, S Chapman, KT Gould, SL Springer, MS Malkowitz, L Schleif, WA Hazuda, D Miller, M Kessler, J Danzeisen, R Holmes, K Lineberger, J Carella, A Carver, G Emini, EA

Citation: Ca. Willoughby et al., Combinatorial synthesis of CCR5 antagonists, BIOORG MED, 11(24), 2001, pp. 3137-3141

1,3,4-trisubstituted pyrrolidine CCR5 receptor antagonists. Part 2: Lead optimization affording selective, orally bioavailable compounds with potent anti-HIV activity

Authors: Hale, JJ Budhu, RJ Holson, EB Finke, PE Oates, B Mills, SG MacCoss, M Gould, SL DeMartino, JA Springer, MS Siciliano, S Malkowitz, L Schleif, WA Hazuda, D Miller, M Kessler, J Danzeisen, R Holmes, K Lineberger, J Carella, A Carver, G Emini, E

Citation: Jj. Hale et al., 1,3,4-trisubstituted pyrrolidine CCR5 receptor antagonists. Part 2: Lead optimization affording selective, orally bioavailable compounds with potent anti-HIV activity, BIOORG MED, 11(20), 2001, pp. 2741-2745

Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 1: Discovery and initial structure-activity relationships for 1-amino-2-phenyl-4-(piperidin-1-yl)butanes

Authors: Dorn, CP Finke, PE Oates, B Budhu, RJ Mills, SG MacCoss, M Malkowitz, L Springer, MS Daugherty, BL Gould, SL DeMartino, JA Siciliano, SJ Carella, A Carver, G Holmes, K Danzeisen, R Hazuda, D Kessler, J Lineberger, J Miller, M Schleif, WA Emini, EA

Citation: Cp. Dorn et al., Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 1: Discovery and initial structure-activity relationships for 1-amino-2-phenyl-4-(piperidin-1-yl)butanes, BIOORG MED, 11(2), 2001, pp. 259-264

Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 2: Structure-activity relationships for substituted 2-aryl-1-[N-(methyl)-N-(phenylsulfonyl) amino]-4-(piperidin-1-yl)butanes

Authors: Finke, PE Meurer, LC Oates, B Mills, SG MacCoss, M Malkowitz, L Springer, MS Daugherty, BL Gould, SL DeMartino, JA Siciliano, SJ Carella, A Carver, G Holmes, K Danzeisen, R Hazuda, D Kessler, J Lineberger, J Miller, M Schleif, WA Emini, EA

Citation: Pe. Finke et al., Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 2: Structure-activity relationships for substituted 2-aryl-1-[N-(methyl)-N-(phenylsulfonyl) amino]-4-(piperidin-1-yl)butanes, BIOORG MED, 11(2), 2001, pp. 265-270

Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 3: A proposed pharmacophore model for 1-[N-(methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)4-[4-(substituted)piperidin-1yl]butanes

Authors: Finke, PE Meurer, LC Oates, B Shah, SK Loebach, JL Mills, SG MacCoss, M Castonguay, L Malkowitz, L Springer, MS Gould, SL DeMartino, JA

Citation: Pe. Finke et al., Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 3: A proposed pharmacophore model for 1-[N-(methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)4-[4-(substituted)piperidin-1yl]butanes, BIOORG MED, 11(18), 2001, pp. 2469-2473

Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 4: Synthesis and structure-activity relationships for 1-[N(methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)-4-(4-(N-(alkyl)-N- (benzyloxycarbonyl)amino)piperidin-1-yl)butanes

Authors: Finke, PE Oates, B Mills, SG MacCoss, M Malkowitz, L Springer, MS Gould, SL DeMartino, JA Carella, A Carver, G Holmes, K Danzeisen, R Hazuda, D Kessler, J Lineberger, J Miller, M Schleif, WA Emini, EA

Citation: Pe. Finke et al., Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 4: Synthesis and structure-activity relationships for 1-[N(methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)-4-(4-(N-(alkyl)-N- (benzyloxycarbonyl)amino)piperidin-1-yl)butanes, BIOORG MED, 11(18), 2001, pp. 2475-2479

1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 1: Discovery of the pyrrolidine scaffold and determination of its stereochemical requirements

Authors: Hale, JJ Budhu, RJ Mills, SG MacCoss, M Malkowitz, L Siciliano, S Gould, SL DeMartino, JA Springer, MS

Citation: Jj. Hale et al., 1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 1: Discovery of the pyrrolidine scaffold and determination of its stereochemical requirements, BIOORG MED, 11(11), 2001, pp. 1437-1440

Mitochondrial versus nuclear gene sequences in deep-level mammalian phylogeny reconstruction

Authors: Springer, MS DeBry, RW Douady, C Amrine, HM Madsen, O de Jong, WW Stanhope, MJ

Citation: Ms. Springer et al., Mitochondrial versus nuclear gene sequences in deep-level mammalian phylogeny reconstruction, MOL BIOL EV, 18(2), 2001, pp. 132-143

Phylogenetics - Which mammalian supertree to bark up?

Authors: Springer, MS de Jong, WW

Citation: Ms. Springer et Ww. De Jong, Phylogenetics - Which mammalian supertree to bark up?, SCIENCE, 291(5509), 2001, pp. 1709

Parallel adaptive radiations in two major clades of placental mammals

Authors: Madsen, O Scally, M Douady, CJ Kao, DJ DeBry, RW Adkins, R Amrine, HM Stanhope, MJ de Jong, WW Springer, MS

Citation: O. Madsen et al., Parallel adaptive radiations in two major clades of placental mammals, NATURE, 409(6820), 2001, pp. 610-614

Integrated fossil and molecular data reconstruct bat echolocation

Authors: Springer, MS Teeling, EC Madsen, O Stanhope, MJ de Jong, WW

Citation: Ms. Springer et al., Integrated fossil and molecular data reconstruct bat echolocation, P NAS US, 98(11), 2001, pp. 6241-6246

CCR5, CXCR4, and CD4 are clustered and closely apposed on microvilli of human macrophages and T cells

Authors: Singer, II Scott, S Kawka, DW Chin, J Daugherty, BL DeMartino, JA DiSalvo, J Gould, SL Lineberger, JE Malkowitz, L Miller, MD Mitnaul, L Siciliano, SJ Staruch, MJ Williams, HR Zweerink, HJ Springer, MS

Citation: Ii. Singer et al., CCR5, CXCR4, and CD4 are clustered and closely apposed on microvilli of human macrophages and T cells, J VIROLOGY, 75(8), 2001, pp. 3779-3790

The chemokine/chemokine-receptor family: potential and progress for therapeutic intervention

Authors: Cascieri, MA Springer, MS

Citation: Ma. Cascieri et Ms. Springer, The chemokine/chemokine-receptor family: potential and progress for therapeutic intervention, CURR OP C B, 4(4), 2000, pp. 420-427

Molecular evidence regarding the origin of echolocation and flight in bats

Authors: Teeling, EC Scally, M Kao, DJ Romagnoli, ML Springer, MS Stanhope, MJ

Citation: Ec. Teeling et al., Molecular evidence regarding the origin of echolocation and flight in bats, NATURE, 403(6766), 2000, pp. 188-192

The CXCR4 agonist ligand stromal derived factor-1 maintains high affinity for receptors in both G(alpha i)-coupled and uncoupled states

Authors: Di Salvo, J Koch, GE Johnson, KE Blake, AD Daugherty, BL DeMartino, JA Sirotina-Meisher, A Liu, Y Springer, MS Cascieri, MA Sullivan, KA

Citation: J. Di Salvo et al., The CXCR4 agonist ligand stromal derived factor-1 maintains high affinity for receptors in both G(alpha i)-coupled and uncoupled states, EUR J PHARM, 409(2), 2000, pp. 143-154

Radiolabeled chemokine binding assays

Authors: Daugherty, BL Siciliano, SJ Springer, MS

Citation: Bl. Daugherty et al., Radiolabeled chemokine binding assays, METH MOL B, 138, 2000, pp. 129-134

Additional support for Afrotheria and Paenungulata, the performance of mitochondrial versus nuclear genes, and the impact of data partitions with heterogeneous base composition

Authors: Springer, MS Amrine, HM Burk, A Stanhope, MJ

Citation: Ms. Springer et al., Additional support for Afrotheria and Paenungulata, the performance of mitochondrial versus nuclear genes, and the impact of data partitions with heterogeneous base composition, SYST BIOL, 48(1), 1999, pp. 65-75

A critical site in the core of the CCR5 chemokine receptor required for binding and infectivity of human immunodeficiency virus type 1

Authors: Siciliano, SJ Kuhmann, SE Weng, YM Madani, N Springer, MS Lineberger, JE Danzeisen, R Miller, MD Kavanaugh, MP DeMartino, JA Kabat, D

Citation: Sj. Siciliano et al., A critical site in the core of the CCR5 chemokine receptor required for binding and infectivity of human immunodeficiency virus type 1, J BIOL CHEM, 274(4), 1999, pp. 1905-1913

Correolide and derivatives are novel immunosuppressants blocking the lymphocyte Kv1.3 potassium channels

Authors: Koo, GC Blake, JT Shah, K Staruch, MJ Dumont, F Wunderler, D Sanchez, M McManus, OB Sirotina-Meisher, A Fischer, P Boltz, RC Goetz, MA Baker, R Bao, JM Kayser, F Rupprecht, KM Parsons, WH Tong, XC Ita, IE Pivnichny, J Vincent, S Cunningham, P Hora, D Feeney, W Kaczorowski, G Springer, MS

Citation: Gc. Koo et al., Correolide and derivatives are novel immunosuppressants blocking the lymphocyte Kv1.3 potassium channels, CELL IMMUN, 197(2), 1999, pp. 99-107

The origin of the Australasian marsupial fauna and the phylogenetic affinities of the enigmatic monito del monte and marsupial mole

Authors: Springer, MS Westerman, M Kavanagh, JR Burk, A Woodburne, MO Kao, DJ Krajewski, C

Citation: Ms. Springer et al., The origin of the Australasian marsupial fauna and the phylogenetic affinities of the enigmatic monito del monte and marsupial mole, P ROY SOC B, 265(1413), 1998, pp. 2381-2386

Risultati: 1-22 |