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Results: 1-12 |
Results: 12
Structure-activity relationship studies on the potent multidrug resistance(MDR) modulator 2-(3,4-dimethoxyphenyl)-2-(methylethyl)-5-[(anthr-9-yl)methylamino]pentanenitrile (MM 36)
Authors: Teodori, E Dei, S Garnier-Suillerot, A Quidu, P Scapecchi, S Budriesi, R
Citation: E. Teodori et al., Structure-activity relationship studies on the potent multidrug resistance(MDR) modulator 2-(3,4-dimethoxyphenyl)-2-(methylethyl)-5-[(anthr-9-yl)methylamino]pentanenitrile (MM 36), MED CHEM RE, 10(9), 2001, pp. 563-576
Structure-activity relationships in 2,2-diphenyl-2-ethylthioacetic acid esters: Unexpected agonistic activity in a series of muscarinic antagonists
Authors: Scapecchi, S Marucci, G Matucci, R Angeli, P Bellucci, C Buccioni, M Dei, S Gualtieri, F Manetti, D Romanelli, MN Teodori, E
Citation: S. Scapecchi et al., Structure-activity relationships in 2,2-diphenyl-2-ethylthioacetic acid esters: Unexpected agonistic activity in a series of muscarinic antagonists, BIO MED CH, 9(5), 2001, pp. 1165-1174
Structure-activity relationships and optimisation of the selective MDR modulator 2-(3,4-dimethoxyphenyl)-5-(9-fluorenylamino)-2-(methylethyl) pentanenitrile and its N-methyl derivative
Authors: Dei, S Teodori, E Garnier-Suillerot, A Gualtieri, F Scapecchi, S Budriesi, R Chiarini, A
Citation: S. Dei et al., Structure-activity relationships and optimisation of the selective MDR modulator 2-(3,4-dimethoxyphenyl)-5-(9-fluorenylamino)-2-(methylethyl) pentanenitrile and its N-methyl derivative, BIO MED CH, 9(10), 2001, pp. 2673-2682
Fluorescent verapamil analogue for monitoring acidic intracellular organelles in Multidrug resistant and sensitive cells
Authors: Mankhetkorn, S Teodori, E Garnier-Suillerot, A
Citation: S. Mankhetkorn et al., Fluorescent verapamil analogue for monitoring acidic intracellular organelles in Multidrug resistant and sensitive cells, CHEM-BIO IN, 137(1), 2001, pp. 1-13
Molecular simplification of 1,4-diazabicyclo[4.3,0]nonan-9-ones gives piperazine derivatives that maintain high nootropic activity
Authors: Manetti, D Ghelardini, C Bartolini, A Dei, S Galeotti, N Gualtieri, F Romanelli, MN Teodori, E
Citation: D. Manetti et al., Molecular simplification of 1,4-diazabicyclo[4.3,0]nonan-9-ones gives piperazine derivatives that maintain high nootropic activity, J MED CHEM, 43(23), 2000, pp. 4499-4507
Design, synthesis, and preliminary pharmacological evaluation of 1,4-diazabicyclo[4.3.0]nonan-9-ones as a new class of highly potent nootropic agents
Authors: Manetti, D Ghelardini, C Bartolini, A Bellucci, C Dei, S Galeotti, N Gualtieri, F Romanelli, MN Scapecchi, S Teodori, E
Citation: D. Manetti et al., Design, synthesis, and preliminary pharmacological evaluation of 1,4-diazabicyclo[4.3.0]nonan-9-ones as a new class of highly potent nootropic agents, J MED CHEM, 43(10), 2000, pp. 1969-1974
Synthesis and binding properties of photoactivable biotin-conjugated verapamil derivatives for the study of P-170 glycoprotein
Authors: Teodori, E Ettori, D Garnier-Suillerot, A Gualtieri, F Manetti, D Romanelli, MN Scapecchi, S
Citation: E. Teodori et al., Synthesis and binding properties of photoactivable biotin-conjugated verapamil derivatives for the study of P-170 glycoprotein, BIO MED CH, 7(9), 1999, pp. 1873-1880
Hybridized and isosteric analogues of N-1-acetyl-N-4-dimethy-piperazinium iodide (ADMP) and N-1-phenyl-N-4-dimethy-piperazinium iodide (DMPP) with central nicotinic action
Authors: Manetti, D Bartolini, A Borea, PA Bellucci, C Dei, S Ghelardini, C Gualtieri, F Romanelli, MN Scapecchi, S Teodori, E Varani, K
Citation: D. Manetti et al., Hybridized and isosteric analogues of N-1-acetyl-N-4-dimethy-piperazinium iodide (ADMP) and N-1-phenyl-N-4-dimethy-piperazinium iodide (DMPP) with central nicotinic action, BIO MED CH, 7(3), 1999, pp. 457-465
Design, synthesis, and in vitro activity of catamphiphilic reverters of multidrug resistance: Discovery of a selective, highly efficacious chemosensitizer with potency in the nanomolar range
Authors: Teodori, E Dei, S Quidu, P Budriesi, R Chiarini, A Garnier-Suillerot, A Gualtieri, F Manetti, D Romanelli, MN Scapecchi, S
Citation: E. Teodori et al., Design, synthesis, and in vitro activity of catamphiphilic reverters of multidrug resistance: Discovery of a selective, highly efficacious chemosensitizer with potency in the nanomolar range, J MED CHEM, 42(10), 1999, pp. 1687-1697
Partial inhibition of the P-glycoprotein-mediated transport of anthracyclines in viable resistant K562 cells after irradiation in the presence of a verapamil analogue
Authors: Mankhetkorn, S Teodori, E Garnier-Suillerot, A
Citation: S. Mankhetkorn et al., Partial inhibition of the P-glycoprotein-mediated transport of anthracyclines in viable resistant K562 cells after irradiation in the presence of a verapamil analogue, CHEM-BIO IN, 121(2), 1999, pp. 125-140
Binding profiles of a series of 2-arylpropionic acid esters on cloned human muscarinic receptor subtypes (m(1)-m(5)) and their relationship to nootropic activity
Authors: Ghelardini, C Mizuma, I Gualtieri, F Bartolini, A Galeotti, N Romanelli, MN Teodori, E
Citation: C. Ghelardini et al., Binding profiles of a series of 2-arylpropionic acid esters on cloned human muscarinic receptor subtypes (m(1)-m(5)) and their relationship to nootropic activity, ARZNEI-FOR, 49(6), 1999, pp. 483-488
Further structure-activity relationships in the series of tropanyl esters endowed with potent antinociceptive activity
Authors: Scapecchi, S Giorgi, A Bellucci, C Dei, S Ghelardini, C Manetti, D Romanelli, MN Teodori, E
Citation: S. Scapecchi et al., Further structure-activity relationships in the series of tropanyl esters endowed with potent antinociceptive activity, FARMACO, 53(12), 1998, pp. 764-772
Risultati: 1-12 |