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Results: 1-21 |
Results: 21
Synthesis and anti-HIV activity of cosalane analogues incorporating two dichlorodisalicylmethane pharmacophore fragments
Authors: Casimiro-Garcia, A De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Fanwick, PE Cushman, M
Citation: A. Casimiro-garcia et al., Synthesis and anti-HIV activity of cosalane analogues incorporating two dichlorodisalicylmethane pharmacophore fragments, BIO MED CH, 9(11), 2001, pp. 2827-2841
SJ-3366, a unique and highly potent nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1 (HIV-1) that also inhibits HIV-2
Authors: Buckheit, RW Watson, K Fliakas-Boltz, V Russell, J Loftus, TL Osterling, MC Turpin, JA Pallansch, LA White, EL Lee, JW Lee, SH Oh, JW Kwon, HS Chung, SG Cho, EH
Citation: Rw. Buckheit et al., SJ-3366, a unique and highly potent nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1 (HIV-1) that also inhibits HIV-2, ANTIM AG CH, 45(2), 2001, pp. 393-400
Synthesis and anti-HIV activity of a bile acid analog of cosalane
Authors: Kannan, A De Clercq, E Pannecouque, C Witvrouw, M Hartman, TL Turpin, JA Buckheit, RW Cushman, M
Citation: A. Kannan et al., Synthesis and anti-HIV activity of a bile acid analog of cosalane, TETRAHEDRON, 57(46), 2001, pp. 9385-9391
The secondary amine/nitric oxide complex ion R2N[N(O)NO](-) as nucleophileand leaving group in SNAr reactions
Authors: Saavedra, JE Srinivasan, A Bonifant, CL Chu, JX Shanklin, AP Flippen-Anderson, JL Rice, WG Turpin, JA Davies, KM Keefer, LK
Citation: Je. Saavedra et al., The secondary amine/nitric oxide complex ion R2N[N(O)NO](-) as nucleophileand leaving group in SNAr reactions, J ORG CHEM, 66(9), 2001, pp. 3090-3098
Solid-phase synthesis of the alkenyldiarylmethane (ADAM) series of non-nucleoside HIV-1 reverse transcriptase inhibitors
Authors: Xu, GZ Loftus, TL Wargo, H Turpin, JA Buckheit, RW Cushman, M
Citation: Gz. Xu et al., Solid-phase synthesis of the alkenyldiarylmethane (ADAM) series of non-nucleoside HIV-1 reverse transcriptase inhibitors, J ORG CHEM, 66(18), 2001, pp. 5958-5964
Correlation of anti-HIV activity with anion spacing in a series of cosalane analogues with extended polycarboxylate pharmacophores
Authors: Santhosh, KC Paul, GC De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Kc. Santhosh et al., Correlation of anti-HIV activity with anion spacing in a series of cosalane analogues with extended polycarboxylate pharmacophores, J MED CHEM, 44(5), 2001, pp. 703-714
The biological effects of structural variation at the meta position of thearomatic rings and at the end of the alkenyl chain in the alkenyldiarylmethane series of non-nucleoside reverse transcriptase inhibitors
Authors: Xu, GZ Micklatcher, M Silvestri, MA Hartman, TL Burrier, J Osterling, MC Wargo, H Turpin, JA Buckheit, RW Cushman, M
Citation: Gz. Xu et al., The biological effects of structural variation at the meta position of thearomatic rings and at the end of the alkenyl chain in the alkenyldiarylmethane series of non-nucleoside reverse transcriptase inhibitors, J MED CHEM, 44(24), 2001, pp. 4092-4113
Inhibitors of HIV cellular fusion
Authors: Turpin, JA Howard, OMZ
Citation: Ja. Turpin et Omz. Howard, Inhibitors of HIV cellular fusion, EXPERT OP T, 10(12), 2000, pp. 1899-1909
Synthesis and anti-HIV activity of cosalane analogues incorporating nitrogen in the linker chain
Authors: Casimiro-Garcia, A De Clercq, E Pannecouque, C Witvrouw, M Stup, TL Turpin, JA Buckheit, RW Cushman, M
Citation: A. Casimiro-garcia et al., Synthesis and anti-HIV activity of cosalane analogues incorporating nitrogen in the linker chain, BIO MED CH, 8(1), 2000, pp. 191-200
Anti-HIV activity of a series of cosalane amino acid conjugates
Authors: Santhosh, KC De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Kc. Santhosh et al., Anti-HIV activity of a series of cosalane amino acid conjugates, BIOORG MED, 10(22), 2000, pp. 2505-2508
Identification of optimal anion spacing for anti-HIV activity in a series of cosalane tetracarboxylates
Authors: Paul, GC De Clercq, E Pannecouque, C Witvrouw, M Loftus, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Gc. Paul et al., Identification of optimal anion spacing for anti-HIV activity in a series of cosalane tetracarboxylates, BIOORG MED, 10(18), 2000, pp. 2149-2152
Inactivation of HIV-1 nucleocapsid protein P7 by pyridinioalkanoyl thioesters - Characterization of reaction products and proposed mechanism of action
Authors: Basrur, V Song, YS Mazur, SJ Higashimoto, Y Turpin, JA Rice, WG Inman, JK Appella, E
Citation: V. Basrur et al., Inactivation of HIV-1 nucleocapsid protein P7 by pyridinioalkanoyl thioesters - Characterization of reaction products and proposed mechanism of action, J BIOL CHEM, 275(20), 2000, pp. 14890-14897
Oral Montelukast compared with inhaled salmeterol to prevent exercise-induced bronchoconstriction - A randomized, double-blind trial
Authors: Edelman, JM Turpin, JA Bronsky, EA Grossman, J Kemp, JP Ghannam, AF DeLucca, PT Gormley, GJ Pearlman, DS
Citation: Jm. Edelman et al., Oral Montelukast compared with inhaled salmeterol to prevent exercise-induced bronchoconstriction - A randomized, double-blind trial, ANN INT MED, 132(2), 2000, pp. 97-104
Synthesis of (R)-(-)-1-piperidino-3,3-dimethylbutan-2-ol: Application in the molar scale asymmetric ethylation of trans-crotonaldehyde
Authors: Hoard, DW Moher, ED Turpin, JA
Citation: Dw. Hoard et al., Synthesis of (R)-(-)-1-piperidino-3,3-dimethylbutan-2-ol: Application in the molar scale asymmetric ethylation of trans-crotonaldehyde, ORG PROC R, 3(1), 1999, pp. 64-66
Synthesis and anti-HIV activity of cosalane analogues with substituted benzoic acid rings attached to the pharmacophore through methylene and amide linkers
Authors: Ruell, JA De Clercq, E Pannecouque, C Witvrouw, M Stup, TL Turpin, JA Buckheit, RW Cushman, M
Citation: Ja. Ruell et al., Synthesis and anti-HIV activity of cosalane analogues with substituted benzoic acid rings attached to the pharmacophore through methylene and amide linkers, J ORG CHEM, 64(16), 1999, pp. 5858-5866
Chicoric acid analogues as HIV-1 integrase inhibitors
Authors: Lin, ZW Neamati, N Zhao, H Kiryu, Y Turpin, JA Aberham, C Strebel, K Kohn, K Witvrouw, M Pannecouque, C Debyser, Z De Clercq, E Rice, WG Pommier, Y Burke, TR
Citation: Zw. Lin et al., Chicoric acid analogues as HIV-1 integrase inhibitors, J MED CHEM, 42(8), 1999, pp. 1401-1414
Novel modifications in the alkenyldiarylmethane (ADAM) series of non-nucleoside reverse transcriptase inhibitors
Authors: Casimiro-Garcia, A Micklatcher, M Turpin, JA Stup, TL Watson, K Buckheit, RW Cushman, M
Citation: A. Casimiro-garcia et al., Novel modifications in the alkenyldiarylmethane (ADAM) series of non-nucleoside reverse transcriptase inhibitors, J MED CHEM, 42(23), 1999, pp. 4861-4874
Thiazolothiazepine inhibitors of HIV-1 integrase
Authors: Neamati, N Turpin, JA Winslow, HE Christensen, JL Williamson, K Orr, A Rice, WG Pommier, Y Garofalo, A Brizzi, A Campiani, G Fiorini, I Nacci, V
Citation: N. Neamati et al., Thiazolothiazepine inhibitors of HIV-1 integrase, J MED CHEM, 42(17), 1999, pp. 3334-3341
Extension of the polyanionic cosalane pharmacophore as a strategy for increasing anti-HIV potency
Authors: Cushman, M Insaf, S Paul, G Ruell, JA De Clercq, E Schols, D Pannecouque, C Witvrouw, M Schaeffer, CA Turpin, JA Williamson, K Rice, WG
Citation: M. Cushman et al., Extension of the polyanionic cosalane pharmacophore as a strategy for increasing anti-HIV potency, J MED CHEM, 42(10), 1999, pp. 1767-1777
Synthesis and biological properties of novel pyridinioalkanoyl thiolesters(PATE) as anti-HTV-1 agents that target the viral nucleocapsid protein zinc fingers
Authors: Turpin, JA Song, YS Inman, JK Huang, MJ Wallqvist, A Maynard, A Covell, DG Rice, WG Appella, E
Citation: Ja. Turpin et al., Synthesis and biological properties of novel pyridinioalkanoyl thiolesters(PATE) as anti-HTV-1 agents that target the viral nucleocapsid protein zinc fingers, J MED CHEM, 42(1), 1999, pp. 67-86
Naturally occurring CCR5 extracellular and transmembrane domain variants affect HIV-1 co-receptor and ligand binding function
Authors: Howard, OMZ Shirakawa, AK Turpin, JA Maynard, A Tobin, GJ Carrington, M Oppenheim, JJ Dean, M
Citation: Omz. Howard et al., Naturally occurring CCR5 extracellular and transmembrane domain variants affect HIV-1 co-receptor and ligand binding function, J BIOL CHEM, 274(23), 1999, pp. 16228-16234
Risultati: 1-21 |