Authors:
Lobaton, E
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Perez-Perez, MJ
Jimeno, ML
San-Felix, A
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: E. Lobaton et al., "Second generation" of TSAO compounds directed against HIV-1 TSAO-resistant strains, NUCLEOS NUC, 20(4-7), 2001, pp. 707-710
Authors:
Chamorro, C
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De Clercq, E
Balzarini, J
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San-Felix, A
Camarasa, MJ
Citation: C. Chamorro et al., Identification of a novel family of nucleosides that specifically inhibit HIV-1 reverse transcriptase, BIOORG MED, 11(23), 2001, pp. 3085-3088
Authors:
Pelemans, H
Aertsen, A
Van Laethem, K
Vandamme, AM
De Clercq, E
Perez-Perez, MJ
San-Felix, A
Velazquez, S
Camarasa, MJ
Balzarini, J
Citation: H. Pelemans et al., Site-directed mutagenesis of human immunodeficiency virus type 1 reverse transcriptase at amino acid position 138, VIROLOGY, 280(1), 2001, pp. 97-106
Authors:
Balzarini, J
Camarasa, MJ
Perez-Perez, MJ
San-Fleix, A
Velazquez, S
Perno, CF
De Clercq, E
Anderson, JN
Karlsson, A
Citation: J. Balzarini et al., Exploitation of the low fidelity of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase and the nucleotide composition bias in the HIV-1 genome to alter the drug resistance development of HIV, J VIROLOGY, 75(13), 2001, pp. 5772-5777
Authors:
Rodriguez-Barrios, F
Perez, C
Lobaton, E
Velazquez, S
Chamorro, C
San-Felix, A
Perez-Perez, MJ
Camarasa, MJ
Pelemans, H
Balzarini, J
Gago, F
Citation: F. Rodriguez-barrios et al., Identification of a putative binding site for [2 ',5 '-bis-O-(tert-butyldimethylsilyl)beta-D-ribofuranosyl]-3 '-spiro-5 ''-(4 ''-amino-1 '',2 ''-oxathiole-2 '',2 ''-dioxide)thymine (TSAO) derivatives at the p51-p66 interfaceof HIV-1 reverse transcriptase, J MED CHEM, 44(12), 2001, pp. 1853-1865
Citation: E. Lobaton et al., An efficient synthesis of 3 '-spiro sultone nucleosides functionalized on the sultone moiety via Pd-catalyzed cross-coupling reaction, SYNLETT, (9), 2000, pp. 1312-1314
Authors:
Camarasa, MJ
San-Felix, A
Perez-Perez, MJ
Velazquez, S
Alvarez, R
Chamorro, C
Jimeno, ML
Perez, C
Gago, F
De Clercq, E
Balzarini, J
Citation: Mj. Camarasa et al., HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique?, J CARB CHEM, 19(4-5), 2000, pp. 451-469
Authors:
McGuigan, C
Brancale, A
Barucki, H
Srinivasan, S
Jones, G
Pathirana, R
Blewett, S
Alvarez, R
Yarnold, CJ
Carangio, A
Velazquez, S
Andrei, G
Snoeck, R
De Clercq, E
Balzarini, J
Citation: C. Mcguigan et al., Fluorescent bicyclic furo pyrimidine deoxynucleoside analogs as potent andselective inhibitors of VZV and potential future drugs for the treatment of chickenpox and shingles, DRUG FUTURE, 25(11), 2000, pp. 1151-1161
Authors:
Chamorro, C
Velazquez, S
Jimeno, ML
Perez-Perez, MJ
Lobaton, E
Tunon, V
Esteban-Gamboa, A
Gago, F
De Clercq, E
Balzarini, J
Camarasa, MJ
San-Felix, A
Citation: C. Chamorro et al., Unexpected results in the reaction of 5 '-tosyl TSAO-m(3)t with amines, NUCLEOS NUC, 18(4-5), 1999, pp. 715-716
Authors:
Velazquez, S
Tunon, V
Jimeno, ML
Perez-Perez, MJ
San-Felix, A
Chamorro, C
Lobaton, E
Esteban-Gamboa, A
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: S. Velazquez et al., Novel series of [ddN]-[TSAO-T] heterodimers as potential bi-functional inhibitors of HIV-1 RT. Studies in the linker and ddN region, NUCLEOS NUC, 18(4-5), 1999, pp. 1029-1030
Authors:
Camarasa, MJ
Jimeno, ML
Perez-Perez, MJ
Alvarez, R
Velazquez, S
Lozano, A
Citation: Mj. Camarasa et al., Synthesis, NMR studies and theoretical calculations of novel 3-spiro-branched ribofuranoses, TETRAHEDRON, 55(41), 1999, pp. 12187-12200
Authors:
Saboulard, D
Naesens, L
Cahard, D
Salgado, A
Pathirana, R
Velazquez, S
McGuigan, C
De Clercq, E
Balzarini, J
Citation: D. Saboulard et al., Characterization of the activation pathway of phosphoramidate triester prodrugs of stavudine and zidovudine, MOLEC PHARM, 56(4), 1999, pp. 693-704
Authors:
Velazquez, S
Tunon, V
Jimeno, ML
Chamorro, C
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: S. Velazquez et al., Potential multifunctional inhibitors of HIV-1 reverse transcriptase. Novel[AZT]-[TSAO-T] and [d4T]-[TSAO-T] heterodimers modified in the linker and in the dideoxynucleoside region, J MED CHEM, 42(25), 1999, pp. 5188-5196
Authors:
McGuigan, C
Yarnold, CJ
Jones, G
Velazquez, S
Barucki, H
Brancale, A
Andrei, G
Snoeck, R
De Clercq, E
Balzarini, J
Citation: C. Mcguigan et al., Potent and selective inhibition of varicella-zoster virus (VZV) by nucleoside analogues with an unusual bicyclic base, J MED CHEM, 42(22), 1999, pp. 4479-4484
Authors:
Velazquez, S
Alvarez, R
Perez, C
Gago, F
De Clercq, E
Balzarini, J
Camarasa, MJ
Citation: S. Velazquez et al., Regiospecific synthesis and anti-human immunodeficiency virus activity of novel 5-substituted N-alkylcarbamoyl and N,N-dialkyl carbamoyl 1,2,3-triazole-TSAO analogues, ANTIVIR CHE, 9(6), 1998, pp. 481-489
Authors:
Gomez, AM
Mantecon, S
Velazquez, S
Valverde, S
Herczegh, P
Lopez, JC
Citation: Am. Gomez et al., Carbohydrates to carbocycles: Regio- and stereoselectivity in the intramolecular [2+2] photocycloaddition of dienic 2-enono-delta-lactones, SYNLETT, (12), 1998, pp. 1402-1404