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Results: 1-25 | 26-33
Results: 1-25/33
N-(2-(4-HYDROXYPHENYL)ETHYL)-4-CHLOROCINNAMIDE - A NOVEL ANTAGONIST AT THE 1A 2B NMDA RECEPTOR SUBTYPE/
Authors: TAMIZ AP WHITTEMORE ER SCHELKUN RM YUEN PW WOODWARD RM CAI SX WEBER E KEANA JFW
Citation: Ap. Tamiz et al., N-(2-(4-HYDROXYPHENYL)ETHYL)-4-CHLOROCINNAMIDE - A NOVEL ANTAGONIST AT THE 1A 2B NMDA RECEPTOR SUBTYPE/, Bioorganic & medicinal chemistry letters, 8(2), 1998, pp. 199-200
SUBSTITUTED 3-BETA-PHENYLETHYNYL DERIVATIVES OF 3-ALPHA-HYDROXY-5-ALPHA-PREGNAN-20-ONE - REMARKABLY POTENT NEUROACTIVE STEROID MODULATORS OF GAMMA-AMINOBUTYRIC ACID(A) RECEPTORS
Authors: HAWKINSON JE ACOSTABURRUEL M YANG KC HOGENKAMP DJ CHEN JS LAN NC DREWE JA WHITTEMORE ER WOODWARD RM CARTER RB UPASANI RB
Citation: Je. Hawkinson et al., SUBSTITUTED 3-BETA-PHENYLETHYNYL DERIVATIVES OF 3-ALPHA-HYDROXY-5-ALPHA-PREGNAN-20-ONE - REMARKABLY POTENT NEUROACTIVE STEROID MODULATORS OF GAMMA-AMINOBUTYRIC ACID(A) RECEPTORS, The Journal of pharmacology and experimental therapeutics, 287(1), 1998, pp. 198-207
STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF BIS(PHENYLALKYL)AMINES - POTENT SUBTYPE-SELECTIVE INHIBITORS OF N-METHYL-D-ASPARTATE RECEPTORS
Authors: TAMIZ AP WHITTEMORE ER ZHOU ZL HUANG JC DREWE JA CHEN JC CAI SX WEBER E WOODWARD RM KEANA JFW
Citation: Ap. Tamiz et al., STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF BIS(PHENYLALKYL)AMINES - POTENT SUBTYPE-SELECTIVE INHIBITORS OF N-METHYL-D-ASPARTATE RECEPTORS, Journal of medicinal chemistry, 41(18), 1998, pp. 3499-3506
SYNTHESIS OF -1-PHENYL-3,5-DIHYDRO-4H-2,3-BENZODIAZEPINE-4-ONES AS NOVEL AND POTENT NONCOMPETITIVE AMPA RECEPTOR ANTAGONISTS
Authors: WANG Y KONKOY CS ILYIN VI VANOVER KE CARTER RB WEBER E KEANA JFW WOODWARD RM CAI SX
Citation: Y. Wang et al., SYNTHESIS OF -1-PHENYL-3,5-DIHYDRO-4H-2,3-BENZODIAZEPINE-4-ONES AS NOVEL AND POTENT NONCOMPETITIVE AMPA RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 41(14), 1998, pp. 2621-2625
ANTINOCICEPTIVE EFFECTS OF NMDA AND NON-NMDA RECEPTOR ANTAGONISTS IN THE TAIL-FLICK TEST IN MICE
Authors: LUTFY K CAI SX WOODWARD RM WEBER E
Citation: K. Lutfy et al., ANTINOCICEPTIVE EFFECTS OF NMDA AND NON-NMDA RECEPTOR ANTAGONISTS IN THE TAIL-FLICK TEST IN MICE, Pain, 70(1), 1997, pp. 31-40
ANTAGONISM OF N-METHYL-D-ASPARTATE RECEPTORS BY SIGMA-SITE LIGANDS - POTENCY, SUBTYPE-SELECTIVITY AND MECHANISMS OF INHIBITION
Authors: WHITTEMORE ER ILYIN VI WOODWARD RM
Citation: Er. Whittemore et al., ANTAGONISM OF N-METHYL-D-ASPARTATE RECEPTORS BY SIGMA-SITE LIGANDS - POTENCY, SUBTYPE-SELECTIVITY AND MECHANISMS OF INHIBITION, The Journal of pharmacology and experimental therapeutics, 282(1), 1997, pp. 326-338
PARTIAL AGONISM BY 3-ALPHA,21-DIHYDROXY-5-BETA-PREGNAN-20-ONE AT THE GAMMA-AMINOBUTYRIC-ACID, RECEPTOR NEUROSTEROID SITE
Authors: XUE BG WHITTEMORE ER PARK CH WOODWARD RM LAN NC GEE KW
Citation: Bg. Xue et al., PARTIAL AGONISM BY 3-ALPHA,21-DIHYDROXY-5-BETA-PREGNAN-20-ONE AT THE GAMMA-AMINOBUTYRIC-ACID, RECEPTOR NEUROSTEROID SITE, The Journal of pharmacology and experimental therapeutics, 281(3), 1997, pp. 1095-1101
STRUCTURE-ACTIVITY-RELATIONSHIPS OF ALKYL-SUBSTITUTED AND ALKOXY-SUBSTITUTED 1,4-DIHYDROQUINOXALINE-2,3-DIONES - POTENT AND SYSTEMICALLY ACTIVE ANTAGONISTS FOR THE GLYCINE SITE OF THE NMDA RECEPTOR
Authors: CAI SX KHER SM ZHOU ZL ILYIN V ESPITIA SA TRAN M HAWKINSON JE WOODWARD RM WEBER E KEANA JFW
Citation: Sx. Cai et al., STRUCTURE-ACTIVITY-RELATIONSHIPS OF ALKYL-SUBSTITUTED AND ALKOXY-SUBSTITUTED 1,4-DIHYDROQUINOXALINE-2,3-DIONES - POTENT AND SYSTEMICALLY ACTIVE ANTAGONISTS FOR THE GLYCINE SITE OF THE NMDA RECEPTOR, Journal of medicinal chemistry, 40(5), 1997, pp. 730-738
A)-7-SUBSTITUTED-1,4-DIHYDROQUINOXALINE-2,3-DIONES - NOVEL, SYSTEMICALLY ACTIVE AND BROAD-SPECTRUM ANTAGONISTS FOR NMDA GLYCINE, AMPA, AND KAINATE RECEPTORS/
Authors: CAI SX HUANG JC ESPITIA SA TRAN M ILYIN VI HAWKINSON JE WOODWARD RM WEBER E KEANA JFW
Citation: Sx. Cai et al., A)-7-SUBSTITUTED-1,4-DIHYDROQUINOXALINE-2,3-DIONES - NOVEL, SYSTEMICALLY ACTIVE AND BROAD-SPECTRUM ANTAGONISTS FOR NMDA GLYCINE, AMPA, AND KAINATE RECEPTORS/, Journal of medicinal chemistry, 40(22), 1997, pp. 3679-3686
SYNTHESIS OF RACEMIC 9-TETRAHYDRO-3-HYDROXY-1H-1-BENZAZEPINE-2,5-DIONES AS ANTAGONISTS OF N-METHYL-D-ASPARTATE (NMDA) AND LPHA-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID (AMPA) RECEPTORS
Authors: GUZIKOWSKI AP WHITTEMORE ER WOODWARD RM WEBER E KEANA JFW
Citation: Ap. Guzikowski et al., SYNTHESIS OF RACEMIC 9-TETRAHYDRO-3-HYDROXY-1H-1-BENZAZEPINE-2,5-DIONES AS ANTAGONISTS OF N-METHYL-D-ASPARTATE (NMDA) AND LPHA-AMINO-3-HYDROXY-5-METHYLISOXAZOLE-4-PROPIONIC ACID (AMPA) RECEPTORS, Journal of medicinal chemistry, 40(15), 1997, pp. 2424-2429
SYNTHESIS AND IN-VITRO ACTIVITY OF 3-BETA-SUBSTITUTED-3-ALPHA-HYDROXYPREGNAN-20-ONES - ALLOSTERIC MODULATORS OF THE GABA(A) RECEPTOR
Authors: HOGENKAMP DJ TAHIR SH HAWKINSON JE UPASANI RB ALAUDDIN M KIMBROUGH CL ACOSTABURRUEL M WHITTEMORE ER WOODWARD RM LAN NC GEE KW BOLGER MB
Citation: Dj. Hogenkamp et al., SYNTHESIS AND IN-VITRO ACTIVITY OF 3-BETA-SUBSTITUTED-3-ALPHA-HYDROXYPREGNAN-20-ONES - ALLOSTERIC MODULATORS OF THE GABA(A) RECEPTOR, Journal of medicinal chemistry, 40(1), 1997, pp. 61-72
ROXY-3-BETA-(PHENYLETHYNYL)-5-BETA-PREGNAN-20-ONES - SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF NEUROACTIVE STEROIDS WITH HIGH-AFFINITY FOR GABA(A) RECEPTORS
Authors: UPASANI RB YANG KC ACOSTABURRUEL M KONKOY CS MCLELLAN JA WOODWARD RM LAN NC CARTER RB HAWKINSON JE
Citation: Rb. Upasani et al., ROXY-3-BETA-(PHENYLETHYNYL)-5-BETA-PREGNAN-20-ONES - SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF NEUROACTIVE STEROIDS WITH HIGH-AFFINITY FOR GABA(A) RECEPTORS, Journal of medicinal chemistry, 40(1), 1997, pp. 73-84
SUBTYPE-SELECTIVE ANTAGONISM OF NMDA RECEPTORS BY NYLIDRIN
Authors: WHITTEMORE ER ILYIN VI KONKOY CS WOODWARD RM
Citation: Er. Whittemore et al., SUBTYPE-SELECTIVE ANTAGONISM OF NMDA RECEPTORS BY NYLIDRIN, European journal of pharmacology, 337(2-3), 1997, pp. 197-208
1-HYDROXY-1,4-DIHYDROQUINOXALINE-2,3-DIONES - NOVEL ANTAGONISTS AT NMDA RECEPTOR GLYCINE SITES
Authors: ZHENG H ESPITIA SA ILYIN V HAWKINSON JE WOODWARD RM WEBER E KEANA JFW
Citation: H. Zheng et al., 1-HYDROXY-1,4-DIHYDROQUINOXALINE-2,3-DIONES - NOVEL ANTAGONISTS AT NMDA RECEPTOR GLYCINE SITES, Bioorganic & medicinal chemistry letters, 6(4), 1996, pp. 439-440
THE FIRST SELECTIVE ANTAGONIST FOR A GABA(C) RECEPTOR
Authors: MURATA Y WOODWARD RM MILEDI R OVERMAN LE
Citation: Y. Murata et al., THE FIRST SELECTIVE ANTAGONIST FOR A GABA(C) RECEPTOR, Bioorganic & medicinal chemistry letters, 6(17), 1996, pp. 2073-2076
SUBTYPE-SELECTIVE INHIBITION OF N-METHYL-D-ASPARTATE RECEPTORS BY HALOPERIDOL
Authors: ILYIN VI WHITTEMORE ER GUASTELLA J WEBER E WOODWARD RM
Citation: Vi. Ilyin et al., SUBTYPE-SELECTIVE INHIBITION OF N-METHYL-D-ASPARTATE RECEPTORS BY HALOPERIDOL, Molecular pharmacology, 50(6), 1996, pp. 1541-1550
PHARMACOLOGY OF THE HUMAN GAMMA-AMINOBUTYRIC ACID(A) RECEPTOR ALPHA-4SUBUNIT EXPRESSED IN XENOPUS-LAEVIS OOCYTES
Authors: WHITTEMORE ER YANG W DREWE JA WOODWARD RM
Citation: Er. Whittemore et al., PHARMACOLOGY OF THE HUMAN GAMMA-AMINOBUTYRIC ACID(A) RECEPTOR ALPHA-4SUBUNIT EXPRESSED IN XENOPUS-LAEVIS OOCYTES, Molecular pharmacology, 50(5), 1996, pp. 1364-1375
DESIGN AND IN-VITRO PHARMACOLOGY OF A SELECTIVE GAMMA-AMINOBUTYRIC ACID(C) RECEPTOR ANTAGONIST
Authors: RAGOZZINO D WOODWARD RM MURATA Y EUSEBI F OVERMAN LE MILEDI R
Citation: D. Ragozzino et al., DESIGN AND IN-VITRO PHARMACOLOGY OF A SELECTIVE GAMMA-AMINOBUTYRIC ACID(C) RECEPTOR ANTAGONIST, Molecular pharmacology, 50(4), 1996, pp. 1024-1030
ROXY-3-BETA-TRIFLUOROMETHYL-5-ALPHA-PREGNAN-20-ONE (CO-2-1970) - A PARTIAL AGONIST AT THE NEUROACTIVE STEROID SITE OF THE GAMMA-AMINOBUTYRIC-ACID(A) RECEPTOR
Authors: HAWKINSON JE DREWE JA KIMBROUGH CL CHEN JS HOGENKAMP DJ LAN NC GEE KW SHEN KZ WHITTEMORE ER WOODWARD RM
Citation: Je. Hawkinson et al., ROXY-3-BETA-TRIFLUOROMETHYL-5-ALPHA-PREGNAN-20-ONE (CO-2-1970) - A PARTIAL AGONIST AT THE NEUROACTIVE STEROID SITE OF THE GAMMA-AMINOBUTYRIC-ACID(A) RECEPTOR, Molecular pharmacology, 49(5), 1996, pp. 897-906
ANALOGS OF 3-HYDROXY-1H-1-BENZAZEPINE-2,5-DIONE - STRUCTURE-ACTIVITY RELATIONSHIP AT N-METHYL-D-ASPARTATE RECEPTOR GLYCINE SITES
Authors: GUZIKOWSKI AP CAI SX ESPITIA SA HAWKINSON JE HUETTNER JE NOGALES DF TRAN M WOODWARD RM WEBER E KEANA JFW
Citation: Ap. Guzikowski et al., ANALOGS OF 3-HYDROXY-1H-1-BENZAZEPINE-2,5-DIONE - STRUCTURE-ACTIVITY RELATIONSHIP AT N-METHYL-D-ASPARTATE RECEPTOR GLYCINE SITES, Journal of medicinal chemistry, 39(23), 1996, pp. 4643-4653
STRUCTURE-ACTIVITY RELATIONSHIPS OF 4-HYDROXY-3-NITROQUINOLIN-2(1H)-ONES AS NOVEL ANTAGONISTS AT THE GLYCINE SITE OF N-METHYL-D-ASPARTATE RECEPTORS
Authors: CAI SX ZHOU ZL HUANG JC WHITTEMORE ER EGBUWOKU ZO HAWKINSON JE WOODWARD RM WEBER E KEANA JFW
Citation: Sx. Cai et al., STRUCTURE-ACTIVITY RELATIONSHIPS OF 4-HYDROXY-3-NITROQUINOLIN-2(1H)-ONES AS NOVEL ANTAGONISTS AT THE GLYCINE SITE OF N-METHYL-D-ASPARTATE RECEPTORS, Journal of medicinal chemistry, 39(23), 1996, pp. 4682-4686
SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE 3-OXIMES - NOVEL AND HIGHLY POTENT ANTAGONISTS FOR NMDA RECEPTOR GLYCINE SITE
Authors: CAI SX ZHOU ZL HUANG JC WHITTEMORE ER EGBUWOKU ZO LU YX HAWKINSON JE WOODWARD RM WEBER E KEANA JFW
Citation: Sx. Cai et al., SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE 3-OXIMES - NOVEL AND HIGHLY POTENT ANTAGONISTS FOR NMDA RECEPTOR GLYCINE SITE, Journal of medicinal chemistry, 39(17), 1996, pp. 3248-3255
PHARMACOLOGY OF ACEA-1416 - A POTENT SYSTEMICALLY ACTIVE NMDA RECEPTOR GLYCINE SITE ANTAGONIST
Authors: ILYIN VI WHITTEMORE ER TRAN M SHEN KZ CAI SX KHER SM KEANA JFW WEBER E WOODWARD RM
Citation: Vi. Ilyin et al., PHARMACOLOGY OF ACEA-1416 - A POTENT SYSTEMICALLY ACTIVE NMDA RECEPTOR GLYCINE SITE ANTAGONIST, European journal of pharmacology, 310(2-3), 1996, pp. 107-114
INHIBITION OF MORPHINE-TOLERANCE BY NMDA RECEPTOR ANTAGONISTS IN THE FORMALIN TEST
Authors: LUTFY K SHEN KZ WOODWARD RM WEBER E
Citation: K. Lutfy et al., INHIBITION OF MORPHINE-TOLERANCE BY NMDA RECEPTOR ANTAGONISTS IN THE FORMALIN TEST, Brain research, 731(1-2), 1996, pp. 171-181
IN-VITRO PHARMACOLOGY OF ACEA-1021 AND ACEA-1031 - SYSTEMICALLY ACTIVE QUINOXALINEDIONES WITH HIGH-AFFINITY AND SELECTIVITY FOR N-METHYL-D-ASPARTATE RECEPTOR GLYCINE SITES
Authors: WOODWARD RM HUETTNER JE GUASTELLA J KEANA JFW WEBER E
Citation: Rm. Woodward et al., IN-VITRO PHARMACOLOGY OF ACEA-1021 AND ACEA-1031 - SYSTEMICALLY ACTIVE QUINOXALINEDIONES WITH HIGH-AFFINITY AND SELECTIVITY FOR N-METHYL-D-ASPARTATE RECEPTOR GLYCINE SITES, Molecular pharmacology, 47(3), 1995, pp. 568-581
Risultati: 1-25 | 26-33