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Results: 1-25 | 26-29
Results: 1-25/29
EFFECTS OF SR140333, A SELECTIVE NONPEPTIDE NK1 RECEPTOR ANTAGONIST, ON TRIGEMINO-THALAMIC NOCICEPTIVE PATHWAYS IN THE RAT
Authors: MICHAUD JC ALONSO R GUEUDET C FOURNIER M CALASSI R BRELIERE JC LEFUR G SOUBRIE P
Citation: Jc. Michaud et al., EFFECTS OF SR140333, A SELECTIVE NONPEPTIDE NK1 RECEPTOR ANTAGONIST, ON TRIGEMINO-THALAMIC NOCICEPTIVE PATHWAYS IN THE RAT, Fundamental and clinical pharmacology, 12(1), 1998, pp. 88-94
SR-144528, THE FIRST POTENT AND SELECTIVE ANTAGONIST OF THE CB2 CANNABINOID RECEPTOR
Authors: RINALDICARMONA M BARTH F MILLAN J DEROCQ JM CASELLAS P CONGY C OUSTRIC D SARRAN M BOUABOULA M CALANDRA B PORTIER M SHIRE D BRELIERE JC LEFUR G
Citation: M. Rinaldicarmona et al., SR-144528, THE FIRST POTENT AND SELECTIVE ANTAGONIST OF THE CB2 CANNABINOID RECEPTOR, The Journal of pharmacology and experimental therapeutics, 284(2), 1998, pp. 644-650
BIOCHEMICAL AND PHARMACOLOGICAL ACTIVITIES OF SR-144190, A NEW POTENTNONPEPTIDE TACHYKININ NK2 RECEPTOR ANTAGONIST
Authors: EMONDSALT X ADVENIER C COGNON C CROCI T DAOUI S DUCOUX JP LANDI M NALINE E NELIAT G PONCELET M PROLETTO V VANBROECK D VILAIN P SOUBRIE P LEFUR G MAFFRAND JP BRELIERE JC
Citation: X. Emondsalt et al., BIOCHEMICAL AND PHARMACOLOGICAL ACTIVITIES OF SR-144190, A NEW POTENTNONPEPTIDE TACHYKININ NK2 RECEPTOR ANTAGONIST, Neuropeptides, 31(5), 1997, pp. 449-458
TACHYKININ-INDUCED CONTRACTIONS OF THE GUINEA-PIG ILEUM LONGITUDINAL SMOOTH-MUSCLE - TONIC AND PHASIC MUSCULAR ACTIVITIES
Authors: VILAIN P EMONDSALT X LEFUR G BRELIERE JC
Citation: P. Vilain et al., TACHYKININ-INDUCED CONTRACTIONS OF THE GUINEA-PIG ILEUM LONGITUDINAL SMOOTH-MUSCLE - TONIC AND PHASIC MUSCULAR ACTIVITIES, Canadian journal of physiology and pharmacology, 75(6), 1997, pp. 587-590
PHARMACOLOGICAL CHARACTERIZATION OF SR-142801 - A NEW NONPEPTIDE ANTAGONIST OF THE NEUROKININ NK-3 RECEPTOR
Authors: NGUYENLE XK NGUYEN QT GOBEIL F PHENG LH EMONDSALT X BRELIERE JC REGOLI D
Citation: Xk. Nguyenle et al., PHARMACOLOGICAL CHARACTERIZATION OF SR-142801 - A NEW NONPEPTIDE ANTAGONIST OF THE NEUROKININ NK-3 RECEPTOR, Pharmacology, 52(5), 1996, pp. 283-291
CHARACTERIZATION AND DISTRIBUTION OF BINDING-SITES FOR [H-3] SR 141716A, A SELECTIVE BRAIN (CB1) CANNABINOID RECEPTOR ANTAGONIST, IN RODENTBRAIN
Authors: RINALDICARMONA M PIALOT F CONGY C REDON E BARTH F BACHY A BRELIERE JC SOUBRIE P LEFUR G
Citation: M. Rinaldicarmona et al., CHARACTERIZATION AND DISTRIBUTION OF BINDING-SITES FOR [H-3] SR 141716A, A SELECTIVE BRAIN (CB1) CANNABINOID RECEPTOR ANTAGONIST, IN RODENTBRAIN, Life sciences, 58(15), 1996, pp. 1239-1247
EFFECT OF SUBSTANCE-P ON CYTOKINE PRODUCTION BY HUMAN ASTROCYTIC CELLS AND BLOOD MONONUCLEAR-CELLS - CHARACTERIZATION OF NOVEL TACHYKININ RECEPTOR ANTAGONISTS
Authors: DEROCQ JM SEGUI M BLAZY C EMONDSALT X LEFUR G BRELIERE JC CASELLAS P
Citation: Jm. Derocq et al., EFFECT OF SUBSTANCE-P ON CYTOKINE PRODUCTION BY HUMAN ASTROCYTIC CELLS AND BLOOD MONONUCLEAR-CELLS - CHARACTERIZATION OF NOVEL TACHYKININ RECEPTOR ANTAGONISTS, FEBS letters, 399(3), 1996, pp. 321-325
BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF SR141716A, THE FIRST POTENT AND SELECTIVE BRAIN CANNABINOID RECEPTOR ANTAGONIST
Authors: RINALDICARMONA M BARTH F HEAULME M ALONSO R SHIRE D CONGY C SOUBRIE P BRELIERE JC LEFUR G
Citation: M. Rinaldicarmona et al., BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF SR141716A, THE FIRST POTENT AND SELECTIVE BRAIN CANNABINOID RECEPTOR ANTAGONIST, Life sciences, 56(23-24), 1995, pp. 1941-1947
EFFECTS OF SR-142801, A POTENT NONPEPTIDE TACHYKININ NK3 RECEPTOR ANTAGONIST, ON CARDIOVASCULAR-RESPONSES INDUCED BY SENKTIDE IN CONSCIOUS GUINEA-PIGS
Authors: NISATO D ROCCON A MARCHIONNI D EMONDSALT X BRELIERE JC LEFUR G
Citation: D. Nisato et al., EFFECTS OF SR-142801, A POTENT NONPEPTIDE TACHYKININ NK3 RECEPTOR ANTAGONIST, ON CARDIOVASCULAR-RESPONSES INDUCED BY SENKTIDE IN CONSCIOUS GUINEA-PIGS, British Journal of Pharmacology, 114, 1995, pp. 42-42
DEVELOPMENT OF TETRAZOLE BIOISOSTERES IN ANGIOTENSIN-II ANTAGONISTS
Authors: FERRARI B TAILLADES J PERREAUT P BERNHART C GOUGAT J GUIRAUDOU P CAZAUBON C ROCCON A NISATO D LEFUR G BRELIERE JC
Citation: B. Ferrari et al., DEVELOPMENT OF TETRAZOLE BIOISOSTERES IN ANGIOTENSIN-II ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 45-50
CYCLOPENTANESPIRO-3H-DIHYDRO-PYRIMIDINONES AS ANGIOTENSIN-II AT(1) RECEPTOR ANTAGONISTS
Authors: BERNHART CA HAUDRICOURT FB ASSENS JL GOUGAT J LACOUR C ROCCON A CAZAUBON C BRELIERE JC LEFUR G NISATO D
Citation: Ca. Bernhart et al., CYCLOPENTANESPIRO-3H-DIHYDRO-PYRIMIDINONES AS ANGIOTENSIN-II AT(1) RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 157-162
DIHYDRO-IMIDAZOLONE DERIVATIVES AS ANGIOTENSIN-II RECEPTOR ANTAGONISTS - CHIRAL EFFECT ON THE ACTIVITY
Authors: PERREAUT P CLEMENT J MUNEAUX C MUNEAUX Y CAZAUBON C GOUGAT J GUIRAUDOU P LACOUR C NISATO D LEFUR G BRELIERE JC
Citation: P. Perreaut et al., DIHYDRO-IMIDAZOLONE DERIVATIVES AS ANGIOTENSIN-II RECEPTOR ANTAGONISTS - CHIRAL EFFECT ON THE ACTIVITY, Bioorganic & medicinal chemistry letters, 4(1), 1994, pp. 163-168
ALLOSTERIC MODULATION OF PERIPHERAL SIGMA-BINDING SITES BY A NEW SELECTIVE LIGAND - SR-31747
Authors: PAUL R LAVASTRE S FLOUTARD D FLOUTARD R CANAT X CASELLAS P LEFUR G BRELIERE JC
Citation: R. Paul et al., ALLOSTERIC MODULATION OF PERIPHERAL SIGMA-BINDING SITES BY A NEW SELECTIVE LIGAND - SR-31747, Journal of neuroimmunology, 52(2), 1994, pp. 183-192
IMMUNOPHARMACOLOGICAL PROFILE OF SR-31747 - IN-VITRO AND IN-VIVO STUDIES ON HUMORAL AND CELLULAR-RESPONSES
Authors: CASELLAS P BOURRIE B CANAT X CARAYON P BUISSON I PAUL R BRELIERE JC LEFUR G
Citation: P. Casellas et al., IMMUNOPHARMACOLOGICAL PROFILE OF SR-31747 - IN-VITRO AND IN-VIVO STUDIES ON HUMORAL AND CELLULAR-RESPONSES, Journal of neuroimmunology, 52(2), 1994, pp. 193-203
NEUROPHARMACOLOGICAL CHARACTERIZATION OF SR-140333, A NON PEPTIDE ANTAGONIST OF NK1 RECEPTORS
Authors: JUNG M CALASSI R MARUANI J BARNOUIN MC SOUILHAC J PONCELET M GUEUDET C EMONDSALT X SOUBRIE P BRELIERE JC LEFUR G
Citation: M. Jung et al., NEUROPHARMACOLOGICAL CHARACTERIZATION OF SR-140333, A NON PEPTIDE ANTAGONIST OF NK1 RECEPTORS, Neuropharmacology, 33(2), 1994, pp. 167-179
EVIDENCE FOR A COMMON MOLECULAR-MODE OF ACTION FOR CHEMICALLY DISTINCT NONPEPTIDE ANTAGONISTS AT THE NEUROKININ-1 (SUBSTANCE-P) RECEPTOR
Authors: GETHER U EMONDSALT X BRELIERE JC FUJII T HAGIWARA D PRADIER L GARRET C JOHANSEN TE SCHWARTZ TW
Citation: U. Gether et al., EVIDENCE FOR A COMMON MOLECULAR-MODE OF ACTION FOR CHEMICALLY DISTINCT NONPEPTIDE ANTAGONISTS AT THE NEUROKININ-1 (SUBSTANCE-P) RECEPTOR, Molecular pharmacology, 45(3), 1994, pp. 500-508
SR-142801, THE FIRST POTENT NONPEPTIDE ANTAGONIST OF THE TACHYKININ NK3 RECEPTOR
Authors: EMONDSALT X BICHON D DUCOUX JP HEAULME M MILOUX B PONCELET M PROIETTO V VANBROECK D VILAIN P NELIAT G SOUBRIE P LEFUR G BRELIERE JC
Citation: X. Emondsalt et al., SR-142801, THE FIRST POTENT NONPEPTIDE ANTAGONIST OF THE TACHYKININ NK3 RECEPTOR, Life sciences, 56(1), 1994, pp. 161200027-161200032
IDENTIFICATION OF BINDING-SITES FOR SR-46349B, A 5-HYDROXYTRYPTAMINE(2) RECEPTOR ANTAGONIST, IN RODENT BRAIN
Authors: RINALDICARMONA M CONGY C POINTEAU P VIDAL H BRELIERE JC LEFUR G
Citation: M. Rinaldicarmona et al., IDENTIFICATION OF BINDING-SITES FOR SR-46349B, A 5-HYDROXYTRYPTAMINE(2) RECEPTOR ANTAGONIST, IN RODENT BRAIN, Life sciences, 54(2), 1994, pp. 119-127
SR141716A, A POTENT AND SELECTIVE ANTAGONIST OF THE BRAIN CANNABINOIDRECEPTOR
Authors: RINALDICARMONA M BARTH F HEAULME M SHIRE D CALANDRA B CONGY C MARTINEZ S MARUANI J NELIAT G CAPUT D FERRARA P SOUBRIE P BRELIERE JC LEFUR G
Citation: M. Rinaldicarmona et al., SR141716A, A POTENT AND SELECTIVE ANTAGONIST OF THE BRAIN CANNABINOIDRECEPTOR, FEBS letters, 350(2-3), 1994, pp. 240-244
PHARMACOLOGICAL PROFILE AND CHEMICAL SYNTHESIS OF SR-48968, A NONPEPTIDE ANTAGONIST OF THE NEUROKININ-A NK(2) RECEPTOR
Authors: EDMONDSALT X PROIETTO V VANBROECK D VILAIN P ADVENIER C NELIAT G LEFUR G BRELIERE JC
Citation: X. Edmondsalt et al., PHARMACOLOGICAL PROFILE AND CHEMICAL SYNTHESIS OF SR-48968, A NONPEPTIDE ANTAGONIST OF THE NEUROKININ-A NK(2) RECEPTOR, Bioorganic & medicinal chemistry letters, 3(5), 1993, pp. 925-930
UP-REGULATION OF 5-HT(2) RECEPTORS IN THE RAT-BRAIN BY REPEATED ADMINISTRATION OF SR-46349B, A SELECTIVE 5-HT(2) RECEPTOR ANTAGONIST
Authors: RINALDICARMONA M BOUABOULA M CONGY C OURYDONAT F SIMIAND J SHIRE D CASELLAS P SOUBRIE P BRELIERE JC LEFUR G
Citation: M. Rinaldicarmona et al., UP-REGULATION OF 5-HT(2) RECEPTORS IN THE RAT-BRAIN BY REPEATED ADMINISTRATION OF SR-46349B, A SELECTIVE 5-HT(2) RECEPTOR ANTAGONIST, European journal of pharmacology. Molecular pharmacology section, 246(1), 1993, pp. 73-80
THE STAMINA OF DRUGS
Authors: MAFFRAND JP BRELIERE JC
Citation: Jp. Maffrand et Jc. Breliere, THE STAMINA OF DRUGS, New scientist, 138(1870), 1993, pp. 12-13
SR-48968, A NEUROKININ-A (NK2) RECEPTOR ANTAGONIST
Authors: EMONDSALT X ADVENIER C CROCI T MANARA L NELIAT G PONCELET M PROIETTO V SANTUCCI V SOUBRIE P VANBROECK D VILAIN P LEFUR G BRELIERE JC
Citation: X. Emondsalt et al., SR-48968, A NEUROKININ-A (NK2) RECEPTOR ANTAGONIST, Regulatory peptides, 46(1-2), 1993, pp. 31-36
NEUROPHARMACOLOGICAL PROFILE OF A NOVEL AND SELECTIVE LIGAND OF THE SIGMA SITE - SR 31742A
Authors: PONCELET M SANTUCCI V PAUL R GUEUDET C LAVASTRE S GUITARD J STEINBERG R TERRANOVA JP BRELIERE JC SOUBRIE P LEFUR G
Citation: M. Poncelet et al., NEUROPHARMACOLOGICAL PROFILE OF A NOVEL AND SELECTIVE LIGAND OF THE SIGMA SITE - SR 31742A, Neuropharmacology, 32(6), 1993, pp. 605-615
2 NONPEPTIDE TACHYKININ ANTAGONISTS ACT THROUGH EPITOPES ON CORRESPONDING SEGMENTS OF THE NK1 AND NK2 RECEPTORS
Authors: GETHER U YOKOTA Y EMONDSALT X BRELIERE JC LOWE JA SNIDER RM NAKANISHI S SCHWARTZ TW
Citation: U. Gether et al., 2 NONPEPTIDE TACHYKININ ANTAGONISTS ACT THROUGH EPITOPES ON CORRESPONDING SEGMENTS OF THE NK1 AND NK2 RECEPTORS, Proceedings of the National Academy of Sciences of the United Statesof America, 90(13), 1993, pp. 6194-6198
Risultati: 1-25 | 26-29