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Results: 1-25/69
Authors:
Boger, DL
Tse, WC
Citation: Dl. Boger et Wc. Tse, Thiazole orange as the fluorescent intercalator in a high resolution FID assay for determining DNA binding affinity and sequence selectivity of smallmolecules, BIO MED CH, 9(9), 2001, pp. 2511-2518
Authors:
Boger, DL
Goldberg, J
Citation: Dl. Boger et J. Goldberg, Cytokine receptor dimerization and activation: Prospects for small molecule agonists, BIO MED CH, 9(3), 2001, pp. 557-562
Authors:
Boger, DL
Stauffer, F
Hedrick, MP
Citation: Dl. Boger et al., Substituent effects within the DNA binding subunit of CBI analogues of theduocarmycins and CC-1065, BIOORG MED, 11(15), 2001, pp. 2021-2024
Authors:
Boger, DL
Miyauchi, H
Hedrick, MP
Citation: Dl. Boger et al., alpha-Keto heterocycle inhibitors of fatty acid amide hydrolase: Carbonyl group modification and alpha-substitution, BIOORG MED, 11(12), 2001, pp. 1517-1520
Authors:
Boger, DL
Citation: Dl. Boger, Symposium-in-Print - Recent advances in bioorganic and medicinal chemistry- Preface, BIOORG MED, 11(12), 2001, pp. IX-IX
Authors:
Boger, DL
Citation: Dl. Boger, Vancomycin, teicoplanin, and ramoplanin: Synthetic and mechanistic studies, MED RES REV, 21(5), 2001, pp. 356-381
Authors:
Mori, Y
McAtee, JJ
Rogel, O
Boger, DL
Citation: Y. Mori et al., Alternative synthesis and thermal atropisomerism of a fully functionalizedDEFG ring system of teicoplanin, TETRAHEDR L, 42(35), 2001, pp. 6061-6064
Authors:
Silletti, S
Kessler, T
Goldberg, J
Boger, DL
Cheresh, DA
Citation: S. Silletti et al., Disruption of matrix metalloproteinase 2 binding to integrin alpha(v)beta(3) by an organic molecule inhibits angiogenesis and tumor growth in vivo, P NAS US, 98(1), 2001, pp. 119-124
Authors:
Fedorova, I
Hashimoto, A
Fecik, RA
Hedrick, MP
Hanus, LO
Boger, DL
Rice, KC
Basile, AS
Citation: I. Fedorova et al., Behavioral evidence for the interaction of oleamide with multiple neurotransmitter systems, J PHARM EXP, 299(1), 2001, pp. 332-342
Authors:
Boger, DL
Hughes, TV
Hedrick, MP
Citation: Dl. Boger et al., Synthesis, chemical properties, and biological evaluation of CC-1065 and duocarmycin analogues incorporating the 5-methoxycarbonyl-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one alkylation subunit, J ORG CHEM, 66(7), 2001, pp. 2207-2216
Authors:
Boger, DL
Schmitt, HW
Fink, BE
Hedrick, MP
Citation: Dl. Boger et al., Parallel synthesis and evaluation of 132 (+)-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one (CBI) analogues of CC-1065 and the duocarmycins defining the contribution of the DNA-binding domain, J ORG CHEM, 66(20), 2001, pp. 6654-6661
Synthesis and evaluation of a series of C3-substituted CBI analogues of CC-1065 and the duocarmycins
Authors:
Boger, DL
Brunette, SR
Garbaccio, RM
Citation: Dl. Boger et al., Synthesis and evaluation of a series of C3-substituted CBI analogues of CC-1065 and the duocarmycins, J ORG CHEM, 66(15), 2001, pp. 5163-5173
Authors:
Greasley, SE
Marsilje, TH
Cai, H
Baker, S
Benkovic, SJ
Boger, DL
Wilson, IA
Citation: Se. Greasley et al., Unexpected formation of an epoxide-derived multisubstrate adduct inhibitoron the active site of GAR transformylase, BIOCHEM, 40(45), 2001, pp. 13538-13547
Authors:
Boger, DL
Kim, SH
Mori, Y
Weng, JH
Rogel, O
Castle, SL
McAtee, JJ
Citation: Dl. Boger et al., First and second generation total synthesis of the teicoplanin aglycon, J AM CHEM S, 123(9), 2001, pp. 1862-1871
Authors:
Boger, DL
Goldberg, J
Silletti, S
Kessler, T
Cheresh, DA
Citation: Dl. Boger et al., Identification of a novel class of small-molecule antiangiogenic agents through the screening of combinatorial libraries which function by inhibitingthe binding and localization of proteinase MMP2 to integrin alpha(v)beta(3), J AM CHEM S, 123(7), 2001, pp. 1280-1288
Authors:
Boger, DL
Ichikawa, S
Tse, WC
Hedrick, MP
Jin, Q
Citation: Dl. Boger et al., Total syntheses of thiocoraline and BE-22179 and assessment of their DNA binding and biological properties, J AM CHEM S, 123(4), 2001, pp. 561-568
Authors:
Ellis, DA
Wolkenberg, SE
Boger, DL
Citation: Da. Ellis et al., Metal cation complexation and activation of reversed CPyI analogues of CC-1065 and duocarmycin SA: Partitioning the effects of binding and catalysis, J AM CHEM S, 123(38), 2001, pp. 9299-9306
Authors:
Boger, DL
Hong, JY
Citation: Dl. Boger et Jy. Hong, Asymmetric total synthesis of ent-(-)-roseophilin: Assignment of absolute configuration, J AM CHEM S, 123(35), 2001, pp. 8515-8519
Authors:
Boger, DL
Fink, BE
Brunette, SR
Tse, WC
Hedrick, MP
Citation: Dl. Boger et al., A simple, high-resolution method for establishing DNA binding affinity andsequence selectivity, J AM CHEM S, 123(25), 2001, pp. 5878-5891
Authors:
Boger, DL
Ichikawa, S
Zhong, W
Citation: Dl. Boger et al., Total synthesis of fostriecin (CI-920), J AM CHEM S, 123(18), 2001, pp. 4161-4167
Authors:
Boger, DL
Dechantsreiter, MA
Ishii, T
Fink, BE
Hedrick, MP
Citation: Dl. Boger et al., Assessment of solution-phase positional scanning libraries based on distamycin A for the discovery of new DNA binding agents, BIO MED CH, 8(8), 2000, pp. 2049-2057
Authors:
Boger, DL
Labroli, MA
Marsilje, TH
Jin, Q
Hedrick, MP
Baker, SJ
Shim, JH
Benkovic, SJ
Citation: Dl. Boger et al., Conformationally restricted analogues designed for selective inhibition ofGAR Tfase versus thymidylate synthase or dihydrofolate reductase, BIO MED CH, 8(5), 2000, pp. 1075-1086
Authors:
Boger, DL
Searcey, M
Tse, WC
Jin, Q
Citation: Dl. Boger et al., Bifunctional alkylating agents derived from duocarmycin SA: Potent antitumor activity with altered sequence selectivity, BIOORG MED, 10(5), 2000, pp. 495-498
Authors:
Boger, DL
Fecik, RA
Patterson, JE
Miyauchi, H
Patricelli, MP
Cravatt, BF
Citation: Dl. Boger et al., Fatty acid amide hydrolase substrate specificity, BIOORG MED, 10(23), 2000, pp. 2613-2616
Authors:
Boger, DL
Chen, Y
Foster, CA
Citation: Dl. Boger et al., Synthesis and evaluation of aza HUN-7293, BIOORG MED, 10(15), 2000, pp. 1741-1744