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Results: 1-25 | 26-47 |
Results: 26-47/47
Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes
Authors: Vianello, P Albinati, A Pinna, GA Lavecchia, A Marinelli, L Borea, PA Gessi, S Fadda, P Tronci, S Cignarella, G
Citation: P. Vianello et al., Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes, J MED CHEM, 43(11), 2000, pp. 2115-2123
Synthesis, modelling, and mu-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes
Authors: Pinna, GA Murineddu, G Curzu, MM Villa, S Vianello, P Borea, PA Gessi, S Toma, L Colombo, D Cignarella, G
Citation: Ga. Pinna et al., Synthesis, modelling, and mu-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes, FARMACO, 55(8), 2000, pp. 553-562
Dose and time effects of caffeine intake on human platelet adenosine A(2A)receptors - Functional and biochemical aspects
Authors: Varani, K Portaluppi, F Gessi, S Merighi, S Ongini, E Belardinelli, L Borea, PA
Citation: K. Varani et al., Dose and time effects of caffeine intake on human platelet adenosine A(2A)receptors - Functional and biochemical aspects, CIRCULATION, 102(3), 2000, pp. 285-289
Thermodynamically distinct high and low affinity states of the A(1) adenosine receptor induced by G protein coupling and guanine nucleotide ligation states of G proteins
Authors: Lorenzen, A Guerra, L Campi, F Lang, H Schwabe, U Borea, PA
Citation: A. Lorenzen et al., Thermodynamically distinct high and low affinity states of the A(1) adenosine receptor induced by G protein coupling and guanine nucleotide ligation states of G proteins, BR J PHARM, 130(3), 2000, pp. 595-604
A(2A) adenosine receptors in human peripheral blood cells
Authors: Gessi, S Varani, K Merighi, S Ongini, E Borea, PA
Citation: S. Gessi et al., A(2A) adenosine receptors in human peripheral blood cells, BR J PHARM, 129(1), 2000, pp. 2-11
Can thermodynamic measurements of receptor binding yield information on drug affinity and efficacy?
Authors: Borea, PA Dalpiaz, A Varani, K Gilli, P Gilli, G
Citation: Pa. Borea et al., Can thermodynamic measurements of receptor binding yield information on drug affinity and efficacy?, BIOCH PHARM, 60(11), 2000, pp. 1549-1556
Synthesis and binding of 3-aminopyridine derivatives at central nicotinic receptors
Authors: Balboni, G Marastoni, M Merighi, S Borea, PA Tomatis, R
Citation: G. Balboni et al., Synthesis and binding of 3-aminopyridine derivatives at central nicotinic receptors, ARZNEI-FOR, 50(6), 2000, pp. 507-511
Hybridized and isosteric analogues of N-1-acetyl-N-4-dimethy-piperazinium iodide (ADMP) and N-1-phenyl-N-4-dimethy-piperazinium iodide (DMPP) with central nicotinic action
Authors: Manetti, D Bartolini, A Borea, PA Bellucci, C Dei, S Ghelardini, C Gualtieri, F Romanelli, MN Scapecchi, S Teodori, E Varani, K
Citation: D. Manetti et al., Hybridized and isosteric analogues of N-1-acetyl-N-4-dimethy-piperazinium iodide (ADMP) and N-1-phenyl-N-4-dimethy-piperazinium iodide (DMPP) with central nicotinic action, BIO MED CH, 7(3), 1999, pp. 457-465
Thermodynamic in vitro studies as a method to investigate the pharmacodynamic behavior of adenosine A(1) receptor ligands
Authors: Dalpiaz, A Scatturin, A Pavan, B Varani, K IJzerman, AP Borea, PA
Citation: A. Dalpiaz et al., Thermodynamic in vitro studies as a method to investigate the pharmacodynamic behavior of adenosine A(1) receptor ligands, PHARM RES, 16(7), 1999, pp. 1054-1058
Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension
Authors: Varani, K Gessi, S Caiazza, A Rastelli, G Portaluppi, F Borea, PA
Citation: K. Varani et al., Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension, BR J CL PH, 47(2), 1999, pp. 167-172
Changes in hippocampal and cortical B-1 bradykinin receptor biological activity in two experimental models of epilepsy
Authors: Bregola, G Varani, K Gessi, S Beani, L Bianchi, C Borea, PA Regoli, D Simonato, M
Citation: G. Bregola et al., Changes in hippocampal and cortical B-1 bradykinin receptor biological activity in two experimental models of epilepsy, NEUROSCIENC, 92(3), 1999, pp. 1043-1049
Comparative molecular field analysis (CoMFA) of a series of selective adenosine receptor A(2A) antagonists
Authors: Baraldi, PG Borea, PA Bergonzoni, M Cacciari, B Ongini, E Recanatini, M Spalluto, G
Citation: Pg. Baraldi et al., Comparative molecular field analysis (CoMFA) of a series of selective adenosine receptor A(2A) antagonists, DRUG DEV R, 46(2), 1999, pp. 126-133
4-(4-fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors
Authors: Claudi, F Scoccia, L Giorgioni, G Accorroni, B Marucci, G Gessi, S Siniscalchi, A Borea, PA
Citation: F. Claudi et al., 4-(4-fluorobenzoyl)-1-[2-(4-iodo-2,5-dimethoxyphenyl)ethyl]piperidine and its derivatives: synthesis and affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors, EUR J MED C, 34(10), 1999, pp. 843-852
Early changes in adenosine A(1) receptors in cerebral cortex slices submitted to in vitro ischemia
Authors: Siniscalchi, A Rodi, D Gessi, S Campi, F Borea, PA
Citation: A. Siniscalchi et al., Early changes in adenosine A(1) receptors in cerebral cortex slices submitted to in vitro ischemia, NEUROCHEM I, 34(6), 1999, pp. 517-522
Pharmacology of [Tyr(1)]nociceptin analogs: receptor binding and bioassay studies
Authors: Varani, K Rizzi, A Calo, G Bigoni, R Toth, G Guerrini, R Gessi, S Salvadori, S Borea, PA Regoli, D
Citation: K. Varani et al., Pharmacology of [Tyr(1)]nociceptin analogs: receptor binding and bioassay studies, N-S ARCH PH, 360(3), 1999, pp. 270-277
Temperature dependence and GABA modulation of beta-carboline binding to rat cerebellum benzodiazepine receptors
Authors: Gessi, S Dalpiaz, A Varani, K Borea, PA
Citation: S. Gessi et al., Temperature dependence and GABA modulation of beta-carboline binding to rat cerebellum benzodiazepine receptors, LIFE SCI, 64(16), 1999, pp. PL185-PL192
alpha(2)-adrenergic agonist modulation of [S-35]GTP gamma S binding to guanine-nucleotide-binding-proteins in human platelet membranes
Authors: Gessi, S Campi, F Varani, K Borea, PA
Citation: S. Gessi et al., alpha(2)-adrenergic agonist modulation of [S-35]GTP gamma S binding to guanine-nucleotide-binding-proteins in human platelet membranes, LIFE SCI, 64(16), 1999, pp. 1403-1413
Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]-pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Klotz, KN Leung, E Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]-pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists, J MED CHEM, 42(22), 1999, pp. 4473-4478
Caffeine alters A(2A) adenosine receptors and their function in human platelets
Authors: Varani, K Portaluppi, F Merighi, S Ongini, E Belardinelli, L Borea, PA
Citation: K. Varani et al., Caffeine alters A(2A) adenosine receptors and their function in human platelets, CIRCULATION, 99(19), 1999, pp. 2499-2502
Sixth International Symposium on Adenosine and Adenine Nucleotides: New frontiers in the third millennium
Authors: Borea, PA Baraldi, PG
Citation: Pa. Borea et Pg. Baraldi, Sixth International Symposium on Adenosine and Adenine Nucleotides: New frontiers in the third millennium, DRUG DEV R, 45(3-4), 1998, pp. 85-85
Adenosine A(2a) receptors of human circulating blood elements
Authors: Varani, K Gessi, S Merighi, S Ongini, E Borea, PA
Citation: K. Varani et al., Adenosine A(2a) receptors of human circulating blood elements, DRUG DEV R, 45(3-4), 1998, pp. 253-260
Nociceptin receptor binding in mouse forebrain membranes: thermodynamic characteristics and structure activity relationships
Authors: Varani, K Calo, G Rizzi, A Merighi, S Toth, G Guerrini, R Salvadori, S Borea, PA Regoli, D
Citation: K. Varani et al., Nociceptin receptor binding in mouse forebrain membranes: thermodynamic characteristics and structure activity relationships, BR J PHARM, 125(7), 1998, pp. 1485-1490
Risultati: 1-25 | 26-47 |