Authors:
UNANGST PC
CAPIRIS T
CONNOR DT
DOUBLEDAY R
HEFFNER TG
MACKENZIE RG
MILLER SR
PUGSLEY TA
WISE LD
Citation: Pc. Unangst et al., (ARYLOXY)ALKYLAMINES AS SELECTIVE HUMAN DOPAMINE D-4 RECEPTOR ANTAGONISTS - POTENTIAL ANTIPSYCHOTIC AGENTS, Journal of medicinal chemistry, 40(25), 1997, pp. 4026-4029
Authors:
UNANGST PC
CAPIRIS T
CONNOR DT
HEFFNER TG
MACKENZIE RG
MILLER SR
PUGSLEY TA
WISE LD
Citation: Pc. Unangst et al., CHROMENO[3,4-C]PYRIDIN-5-ONES - SELECTIVE HUMAN DOPAMINE D-4 RECEPTORANTAGONISTS AS POTENTIAL ANTIPSYCHOTIC AGENTS, Journal of medicinal chemistry, 40(17), 1997, pp. 2688-2693
Authors:
FUJIMORI T
CONNOR DT
CETENKO WA
MARLETTA MA
HUPE DJ
DYER RD
Citation: T. Fujimori et al., A NOVEL ANTIINFLAMMATORY COMPOUND EXTENDS THE LAG PHASE OF PROSTAGLANDIN-H SYNTHASE-2 (PGHS-2) KINETICS, The FASEB journal, 10(6), 1996, pp. 1495-1495
Authors:
KHATANA SS
BOSCHELLI DH
KRAMER JB
CONNOR DT
BARTH H
STOSS P
Citation: Ss. Khatana et al., PREPARATION OF BENZOTHIENO[2,3-F]-1,4-OXAZEPIN-5(2H)-ONES AND BENZOTHIENO[2,3-F]-1,4-THIAZEPIN-5(2H)-ONES AND OF BENZOTHIENO[3,2-E]-1,4-DIAZEPIN-5-ONES, Journal of organic chemistry, 61(17), 1996, pp. 6060-6062
Citation: Pc. Unangst et al., SYNTHESIS OF NOVEL 5-HYDROXY-3-ALKOXY-INDOLE-2-CARBOXAMIDES AND 5-HYDROXY-3-ALKYLTHIO-INDOLE-2-CARBOXAMIDES, Journal of heterocyclic chemistry, 33(6), 1996, pp. 1627-1630
Citation: Pc. Unangst et al., SYNTHESIS OF NOVEL 3-ALKOXYTHIOINDOLE AND 3-ALKYLTHIOINDOLE AND -BENZOFURAN-2-CARBOXAMIDES, Journal of heterocyclic chemistry, 33(6), 1996, pp. 2025-2030
Authors:
BOSCHELLI DH
KRAMER JB
KHATANA SS
SORENSON RJ
CONNOR DT
FERIN MA
WRIGHT CD
LESCH ME
IMRE K
OKONKWO GC
SCHRIER DJ
CONROY MC
FERGUSON E
WOELLE J
SAXENA U
Citation: Dh. Boschelli et al., INHIBITION OF E-SELECTIN-MEDIATED, ICAM-1-MEDIATED, AND VCAM-1-MEDIATED CELL-ADHESION BY BENZO[B]THIOPHENE-CARBOXAMIDES, BENZOFURAN-CARBOXAMIDES, INDOLE-, AND NAPHTHALENE-2-CARBOXAMIDES - IDENTIFICATION OF PD-144795 AS AN ANTIINFLAMMATORY AGENT, Journal of medicinal chemistry, 38(22), 1995, pp. 4597-4614
Authors:
UNANGST PC
CONNOR DT
KOSTLAN CR
SHRUM GP
MILLER SR
KANTER G
Citation: Pc. Unangst et al., SYNTHESIS OF PYRIMIDINE ANALOGS OF 2,6-DI-TERT-BUTYLPHENOL ANTIINFLAMMATORY AGENTS, Journal of heterocyclic chemistry, 32(4), 1995, pp. 1197-1200
Authors:
SCHRIER DJ
BARAGI VM
CONNOR DT
DYER RD
JORDAN JH
IMRE KM
LESCH ME
MULLICAN MD
OKONKWO GCN
CONROY MC
Citation: Dj. Schrier et al., THE PHARMACOLOGICAL EFFECTS OF )-4-HYDROXYPHENYL]-1,3,4-THIADIAZOLE-2(3H)-THIONE, CHOLINE SALT (CI-986), A NOVEL INHIBITOR OF ARACHIDONIC-ACID METABOLISM IN MODELS OF INFLAMMATION, ANALGESIA AND GASTRIC IRRITATION, Prostaglandins, 47(1), 1994, pp. 17-30
Authors:
BOSCHELLI DH
KRAMER JB
CONNOR DT
LESCH ME
SCHRIER DJ
FERIN MA
WRIGHT CD
Citation: Dh. Boschelli et al., 3-ALKOXYBENZO[B]THIOPHENE-2-CARBOXAMIDES AS INHIBITORS OF NEUTROPHIL-ENDOTHELIAL CELL-ADHESION, Journal of medicinal chemistry, 37(6), 1994, pp. 717-718
Authors:
UNANGST PC
CONNOR DT
CETENKO WA
SORENSON RJ
KOSTLAN CR
SIRCAR JC
WRIGHT CD
SCHRIER DJ
DYER RD
Citation: Pc. Unangst et al., SYNTHESIS AND BIOLOGICAL EVALUATION OF DIMETHYLETHYL)-4-HYDROXYPHENYL]METHYLENE]OXAZOLES, -THIAZOLES, AND -IMIDAZOLES - NOVEL DUAL 5-LIPOXYGENASE AND CYCLOOXYGENASE INHIBITORS WITH ANTIINFLAMMATORY ACTIVITY, Journal of medicinal chemistry, 37(2), 1994, pp. 322-328
Citation: Jb. Kramer et al., SYNTHESIS OF 2,6-DI-TERT-BUTYLPHENOLS LINKED TO 1,3,4-OXADIAZOLES AND1,3,4-THIADIAZOLES, Journal of heterocyclic chemistry, 31(6), 1994, pp. 1439-1443
Authors:
UNANGST PC
CONNOR DT
CETENKO WA
SORENSON RJ
SIRCAR JC
WRIGHT CD
SCHRIER DJ
DYER RD
Citation: Pc. Unangst et al., OXAZOLE, THIAZOLE, AND IMIDAZOLE DERIVATIVES OF 2,6-DI-TERT-BUTYLPHENOL AS DUAL 5-LIPOXYGENASE AND CYCLOOXYGENASE INHIBITORS, Bioorganic & medicinal chemistry letters, 3(8), 1993, pp. 1729-1734
Authors:
KRAMER JB
BOSCHELLI DH
CONNOR DT
KOSTLAN CR
KUIPERS PJ
KENNEDY JA
WRIGHT CD
BORNEMEIER DA
DYER RD
Citation: Jb. Kramer et al., CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITORY ACTIVITY OF 2,6 DI-T-BUTYLPHENOLS LINKED BY A SULFUR ATOM TO 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES, Bioorganic & medicinal chemistry letters, 3(12), 1993, pp. 2827-2830
Authors:
MULLICAN MD
WILSON MW
CONNOR DT
KOSTLAN CR
SCHRIER DJ
DYER RD
Citation: Md. Mullican et al., DESIGN OF DI-TERT-BUTYL-4-HYDROXYPHENYL)-1,3,4-THIADIAZOLES, 1,3,4-OXADIAZOLES, AND 1,2,4-TRIAZOLES AS ORALLY-ACTIVE, NONULCEROGENIC ANTIINFLAMMATORY AGENTS, Journal of medicinal chemistry, 36(8), 1993, pp. 1090-1099
Authors:
BOSCHELLI DH
CONNOR DT
BORNEMEIER DA
DYER RD
KENNEDY JA
KUIPERS PJ
OKONKWO GC
SCHRIER DJ
WRIGHT CD
Citation: Dh. Boschelli et al., 1,3,4-OXADIAZOLE, 1,3,4-THIADIAZOLE, AND 1,2,4-TRIAZOLE ANALOGS OF THE FENAMATES - IN-VITRO INHIBITION OF CYCLOOXYGENASE AND 5-LIPOXYGENASEACTIVITIES, Journal of medicinal chemistry, 36(13), 1993, pp. 1802-1810
Citation: Pc. Unangst et al., PREPARATION OF NOVEL 1,2,4-THIADIAZOLES BY CYCLIZATION WITH 4-METHYLBENZENESULFONYL CYANIDE (TOSYL CYANIDE) [1], Journal of heterocyclic chemistry, 30(2), 1993, pp. 357-359