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DESIGN AND SYNTHESIS OF IMIDAZOLINE DERIVATIVES ACTIVE ON GLUCOSE-HOMEOSTASIS IN A RAT MODEL OF TYPE-II DIABETES .1. SYNTHESIS AND BIOLOGICAL-ACTIVITIES OF L)-2-(4',5'-DIHYDRO-1'H-IMIDAZOL-2'-YL)PIPERAZINES
Authors: RONDU F LEBIHAN G WANG X LAMOURI A TOUBOUL E DIVE G BELLAHSENE T PFEIFFER B RENARD P GUARDIOLALEMAITRE B MANECHEZ D PENICAUD L KTORZA A GODFROID JJ
Citation: F. Rondu et al., DESIGN AND SYNTHESIS OF IMIDAZOLINE DERIVATIVES ACTIVE ON GLUCOSE-HOMEOSTASIS IN A RAT MODEL OF TYPE-II DIABETES .1. SYNTHESIS AND BIOLOGICAL-ACTIVITIES OF L)-2-(4',5'-DIHYDRO-1'H-IMIDAZOL-2'-YL)PIPERAZINES, Journal of medicinal chemistry, 40(23), 1997, pp. 3793-3803
NOVEL AND SELECTIVE PARTIAL AGONISTS OF 5-HT3 RECEPTORS .2. SYNTHESISAND BIOLOGICAL EVALUATION OF PIPERAZINOPYRIDOPYRROLOPYRAZINES, PIPERAZINOPYRROLOQUINOXALINES, AND PIPERAZINOPYRIDOPYRROLOQUINOXALINES
Authors: PRUNIER H RAULT S LANCELOT JC ROBBA M RENARD P DELAGRANGE P PFEIFFER B CAIGNARD DH MISSLIN R GUARDIOLALEMAITRE B HAMON M
Citation: H. Prunier et al., NOVEL AND SELECTIVE PARTIAL AGONISTS OF 5-HT3 RECEPTORS .2. SYNTHESISAND BIOLOGICAL EVALUATION OF PIPERAZINOPYRIDOPYRROLOPYRAZINES, PIPERAZINOPYRROLOQUINOXALINES, AND PIPERAZINOPYRIDOPYRROLOQUINOXALINES, Journal of medicinal chemistry, 40(12), 1997, pp. 1808-1819
IDENTIFICATION OF MEL(1A) MELATONIN RECEPTORS IN THE HUMAN EMBRYONIC KIDNEY-CELL-LINE-HEK293 - EVIDENCE OF G-PROTEIN-COUPLED MELATONIN RECEPTORS WHICH DO NOT MEDIATE THE INHIBITION OF STIMULATED CYCLIC-AMP LEVELS
Authors: CONWAY S DREW JE CANNING SJ BARRETT P JOCKERS R STROSBERG AD GUARDIOLALEMAITRE B DELAGRANGE P MORGAN PJ
Citation: S. Conway et al., IDENTIFICATION OF MEL(1A) MELATONIN RECEPTORS IN THE HUMAN EMBRYONIC KIDNEY-CELL-LINE-HEK293 - EVIDENCE OF G-PROTEIN-COUPLED MELATONIN RECEPTORS WHICH DO NOT MEDIATE THE INHIBITION OF STIMULATED CYCLIC-AMP LEVELS, FEBS letters, 407(1), 1997, pp. 121-126
CHARACTERIZATION OF A MELATONIN BINDING-SITE IN SIBERIAN HAMSTER BROWN ADIPOSE-TISSUE
Authors: LEGOUIC S ATGIE C VIGUERIEBASCANDS N HANOUN N LARROUY D AMBID L RAIMBAULT S RICQUIER D DELAGRANGE P GUARDIOLALEMAITRE B PENICAUD L CASTEILLA L
Citation: S. Legouic et al., CHARACTERIZATION OF A MELATONIN BINDING-SITE IN SIBERIAN HAMSTER BROWN ADIPOSE-TISSUE, European journal of pharmacology, 339(2-3), 1997, pp. 271-278
DIRECT STIMULATION OF INSULIN RELEASE FROM THE MIN6 BETA-CELL LINE BYA NEW IMIDAZOLINE COMPOUND, S-21663, VIA AN ORIGINAL SITE
Authors: LEBRIGAND L VIRSOLVY A PEYROLLIER K MANECHEZ D GODFROID JJ GUARDIOLALEMAITRE B BATAILLE D
Citation: L. Lebrigand et al., DIRECT STIMULATION OF INSULIN RELEASE FROM THE MIN6 BETA-CELL LINE BYA NEW IMIDAZOLINE COMPOUND, S-21663, VIA AN ORIGINAL SITE, Diabetologia, 40, 1997, pp. 403-403
POTENT ANTIHYPERGLYCEMIC EFFECT OF AN IMIDAZOLINE DERIVATIVE S-22068 IN A RAT MODEL OF TYPE-II DIABETES
Authors: PELE A WANG X RONDU F ILLIC C HELLARY C LAMOURY A TOUBOUL E DOKHAN R MARC S PFEIFFER B MANECHEZ D RENARD P GUARDIOLALEMAITRE B GODFROID JJ PENICAUD L KTORZA A
Citation: A. Pele et al., POTENT ANTIHYPERGLYCEMIC EFFECT OF AN IMIDAZOLINE DERIVATIVE S-22068 IN A RAT MODEL OF TYPE-II DIABETES, Diabetologia, 40, 1997, pp. 1461-1461
STUDIES ON THE VASOCONSTRICTOR ACTION OF MELATONIN AND PUTATIVE MELATONIN RECEPTOR LIGANDS IN THE TAIL ARTERY OF JUVENILE WISTAR RATS
Authors: TING KN DUNN WR DAVIES DJ SUGDEN D DELAGRANGE F GUARDIOLALEMAITRE B SCALBERT E WILSON VG
Citation: Kn. Ting et al., STUDIES ON THE VASOCONSTRICTOR ACTION OF MELATONIN AND PUTATIVE MELATONIN RECEPTOR LIGANDS IN THE TAIL ARTERY OF JUVENILE WISTAR RATS, British Journal of Pharmacology, 122(7), 1997, pp. 1299-1306
STIMULATION OF INSULIN RELEASE FROM THE MIN6 CELL-LINE BY A NEW IMIDAZOLINE COMPOUND, S-21663 - EVIDENCE FOR THE EXISTENCE OF A NOVEL IMIDAZOLINE SITE IN BETA-CELLS
Authors: LEBRIGAND L VIRSOLVY A PEYROLLIER K MANECHEZ D GODFROID JJ GUARDIOLALEMAITRE B BATAILLE D
Citation: L. Lebrigand et al., STIMULATION OF INSULIN RELEASE FROM THE MIN6 CELL-LINE BY A NEW IMIDAZOLINE COMPOUND, S-21663 - EVIDENCE FOR THE EXISTENCE OF A NOVEL IMIDAZOLINE SITE IN BETA-CELLS, British Journal of Pharmacology, 122(4), 1997, pp. 786-791
THE ROLES SF VALINE-208 AND HISTIDINE-211 IN LIGAND-BINDING AND RECEPTOR FUNCTION OF THE OVINE MEL(1A-BETA) MELATONIN RECEPTOR
Authors: CONWAY S CANNING SJ BARRETT P GUARDIOLALEMAITRE B DELAGRANGE P MORGAN PJ
Citation: S. Conway et al., THE ROLES SF VALINE-208 AND HISTIDINE-211 IN LIGAND-BINDING AND RECEPTOR FUNCTION OF THE OVINE MEL(1A-BETA) MELATONIN RECEPTOR, Biochemical and biophysical research communications, 239(2), 1997, pp. 418-423
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CONFORMATIONALLY RESTRICTED TRICYCLIC ANALOGS OF THE HORMONE MELATONIN
Authors: LECLERC V DEPREUX P LESIEUR D CAIGNARD DH RENARD P DELAGRANGE P GUARDIOLALEMAITRE B MORGAN P
Citation: V. Leclerc et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CONFORMATIONALLY RESTRICTED TRICYCLIC ANALOGS OF THE HORMONE MELATONIN, Bioorganic & medicinal chemistry letters, 6(10), 1996, pp. 1071-1076
EFFECTS OF BOTH A MELATONIN AGONIST AND ANTAGONIST ON SEASONAL-CHANGES IN BODY-MASS AND ENERGY-INTAKE IN THE GARDEN DORMOUSE
Authors: LEGOUIC S DELAGRANGE P ATGIE C NIBBELINK M HANOUN N CASTEILLA L RENARD P LESIEUR D GUARDIOLALEMAITRE B AMBID L
Citation: S. Legouic et al., EFFECTS OF BOTH A MELATONIN AGONIST AND ANTAGONIST ON SEASONAL-CHANGES IN BODY-MASS AND ENERGY-INTAKE IN THE GARDEN DORMOUSE, International journal of obesity, 20(7), 1996, pp. 661-667
ENTRAINMENT OF CIRCADIAN-RHYTHMS BY S-20098, A MELATONIN AGONIST, IS DOSE AND PLASMA-CONCENTRATION DEPENDENT
Authors: MARTINET L GUARDIOLALEMAITRE B MOCAER E
Citation: L. Martinet et al., ENTRAINMENT OF CIRCADIAN-RHYTHMS BY S-20098, A MELATONIN AGONIST, IS DOSE AND PLASMA-CONCENTRATION DEPENDENT, Pharmacology, biochemistry and behavior, 54(4), 1996, pp. 713-718
PRECLINICAL PROFILE OF THE MIXED 5-HT1A 5-HT2A RECEPTOR ANTAGONIST S21357/
Authors: GRIEBEL G BLANCHARD DC RETTORI MC GUARDIOLALEMAITRE B BLANCHARD RJ
Citation: G. Griebel et al., PRECLINICAL PROFILE OF THE MIXED 5-HT1A 5-HT2A RECEPTOR ANTAGONIST S21357/, Pharmacology, biochemistry and behavior, 54(2), 1996, pp. 509-516
EFFECT OF S-21663 (PMS812), AN IMIDAZOLINE DERIVATIVE, ON GLUCOSE-TOLERANCE AND INSULIN-SECRETION IN A RAT MODEL OF TYPE-II DIABETES
Authors: WANG XA RONDU F LAMOURI A DOKHAN R MARC S TOUBOUL E PFEIFFER B MANECHEZ D RENARD P GUARDIOLALEMAITRE B GODFROID JJ KTORZA A PENICAUD L
Citation: Xa. Wang et al., EFFECT OF S-21663 (PMS812), AN IMIDAZOLINE DERIVATIVE, ON GLUCOSE-TOLERANCE AND INSULIN-SECRETION IN A RAT MODEL OF TYPE-II DIABETES, The Journal of pharmacology and experimental therapeutics, 278(1), 1996, pp. 82-89
3-AMINO-3,4-DIHYDRO-2H-1-BENZOPYRAN DERIVATIVES AS 5-HT1A RECEPTOR LIGANDS AND POTENTIAL ANXIOLYTIC AGENTS .2. SYNTHESIS AND QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF SPIRO[PYRROLIDINE-2,3'(2'H)-BENZOPYRAN] AND SPIRO[PIPERIDINE-2,3'(2'H)-BENZOPYRAN]
Authors: COMOY C MAROT C PODONA T BAUDIN ML MORINALLORY L GUILLAUMET G PFEIFFER B CAIGNARD DH RENARD P RETTORI MC ADAM G GUARDIOLALEMAITRE B
Citation: C. Comoy et al., 3-AMINO-3,4-DIHYDRO-2H-1-BENZOPYRAN DERIVATIVES AS 5-HT1A RECEPTOR LIGANDS AND POTENTIAL ANXIOLYTIC AGENTS .2. SYNTHESIS AND QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF SPIRO[PYRROLIDINE-2,3'(2'H)-BENZOPYRAN] AND SPIRO[PIPERIDINE-2,3'(2'H)-BENZOPYRAN], Journal of medicinal chemistry, 39(21), 1996, pp. 4285-4298
NOVEL SELECTIVE AND PARTIAL AGONISTS OF 5-HT3 RECEPTORS .1. SYNTHESISAND BIOLOGICAL EVALUATION OF PIPERAZINOPYRROLOTHIENOPYRAZINES
Authors: RAULT S LANCELOT JC PRUNIER H ROBBA M RENARD P DELAGRANGE P PFEIFFER B CAIGNARD DH GUARDIOLALEMAITRE B HAMON M
Citation: S. Rault et al., NOVEL SELECTIVE AND PARTIAL AGONISTS OF 5-HT3 RECEPTORS .1. SYNTHESISAND BIOLOGICAL EVALUATION OF PIPERAZINOPYRROLOTHIENOPYRAZINES, Journal of medicinal chemistry, 39(10), 1996, pp. 2068-2080
MELATONIN ANALOGS AS AGONISTS AND ANTAGONISTS IN THE CIRCADIAN SYSTEMAND OTHER BRAIN-AREAS
Authors: YING SW RUSAK B DELAGRANGE P MOCAER E RENARD P GUARDIOLALEMAITRE B
Citation: Sw. Ying et al., MELATONIN ANALOGS AS AGONISTS AND ANTAGONISTS IN THE CIRCADIAN SYSTEMAND OTHER BRAIN-AREAS, European journal of pharmacology, 296(1), 1996, pp. 33-42
DOSE-DEPENDENT EFFECTS OF S-20098, A MELATONIN AGONIST, ON DIRECTION OF REENTRAINMENT OF RAT CIRCADIAN ACTIVITY RHYTHMS
Authors: REDMAN JR GUARDIOLALEMAITRE B BROWN M DELAGRANGE P ARMSTRONG SM
Citation: Jr. Redman et al., DOSE-DEPENDENT EFFECTS OF S-20098, A MELATONIN AGONIST, ON DIRECTION OF REENTRAINMENT OF RAT CIRCADIAN ACTIVITY RHYTHMS, Psychopharmacology, 118(4), 1995, pp. 385-390
STRUCTURE-ACTIVITY-RELATIONSHIPS OF MELATONIN ANALOGS
Authors: CAIGNARD DH LESIEUR D DEPREUX P RENARD P DELAGRANGE P GUARDIOLALEMAITRE B
Citation: Dh. Caignard et al., STRUCTURE-ACTIVITY-RELATIONSHIPS OF MELATONIN ANALOGS, European journal of medicinal chemistry, 30, 1995, pp. 637-642
MELATONIN ANALOGS - FROM PHARMACOLOGY TO CLINICAL-APPLICATION
Authors: GUARDIOLALEMAITRE B DELAGRANGE P
Citation: B. Guardiolalemaitre et P. Delagrange, MELATONIN ANALOGS - FROM PHARMACOLOGY TO CLINICAL-APPLICATION, European journal of medicinal chemistry, 30, 1995, pp. 643-651
ANTICONFLICT AND DISCRIMINATIVE STIMULUS EFFECTS IN THE PIGEON OF A NEW METHOXY-CHROMAN 5-HT1A AGONIST, (-20244 AND ITS ENANTIOMERS (+)S-20499 AND (-)S-20500()S)
Authors: BARRETT JE GAMBLE EH ZHANG L GUARDIOLALEMAITRE B
Citation: Je. Barrett et al., ANTICONFLICT AND DISCRIMINATIVE STIMULUS EFFECTS IN THE PIGEON OF A NEW METHOXY-CHROMAN 5-HT1A AGONIST, (-20244 AND ITS ENANTIOMERS (+)S-20499 AND (-)S-20500()S), Psychopharmacology, 116(1), 1994, pp. 73-78
3,4-DIHYDRO-3-AMINO-2H-1-BENZOPYRAN DERIVATIVES AS 5-HT1A RECEPTOR LIGANDS AND POTENTIAL ANXIOLYTIC AGENTS .1. SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIP STUDIES
Authors: PODONA T GUARDIOLALEMAITRE B CAIGNARD DH ADAM G PFEIFFER B RENARD P GUILLAUMET G
Citation: T. Podona et al., 3,4-DIHYDRO-3-AMINO-2H-1-BENZOPYRAN DERIVATIVES AS 5-HT1A RECEPTOR LIGANDS AND POTENTIAL ANXIOLYTIC AGENTS .1. SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIP STUDIES, Journal of medicinal chemistry, 37(12), 1994, pp. 1779-1793
EFFECTS OF A NOVEL MELATONIN ANALOG ON CIRCADIAN-RHYTHMS OF BODY-TEMPERATURE AND ACTIVITY IN YOUNG, MIDDLE-AGED, AND OLD RATS
Authors: KOSTERVANHOFFEN GC MIRMIRAN M BOS NPA WITTING W DELAGRANGE P GUARDIOLALEMAITRE B
Citation: Gc. Kostervanhoffen et al., EFFECTS OF A NOVEL MELATONIN ANALOG ON CIRCADIAN-RHYTHMS OF BODY-TEMPERATURE AND ACTIVITY IN YOUNG, MIDDLE-AGED, AND OLD RATS, Neurobiology of aging, 14(6), 1993, pp. 565-569
SUCCESSFUL USE OF S20098 AND MELATONIN IN AN ANIMAL-MODEL OF DELAYED SLEEP-PHASE SYNDROME (DSPS)
Authors: ARMSTRONG SM MCNULTY OM GUARDIOLALEMAITRE B REDMAN JR
Citation: Sm. Armstrong et al., SUCCESSFUL USE OF S20098 AND MELATONIN IN AN ANIMAL-MODEL OF DELAYED SLEEP-PHASE SYNDROME (DSPS), Pharmacology, biochemistry and behavior, 46(1), 1993, pp. 45-49
(-)TERTATOLOL IS A POTENT ANTAGONIST AT PRESYNAPTIC AND POSTSYNAPTIC SEROTONIN 5-HT(1A) RECEPTORS IN THE RAT-BRAIN
Authors: JOLAS T HAJDAHMANE S LANFUMEY L FATTACCINI CM KIDD EJ ADRIEN J GOZLAN H GUARDIOLALEMAITRE B HAMON M
Citation: T. Jolas et al., (-)TERTATOLOL IS A POTENT ANTAGONIST AT PRESYNAPTIC AND POSTSYNAPTIC SEROTONIN 5-HT(1A) RECEPTORS IN THE RAT-BRAIN, Naunyn-Schmiedeberg's archives of pharmacology, 347(5), 1993, pp. 453-463
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